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Recent advances in the development of selective androgen receptor modulators

, PhD, , PhD & , PhD
Pages 1239-1258 | Published online: 08 Jun 2009

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Tommi H Nyrönen & Annu A Söderholm. (2010) Structural basis for computational screening of non-steroidal androgen receptor ligands. Expert Opinion on Drug Discovery 5:1, pages 5-20.
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Marina Komrakova, Janek Nagel, Daniel Bernd Hoffmann, Wolfgang Lehmann, Arndt Friedrich Schilling & Stephan Sehmisch. (2020) Effect of Selective Androgen Receptor Modulator Enobosarm on Bone Healing in a Rat Model for Aged Male Osteoporosis. Calcified Tissue International 107:6, pages 593-602.
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Vito A. Giagulli, Andrea Silvestrini, Carmine Bruno, Vincenzo Triggiani, Alvaro Mordente & Antonio Mancini. (2020) Is There Room for SERMs or SARMs as Alternative Therapies for Adult Male Hypogonadism?. International Journal of Endocrinology 2020, pages 1-9.
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D. B. Hoffmann, M. Komrakova, S. Pflug, M. von Oertzen, D. Saul, L. Weiser, T. A. Walde, M. Wassmann, A. F. Schilling, W. Lehmann & S. Sehmisch. (2018) Evaluation of ostarine as a selective androgen receptor modulator in a rat model of postmenopausal osteoporosis. Journal of Bone and Mineral Metabolism 37:2, pages 243-255.
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Päivi Pihlajamaa, Biswajyoti Sahu & Olli A. Jänne. (2015) Determinants of Receptor- and Tissue-Specific Actions in Androgen Signaling. Endocrine Reviews 36:4, pages 357-384.
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G. G. Mazgarova, K. Yu. Suponitskii & R. R. Gataullin. (2013) Effect of salts on the reaction direction of (2R*,3R*)-2-[(1R*)-1-iodoethyl)]-3-methyl(3,5-dimethyl)-1-(4-methylphenylsulfonyl)-2,3-dihydro-1H-indoles with dimethylformamide. Russian Journal of Organic Chemistry 49:9, pages 1322-1328.
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