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Sonja Nordhoff, Silvia Cerezo-Gálvez, Holger Deppe, Oliver Hill, Meritxell López-Canet, Christian Rummey, Meinolf Thiemann, Victor G. Matassa, Paul J. Edwards & Achim Feurer. (2009) Discovery of β-homophenylalanine based pyrrolidin-2-ylmethyl amides and sulfonamides as highly potent and selective inhibitors of dipeptidyl peptidase IV. Bioorganic & Medicinal Chemistry Letters 19:15, pages 4201-4203.
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Pieter Van der Veken, Ingrid De Meester, Véronique Dubois, Anna Soroka, Sebastiaan Van Goethem, Marie-Berthe Maes, Inger Brandt, Anne-Marie Lambeir, Xin Chen, Achiel Haemers, Simon Scharpé & Koen Augustyns. (2008) Inhibitors of dipeptidyl peptidase 8 and dipeptidyl peptidase 9. Part 1: Identification of dipeptide derived leads. Bioorganic & Medicinal Chemistry Letters 18:14, pages 4154-4158.
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Ki Dong Koo, Min Jung Kim, Sungsub Kim, Kyoung-Hee Kim, Sang Yong Hong, Gwong-Cheung Hur, Hyeon Joo Yim, Geun Tae Kim, Hee Oon Han, O Hwan Kwon, Tae Sik Kwon, Jong Sung Koh & Chang-Seok Lee. (2007) Synthesis, SAR, and X-ray structure of novel potent DPPIV inhibitors: Oxadiazolyl ketones. Bioorganic & Medicinal Chemistry Letters 17:15, pages 4167-4172.
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(2
S
,3
S
)-3-Amino-4-(3,3-difluoropyrrolidin-1-yl)-
N,N
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a
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David R. Magnin, Prakash C. Taunk, James G. Robertson, Aiying Wang, Jovita Marcinkeviciene, Mark S. Kirby & Lawrence G. Hamann. (2006) Seco-prolinenitrile inhibitors of dipeptidyl peptidase IV define minimal pharmacophore requirements at P1. Bioorganic & Medicinal Chemistry Letters 16:6, pages 1731-1734.
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