Advanced search
Publication Cover
Expert Opinion on Therapeutic Patents Volume 13, 2003 - Issue 12
Submit an article Journal homepage
25
Views
11
CrossRef citations to date
0
Altmetric
Review

Non-steroidal progesterone receptor modulators

Puwen Zhang Chemical & Screening Sciences & Women’s Health Research Institute, Wyeth Research, 500 Arcola Road, Collegeville, PA19426, USA. [email protected]
,
Andrew Fensome Chemical & Screening Sciences & Women’s Health Research Institute, Wyeth Research, 500 Arcola Road, Collegeville, PA19426, USA. [email protected]
,
Jay Wrobel Chemical & Screening Sciences & Women’s Health Research Institute, Wyeth Research, 500 Arcola Road, Collegeville, PA19426, USA. [email protected]
,
Richard Winneker Chemical & Screening Sciences & Women’s Health Research Institute, Wyeth Research, 500 Arcola Road, Collegeville, PA19426, USA. [email protected]
&
Zhiming Zhang Chemical & Screening Sciences & Women’s Health Research Institute, Wyeth Research, 500 Arcola Road, Collegeville, PA19426, USA. [email protected]
Pages 1839-1847 | Published online: 02 Mar 2005

Citations (11)

Keep up to date with the latest research on this topic with citation updates for this article.

Subscribe to citation updates

Read on this site (1)

Weiqin Jiang, James J. Fiordeliso & Zhihua Sui. (2007) Facile Synthesis of 3,3‐Dialkyl‐6‐phenyl‐imidazopyridinones. Synthetic Communications 37:8, pages 1237-1249.
Read now

Articles from other publishers (10)

Santosh R. Kshirsagar, Ashok S. Pise, Sagar I. Shinde, Sandip P. Gondake & Valmik S. Kapase. (2020) One-Pot Green Method for the Synthesis of Oxazine Derivatives Under Aqueous Medium. International Journal of Scientific Research in Science and Technology, pages 332-339.
Crossref
Deborah M. Roll, Laurel R. Barbieri, Ramunas Bigelis, Leonard A. McDonald, Daniel A. Arias, Li-Ping Chang, Maya P. Singh, Scott W. Luckman, Thomas J. Berrodin & Matthew R. Yudt. (2009) The Lecanindoles, Nonsteroidal Progestins from the Terrestrial Fungus Verticillium lecanii 6144 . Journal of Natural Products 72:11, pages 1944-1948.
Crossref
Nareshkumar Jain, George Allan, Olivia Linton, Pamela Tannenbaum, Xin Chen, Jun Xu, Peifang Zhu, Joseph Gunnet, Keith Demarest, Scott Lundeen, William Murray & Zhihua Sui. (2009) Synthesis and SAR study of novel pseudo-steroids as potent and selective progesterone receptor antagonists. Bioorganic & Medicinal Chemistry Letters 19:14, pages 3977-3980.
Crossref
Andrew Fensome, William R. Adams, Andrea L. Adams, Tom J. Berrodin, Jeff Cohen, Christine Huselton, Arthur Illenberger, Jeffrey C. Kern, Valerie A. Hudak, Michael A. Marella, Edward G. Melenski, Casey C. McComas, Cheryl A. Mugford, Ov D. Slayden, Matthew Yudt, Zhiming Zhang, Puwen Zhang, Yuan Zhu, Richard C. Winneker & Jay E. Wrobel. (2008) Design, Synthesis, and SAR of New Pyrrole-Oxindole Progesterone Receptor Modulators Leading to 5-(7-Fluoro-3,3-dimethyl-2-oxo-2,3-dihydro-1 H -indol-5-yl)-1-methyl-1 H -pyrrole-2-carbonitrile (WAY-255348) . Journal of Medicinal Chemistry 51:6, pages 1861-1873.
Crossref
Paul P.M.A. Dols, Brigitte J.B. Folmer, Hans Hamersma, Cor W. Kuil, Hans Lucas, Lourdes Ollero, Jos B.M. Rewinkel & Pedro H.H. Hermkens. (2008) SAR study of 2,3,4,14b-tetrahydro-1H-dibenzo[b,f]pyrido[1,2-d][1,4]oxazepines as progesterone receptor agonists. Bioorganic & Medicinal Chemistry Letters 18:4, pages 1461-1467.
Crossref
Puwen Zhang, Eugene Terefenko, Jeffrey Kern, Andrew Fensome, Eugene Trybulski, Ray Unwalla, Jay Wrobel, Susan Lockhead, Yuan Zhu, Jeffrey Cohen, Margaret LaCava, Richard C. Winneker & Zhiming Zhang. (2007) 5-(3-Cyclopentyl-2-thioxo-2,3-dihydro-1H-benzimidazol-5-yl)-1-methyl-1H-pyrrole-2-carbonitrile: A novel, highly potent, selective, and orally active non-steroidal progesterone receptor agonist. Bioorganic & Medicinal Chemistry 15:20, pages 6556-6564.
Crossref
Fu-An Kang, Jihua Guan, Nareshkumar Jain, George Allan, Olivia Linton, Pamela Tannenbaum, Xin Chen, Jun Xu, Peifang Zhu, Joseph Gunnet, Keith Demarest, Scott Lundeen & Zhihua Sui. (2007) Parallel synthesis and SAR study of novel oxa-steroids as potent and selective progesterone receptor antagonists. Bioorganic & Medicinal Chemistry Letters 17:9, pages 2531-2534.
Crossref
Kevin P. Madauss, Eugene L. Stewart & Shawn P. Williams. (2006) The evolution of progesterone receptor ligands. Medicinal Research Reviews 27:3, pages 374-400.
Crossref
Fu-An Kang, George Allan, Jihua Guan, Nareshkumar Jain, Olivia Linton, Pamela Tannenbaum, Jun Xu, Peifang Zhu, Joseph Gunnet, Xin Chen, Keith Demarest, Scott Lundeen & Zhihua Sui. (2007) Synthesis and identification of novel oxa-steroids as progesterone receptor antagonists. Bioorganic & Medicinal Chemistry Letters 17:4, pages 907-910.
Crossref
Weiqin Jiang, James J. Fiordeliso, Xin Chen & Zhihua Sui. (2006) Synthesis of trisubstituted thiophenes designed as progesterone receptor modulator. Journal of Heterocyclic Chemistry 43:5, pages 1391-1396.
Crossref

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Order Reprints Request Corporate Permissions

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

Request Academic Permissions

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.

Related research

People also read lists articles that other readers of this article have read.

Recommended articles lists articles that we recommend and is powered by our AI driven recommendation engine.

Cited by lists all citing articles based on Crossref citations.
Articles with the Crossref icon will open in a new tab.