Citations (34)
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Miguel A. Maestro, Ferdinand Molnár, Antonio Mouriño & Carsten Carlberg. (2016) Vitamin D receptor 2016: novel ligands and structural insights. Expert Opinion on Therapeutic Patents 26:11, pages 1291-1306.
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Ichiro Takada & Makoto Makishima. (2015) Therapeutic application of vitamin D receptor ligands: an updated patent review. Expert Opinion on Therapeutic Patents 25:12, pages 1373-1383.
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Carsten Carlberg, Ferdinand Molnár & Antonio Mouriño. (2012) Vitamin D receptor ligands: the impact of crystal structures. Expert Opinion on Therapeutic Patents 22:4, pages 417-435.
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Mihwa Choi & Makoto Makishima. (2009) Therapeutic applications for novel non-hypercalcemic vitamin D receptor ligands. Expert Opinion on Therapeutic Patents 19:5, pages 593-606.
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Articles from other publishers (30)
Miguel A. Maestro, Ferdinand Molnár & Carsten Carlberg. (2019) Vitamin D and Its Synthetic Analogs. Journal of Medicinal Chemistry 62:15, pages 6854-6875.
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Akiko Nagata, Yusuke Akagi, Shadi Sedghi Masoud, Masahiro Yamanaka, Atsushi Kittaka, Motonari Uesugi, Minami Odagi & Kazuo Nagasawa. (2019) Stereoselective Synthesis of Four Calcitriol Lactone Diastereomers at C23 and C25. The Journal of Organic Chemistry 84:12, pages 7630-7641.
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Wei Wang, Guo-Dong Zhao, Ying-jie Cui, Min-Qi Li & Zhao-Peng Liu. (2019) Synthesis of 1α,25-dihydroxyvitamin D3 analogues with α,α-difluorocycloketone at the CD-ring side chains and their biological properties in ovariectomized rats. The Journal of Steroid Biochemistry and Molecular Biology 186, pages 66-73.
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Marcin Szybinski, Katarzyna Sektas, Rafal R. Sicinski, Lori A. Plum, Jadwiga Frelek & Hector F. DeLuca. (2017) Design, synthesis and biological properties of seco-d-ring modified 1α,25-dihydroxyvitamin D3 analogues. The Journal of Steroid Biochemistry and Molecular Biology 171, pages 144-154.
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Urszula Kulesza, Lori A. Plum, Hector F. DeLuca, Antonio Mouriño & Rafal R. Sicinski. (2015)
Novel 9-Alkyl- and 9-Alkylidene-Substituted 1α,25-Dihydroxyvitamin D
3
Analogues: Synthesis and Biological Examinations
. Journal of Medicinal Chemistry 58:15, pages 6237-6247.
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Norihito Arichi, Kenji Hata, Yoshiji Takemoto, Ken-ichi Yamada, Yousuke Yamaoka & Kiyosei Takasu. (2015) Synthesis of steroidal derivatives bearing a small ring using a catalytic [2+2] cycloaddition and a ring-contraction rearrangement. Tetrahedron 71:2, pages 233-244.
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Diego M. Carballa, Flavia Zacconi, Urszula Kulesza, Antonio Mouriño & Mercedes Torneiro. (2013) Synthesis of 1α,25-dihydroxyvitamin D3 analogues with α-hydroxyalkyl substituents at C12. The Journal of Steroid Biochemistry and Molecular Biology 136, pages 34-38.
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Diego M. Carballa, Samuel Seoane, Flavia Zacconi, Xenxo Pérez, Antonio Rumbo, Silvia Alvarez-Díaz, María Jesús Larriba, Román Pérez-Fernández, Alberto Muñoz, Miguel MaestroAntonio Mouriño & Mercedes Torneiro. (2012)
Synthesis and Biological Evaluation of 1α,25-Dihydroxyvitamin D
3
Analogues with a Long Side Chain at C12 and Short C17 Side Chains
. Journal of Medicinal Chemistry 55:20, pages 8642-8656.
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Diego M. Carballa, Antonio Rumbo, Mercedes Torneiro, Miguel Maestro & Antonio Mouriño. (2012)
Synthesis of (1
α
)‐1,25‐Dihydroxyvitamin D
3
with a
β
‐Positioned Seven‐Carbon Side Chain at C(12)
. Helvetica Chimica Acta 95:10, pages 1842-1850.
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Hirotaka Kashiwagi, Yoshiyuki Ono, Masateru Ohta, Kenji Morikami & Tadakatsu Takahashi. (2012) Systematic SAR study of the side chain of nonsecosteroidal vitamin D3 analogs. Bioorganic & Medicinal Chemistry 20:14, pages 4495-4506.
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Ramón Fraga, Flavia Zacconi, Fredy Sussman, Paloma Ordóñez‐Morán, Alberto Muñoz, Tiphaine Huet, Ferdinand Molnár, Dino Moras, Natacha Rochel, Miguel Maestro & Antonio Mouriño. (2011) Design, Synthesis, Evaluation, and Structure of Vitamin D Analogues with Furan Side Chains. Chemistry – A European Journal 18:2, pages 603-612.
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María A. Regueira, Shaonly Samanta, Peter J. Malloy, Paloma Ordóñez-Morán, Diana Resende, Fredy Sussman, Alberto Muñoz, Antonio Mouriño, David Feldman & Mercedes Torneiro. (2011)
Synthesis and Biological Evaluation of 1α,25-Dihydroxyvitamin D
3
Analogues Hydroxymethylated at C-26
. Journal of Medicinal Chemistry 54:11, pages 3950-3962.
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Yan Chen & Tong Ju. (2010)
Enantioselective Synthesis of A Key A-Ring Intermediate for the Preparation of 1α,25-Dihydroxyvitamin D
3
. Organic Letters 13:1, pages 86-89.
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Marjo Malinen, Jussi Ryynänen, Merja Heinäniemi, Sami Väisänen & Carsten Carlberg. (2011) Cyclical regulation of the insulin-like growth factor binding protein 3 gene in response to 1α,25-dihydroxyvitamin D 3. Nucleic Acids Research 39:2, pages 502-512.
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Jinhu Wang, Ke Tang, Qianqian Hou, Xueli Cheng, Lihua Dong, Yongjun Liu & Chengbu Liu. (2010) 3D-QSAR Studies on C24-Monoalkylated Vitamin D3 26,23-Lactones and their C2α-Modified Derivatives with Inhibitory Activity to Vitamin D Receptor. Molecular Informatics 29:8-9, pages 621-632.
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Antonio Rumbo, Xenxo Pérez-García & Antonio Mouriño. (2010) Stereoselective synthesis of C24-hydroxylated vitamin D3 analogs: A practical and expeditius route to calcipotriol. The Journal of Steroid Biochemistry and Molecular Biology 121:1-2, pages 68-70.
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Daniel Nicoletti, Carlos Gregorio, Antonio Mouriño & Miguel Maestro. (2010) A short practical approach to 24R,25-dihydroxyvitamin D3. The Journal of Steroid Biochemistry and Molecular Biology 121:1-2, pages 43-45.
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Silvina Eduardo-Canosa, Ramón Fraga, Rita Sigüeiro, Maria Marco, Natacha Rochel, Dino Moras & Antonio Mouriño. (2010) Design and synthesis of active vitamin D analogs. The Journal of Steroid Biochemistry and Molecular Biology 121:1-2, pages 7-12.
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Pranjal Gogoi, Rita Sigüeiro, Silvina Eduardo & Antonio Mouriño. (2010)
An Expeditious Route to 1α,25‐Dihydroxyvitamin D
3
and Its Analogues by an Aqueous Tandem Palladium‐Catalyzed A‐Ring Closure and Suzuki Coupling to the C/D Unit
. Chemistry – A European Journal 16:5, pages 1432-1435.
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Daniel Nicoletti, Antonio Mouriño & Mercedes Torneiro. (2009)
Synthesis of 25-Hydroxyvitamin D
3
and 26,26,26,27,27,27-Hexadeutero-25-hydroxyvitamin D
3
on Solid Support
. The Journal of Organic Chemistry 74:13, pages 4782-4786.
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Peter Kolkhof, Lars Bärfacker, Alexander Hillisch, Helmut Haning & Stefan Schäfer. 2008. Nuclear Receptors as Drug Targets. Nuclear Receptors as Drug Targets
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Ricardo Riveiros, Antonio Rumbo, Luis A. Sarandeses & Antonio Mouriño. (2007) Synthesis and Conformational Analysis of 17α,21-Cyclo-22-Unsaturated Analogues of Calcitriol. The Journal of Organic Chemistry 72:15, pages 5477-5485.
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Natacha Rochel, Shinji Hourai, Xenxo Pérez-García, Antonio Rumbo, Antonio Mourino & Dino Moras. (2007) Crystal structure of the vitamin D nuclear receptor ligand binding domain in complex with a locked side chain analog of calcitriol. Archives of Biochemistry and Biophysics 460:2, pages 172-176.
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Carlos Gregorio, Silvina Eduardo, Luis C. Rodrigues, María A. Regueira, Ramón Fraga, Ricardo Riveiros, Miguel Maestro & Antonio Mouriño. (2007) Synthesis of two carboxylic haptens for raising antibodies to 25-hydroxyvitamin D3 and 1α,25-dihydroxyvitamin D3. The Journal of Steroid Biochemistry and Molecular Biology 103:3-5, pages 227-230.
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Ferdinand Molnár, Mikael Peräkylä & Carsten Carlberg. (2006) Vitamin D Receptor Agonists Specifically Modulate the Volume of the Ligand-binding Pocket. Journal of Biological Chemistry 281:15, pages 10516-10526.
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Xosé C. González-Avión, Antonio Mouriño, Natacha Rochel & Dino Moras. (2006)
Novel 1α,25-Dihydroxyvitamin D
3
Analogues with the Side Chain at C12
. Journal of Medicinal Chemistry 49:5, pages 1509-1516.
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Mikael Peräkylä, Marjo Malinen, Karl-Heinz Herzig & Carsten Carlberg. (2005) Gene Regulatory Potential of Nonsteroidal Vitamin D Receptor Ligands. Molecular Endocrinology 19:8, pages 2060-2073.
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M J Larriba & A Muñoz. (2005) SNAIL vs vitamin D receptor expression in colon cancer: therapeutics implications. British Journal of Cancer 92:6, pages 985-989.
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Anton Blencowe & Wayne Hayes. (2005) Development and application of diazirines in biological and synthetic macromolecular systems. Soft Matter 1:3, pages 178.
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Mikael Peräkylä, Ferdinand Molnár & Carsten Carlberg. (2004) A Structural Basis for the Species-Specific Antagonism of 26,23-Lactones on Vitamin D Signaling. Chemistry & Biology 11:8, pages 1147-1156.
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