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Histamine H4 receptor ligands and their potential therapeutic applications

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Pages 119-135 | Published online: 05 Feb 2009

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Róbert Kiss & György M Keserű. (2012) Histamine H4 receptor ligands and their potential therapeutic applications: an update. Expert Opinion on Therapeutic Patents 22:3, pages 205-221.
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Xiaojing Ling, Yongxin Liu, Danxuan Zhu, Weizhen An, Jiaying Geng, Lin Li, Changmin Yu & Ji-Fu Wei. (2022) Colorimetric visualization of histamine secreted by basophils based on DSP-functionalized gold nanoparticles. Analytical Methods 14:27, pages 2698-2702.
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Fernando Valenzuela & Rodrigo Flores. (2021) Antihistamínicos: Usos clásicos, nuevos y anecdóticos en dermatología. Parte 1: Histamina, sus receptores y antagonistas. Piel 36:2, pages 95-103.
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Ruben Vardanyan & Victor Hruby. 2016. Synthesis of Best-Seller Drugs. Synthesis of Best-Seller Drugs 247 263 .
Mark S. Tichenor, Robin L. Thurmond, Jennifer D. Venable & Brad M. Savall. (2015) Functional Profiling of 2-Aminopyrimidine Histamine H 4 Receptor Modulators . Journal of Medicinal Chemistry 58:18, pages 7119-7127.
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Roland Geyer, Melanie Kaske, Paul Baumeister & Armin Buschauer. (2014) Synthesis and Functional Characterization of Imbutamine Analogs as Histamine H 3 and H 4 Receptor Ligands . Archiv der Pharmazie 347:2, pages 77-88.
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Roland Geyer, Patrick Igel, Melanie Kaske, Sigurd Elz & Armin Buschauer. (2014) Synthesis, SAR and selectivity of 2-acyl- and 2-cyano-1-hetarylalkyl-guanidines at the four histamine receptor subtypes: a bioisosteric approach. Med. Chem. Commun. 5:1, pages 72-81.
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Charlotte A.L. Lane, Duncan Hay, Charles E. Mowbray, Michael Paradowski, Matthew D. Selby, Nigel A. Swain & David H. Williams. (2012) Synthesis of novel histamine H4 receptor antagonists. Bioorganic & Medicinal Chemistry Letters 22:2, pages 1156-1159.
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Roland Geyer & Armin Buschauer. (2011) Synthesis and Histamine H 3 and H 4 Receptor Activity of Conformationally Restricted Cyanoguanidines Related to UR‐PI376 . Archiv der Pharmazie 344:12, pages 775-785.
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Charles M. Marson. (2011) Targeting the Histamine H 4 Receptor . Chemical Reviews 111:11, pages 7121-7156.
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Robert L. Hudkins, Rita Raddatz, Ming Tao, Joanne R. Mathiasen, Lisa D. Aimone, Nadine C. Becknell, Catherine P. Prouty, Lars J. S. Knutsen, Mehran Yazdanian, Gilbert Moachon, Mark A. Ator, John P. Mallamo, Michael J. Marino, Edward R. Bacon & Michael Williams. (2011) Discovery and Characterization of 6-{4-[3-( R )-2-Methylpyrrolidin-1-yl)propoxy]phenyl}-2 H -pyridazin-3-one (CEP-26401, Irdabisant): A Potent, Selective Histamine H 3 Receptor Inverse Agonist . Journal of Medicinal Chemistry 54:13, pages 4781-4792.
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Mark B. Abelson, James T. McLaughlin & Paul J. Gomes. (2011) Antihistamines in Ocular Allergy: Are They All Created Equal?. Current Allergy and Asthma Reports 11:3, pages 205-211.
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Phil Lieberman. (2011) The basics of histamine biology. Annals of Allergy, Asthma & Immunology 106:2, pages S2-S5.
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Róbert Kiss & György M. Keserű. 2011. Virtual Screening. Virtual Screening 381 410 .
Farhad Jadidi-Niaragh & Abbas Mirshafiey. (2010) Histamine and histamine receptors in pathogenesis and treatment of multiple sclerosis. Neuropharmacology 59:3, pages 180-189.
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Sue Cramp, Hazel J. Dyke, Christopher Higgs, David E. Clark, Matthew Gill, Pascal Savy, Neil Jennings, Steve Price, Peter M. Lockey, Dennis Norman, Soraya Porres, Francis Wilson, Alison Jones, Nigel Ramsden, Raffaella Mangano, Dan Leggate, Marie Andersson & Richard Hale. (2010) Identification and hit-to-lead exploration of a novel series of histamine H4 receptor inverse agonists. Bioorganic & Medicinal Chemistry Letters 20:8, pages 2516-2519.
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Fakher Rahim. (2010) An in Silico Development of Selective Inhibitor for Histamine Receptors. Biotechnology(Faisalabad) 9:2, pages 157-163.
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K. Sander, T. Kottke, E. Proschak, Y. Tanrikulu, E. H. Schneider, R. Seifert, G. Schneider & H. Stark. (2009) Lead identification and optimization of diaminopyrimidines as histamine H4 receptor ligands. Inflammation Research 59:S2, pages 249-251.
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Kerstin Sander, Tim Kottke, Yusuf Tanrikulu, Ewgenij Proschak, Lilia Weizel, Erich H. Schneider, Roland Seifert, Gisbert Schneider & Holger Stark. (2009) 2,4-Diaminopyrimidines as histamine H4 receptor ligands—Scaffold optimization and pharmacological characterization. Bioorganic & Medicinal Chemistry 17:20, pages 7186-7196.
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