Citations (12)
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Chen Cheng, Salman Jabri, Brandon M Taoka & Christopher J Sinz. (2020) Small molecule glucagon receptor antagonists: an updated patent review (2015–2019). Expert Opinion on Therapeutic Patents 30:7, pages 509-526.
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Kevin J Filipski. (2015) Small molecule glucagon receptor antagonists: a patent review (2011 – 2014). Expert Opinion on Therapeutic Patents 25:7, pages 819-830.
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Dong-Ming Shen, Songnian Lin & Emma R Parmee. (2011) A survey of small molecule glucagon receptor antagonists from recent patents (2006 – 2010). Expert Opinion on Therapeutic Patents 21:8, pages 1211-1240.
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Ravi Kurukulasuriya & JT Link. (2005) Progress towards glucagon receptor antagonist therapy for Type 2 diabetes. Expert Opinion on Therapeutic Patents 15:12, pages 1739-1749.
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Shuangjie Shu, Xiaoqing Cai, Jia Li, Yang Feng, Antao Dai, Jiang Wang, Dehua Yang, Ming-Wei Wang & Hong Liu. (2016) Design, synthesis, structure–activity relationships, and docking studies of pyrazole-containing derivatives as a novel series of potent glucagon receptor antagonists. Bioorganic & Medicinal Chemistry 24:12, pages 2852-2863.
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The Discovery of
N
-((2
H
-Tetrazol-5-yl)methyl)-4-((
R
)-1-((5
r
,8
R
)-8-(
tert
-butyl)-3-(3,5-dichlorophenyl)-2-oxo-1,4-diazaspiro[4.5]dec-3-en-1-yl)-4,4-dimethylpentyl)benzamide (SCH 900822): A Potent and Selective Glucagon Receptor Antagonist
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Ronald M. Kim, Jiang Chang, Ashley R. Lins, Ed Brady, Mari R. Candelore, Qing Dallas-Yang, Victor Ding, Jasminka Dragovic, Susan Iliff, Guoqiang Jiang, Steven Mock, Sajjad Qureshi, Richard Saperstein, Deborah Szalkowski, Constantin Tamvakopoulos, Laurie Tota, Michael Wright, Xiaodong Yang, James R. Tata, Kevin Chapman, Bei B. Zhang & Emma R. Parmee. (2008) Discovery of potent, orally active benzimidazole glucagon receptor antagonists. Bioorganic & Medicinal Chemistry Letters 18:13, pages 3701-3705.
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Rui Liang, Lauren Abrardo, Edward J. Brady, Mari Rios Candelore, Victor Ding, Richard Saperstein, Laurie M. Tota, Michael Wright, Steve Mock, Constantin Tamvakopolous, Sharon Tong, Song Zheng, Bei B. Zhang, James R. Tata & Emma R. Parmee. (2007) Design and synthesis of conformationally constrained tri-substituted ureas as potent antagonists of the human glucagon receptor. Bioorganic & Medicinal Chemistry Letters 17:3, pages 587-592.
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Sheila M. Cohen, Joseph L. Duffy, Corin Miller, Brian A. Kirk, Mari Rios Candelore, Victor D.H. Ding, Gregory Kaczorowski, Laurie M. Tota, Jeffrey G. Werrmann, Michael Wright, Emma R. Parmee, James R. Tata & Bei B. Zhang. (2006) Direct observation (NMR) of the efficacy of glucagon receptor antagonists in murine liver expressing the human glucagon receptor. Bioorganic & Medicinal Chemistry 14:5, pages 1506-1517.
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Dong-Ming Shen, Fengqi Zhang, Edward J. Brady, Mari Rios Candelore, Qing Dallas-Yang, Victor D.-H. Ding, Jasminka Dragovic, William P. Feeney, Guoquiang Jiang, Peggy E. McCann, Steve Mock, Sajjad A. Qureshi, Richard Saperstein, Xiaolan Shen, Constantin Tamvakopoulos, Xinchun Tong, Laurie M. Tota, Michael J. Wright, Xiaodong Yang, Song Zheng, Kevin T. Chapman, Bei B. Zhang, James R. Tata & Emma R. Parmee. (2005) Discovery of novel, potent, and orally active spiro-urea human glucagon receptor antagonists. Bioorganic & Medicinal Chemistry Letters 15:20, pages 4564-4569.
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Ravi Kurukulasuriya, Bryan K Sorensen, James T Link, Jyoti R Patel, Hwan-Soo Jae, Marty X Winn, Jeffrey R Rohde, Nelson D Grihalde, Chun W Lin, Christopher A Ogiela, Andrew L Adler & Christine A Collins. (2004) Biaryl amide glucagon receptor antagonists. Bioorganic & Medicinal Chemistry Letters 14:9, pages 2047-2050.
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