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Expert Opinion on Therapeutic Patents Volume 11, 2001 - Issue 8
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Small molecule antagonists of chemokine receptors as emerging anti-HIV agents

Antonio Mastrolorenzo Università degli Studi, Dipartimento di Scienze Dermatologiche, Centro MTS, via degli Alfani 37, 50121 Firenze, Italy. , Fax: +39 055 2758395; E-mail: [email protected]à degli Studi, Laboratorio di Chimica Inorganica e Bioinorganica, via Gino Capponi 7, I-50121, Florence, Italy. , Fax: +39 055 2757555; , E-mail: [email protected]
,
Andrea Scozzafava Università degli Studi, Dipartimento di Scienze Dermatologiche, Centro MTS, via degli Alfani 37, 50121 Firenze, Italy. , Fax: +39 055 2758395; E-mail: [email protected]à degli Studi, Laboratorio di Chimica Inorganica e Bioinorganica, via Gino Capponi 7, I-50121, Florence, Italy. , Fax: +39 055 2757555; , E-mail: [email protected]
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Claudiu T Supuran Università degli Studi, Laboratorio di Chimica Inorganica e Bioinorganica, via Gino Capponi 7, I-50121, Florence, Italy. , Fax: +39 055 2757555; , E-mail: [email protected]
Pages 1245-1252 | Published online: 25 Feb 2005

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Claudiu T Supuran. (2011) Therapeutic compounds: patent evaluation of WO2011011652A1. Expert Opinion on Therapeutic Patents 21:9, pages 1491-1495.
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Hirokazu Tamamura, Hiroshi Tsutsumi, Wataru Nomura, Tomohiro Tanaka & Nobutaka Fujii. (2008) A future perspective on the development of chemokine receptor CXCR4 antagonists. Expert Opinion on Drug Discovery 3:10, pages 1155-1166.
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Hirokazu Tamamura & Nobutaka Fujii. (2005) The therapeutic potential of CXCR4 antagonists in the treatment of HIV infection, cancer metastasis and rheumatoid arthritis. Expert Opinion on Therapeutic Targets 9:6, pages 1267-1282.
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Jean-Yves Winum, Andrea Scozzafava, Jean-Louis Montero & Claudiu T Supuran. (2004) Therapeutic applications of sulfamates. Expert Opinion on Therapeutic Patents 14:9, pages 1273-1308.
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. (2004) 4,4-Disubstituted-3,4-dihydro-2(1H)-quinazolinones as HIV reverse transcriptase inhibitors. Expert Opinion on Therapeutic Patents 14:8, pages 1237-1240.
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. (2004) Chemokine receptor antagonists as HIV entry inhibitors. Expert Opinion on Therapeutic Patents 14:2, pages 251-255.
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Akira Naya & Toshihiko Saeki. (2004) Chemokine CCR3 antagonists. Expert Opinion on Therapeutic Patents 14:1, pages 7-16.
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. (2003) HIV protease inhibitors based on amino acid derivatives. Expert Opinion on Therapeutic Patents 13:4, pages 547-550.
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Articles from other publishers (11)

David C. Pryde & Christopher G. Barber. 2010. Chemokine Receptors as Drug Targets. Chemokine Receptors as Drug Targets 207 238 .
Chris Barber & David Pryde. 2010. Accounts in Drug Discovery. Accounts in Drug Discovery 183 214 .
Antonio MastrolorenzoAlfonso MarescaStefano RusconiClaudiu T Supuran. (2008) Update on the development of HIV entry inhibitors. Future HIV Therapy 2:5, pages 479-507.
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Hirokazu TamamuraHiroshi TsutsumiWataru NomuraNobutaka Fujii. (2008) Exploratory Studies on Development of the Chemokine Receptor CXCR4 Antagonists toward Downsizing. Perspectives in Medicinal Chemistry 2, pages PMC.S422.
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Hiroshi Tsutsumi, Tomohiro Tanaka, Nami Ohashi, Hiroyuki Masuno, Hirokazu Tamamura, Kenichi Hiramatsu, Takanobu Araki, Satoshi Ueda, Shinya Oishi & Nobutaka Fujii. (2007) Therapeutic potential of the chemokine receptor CXCR4 antagonists as multifunctional agents. Biopolymers 88:2, pages 279-289.
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Jean‐Yves Winum, Andrea Scozzafava, Jean‐Louis Montero & Claudiu T. Supuran. (2004) Sulfamates and their therapeutic potential. Medicinal Research Reviews 25:2, pages 186-228.
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Dong-Ming Shen, Min Shu, Sander G. Mills, Kevin T. Chapman, Lorraine Malkowitz, Martin S. Springer, Sandra L. Gould, Julie A. DeMartino, Salvatore J. Siciliano, Gloria Y. Kwei, Anthony Carella, Gwen Carver, Karen Holmes, William A. Schleif, Renee Danzeisen, Daria Hazuda, Joseph Kessler, Janet Lineberger, Michael D. Miller & Emilio A. Emini. (2004) Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 1: Discovery and SAR study of 4-pyrazolylpiperidine side chains. Bioorganic & Medicinal Chemistry Letters 14:4, pages 935-939.
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Anandan Palani, Sherry Shapiro, John W. Clader, William J. Greenlee, Susan Vice, Stuart McCombie, Kathleen Cox, Julie Strizki & Bahige M. Baroudy. (2003) Oximino-piperidino-piperidine-based CCR5 antagonists. Part 2: synthesis, SAR and biological evaluation of symmetrical heteroaryl carboxamides. Bioorganic & Medicinal Chemistry Letters 13:4, pages 709-712.
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Anandan Palani, Sherry Shapiro, John W. Clader, William J. Greenlee, David Blythin, Kathleen Cox, Nicole E. Wagner, Julie Strizki, Bahige M. Baroudy & Niya Dan. (2003) Biological evaluation and interconversion studies of rotamers of SCH 351125, an orally bioavailable CCR5 antagonist. Bioorganic & Medicinal Chemistry Letters 13:4, pages 705-708.
Crossref
John A. Bender, Nicholas A. Meanwell & Tao Wang. (2002) The mono-functionalization of symmetrical polyamines. Tetrahedron 58:16, pages 3111-3128.
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Nicholas A Meanwell, John F Kadow & Paul M Scola. 2002. Annual Reports in Medicinal Chemistry Volume 37. Annual Reports in Medicinal Chemistry Volume 37 133 147 .

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