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Cheng Jiang & Qidong You. (2013) Kinesin spindle protein inhibitors in cancer: a patent review (2008 – present). Expert Opinion on Therapeutic Patents 23:12, pages 1547-1560.
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Hala Bakr El-Nassan. (2013) Advances in the discovery of kinesin spindle protein (Eg5) inhibitors as antitumor agents. European Journal of Medicinal Chemistry 62, pages 614-631.
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Cheng Jiang, Lei Yang, Wu-Tong Wu, Qing-Long Guo & Qi-Dong You. (2011) De novo design, synthesis and biological evaluation of 1,4-dihydroquinolin-4-ones and 1,2,3,4-tetrahydroquinazolin-4-ones as potent kinesin spindle protein (KSP) inhibitors. Bioorganic & Medicinal Chemistry 19:18, pages 5612-5627.
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Tomoki Takeuchi, Shinya Oishi, Toshiaki Watanabe, Hiroaki Ohno, Jun-ichi Sawada, Kenji Matsuno, Akira Asai, Naoya Asada, Kazuo Kitaura & Nobutaka Fujii. (2011) Structure–Activity Relationships of Carboline and Carbazole Derivatives as a Novel Class of ATP-Competitive Kinesin Spindle Protein Inhibitors. Journal of Medicinal Chemistry 54:13, pages 4839-4846.
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Makiko Shimizu, Hirosuke Ishii, Naohisa Ogo, Yuka Unno, Kenji Matsuno, Jun-ichi Sawada, Yasuto Akiyama & Akira Asai. (2010) S-trityl-L-cysteine derivative induces caspase-independent cell death in K562 human chronic myeloid leukemia cell line. Cancer Letters 298:1, pages 99-106.
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Shinya Oishi, Toshiaki Watanabe, Jun-ichi Sawada, Akira Asai, Hiroaki Ohno & Nobutaka Fujii. (2010) Kinesin Spindle Protein (KSP) Inhibitors with 2,3-Fused Indole Scaffolds. Journal of Medicinal Chemistry 53:13, pages 5054-5058.
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Xiangping Qian, Andrew McDonald, Han-Jie Zhou, Nicholas D. Adams, Cynthia A. Parrish, Kevin J. Duffy, Duke M. Fitch, Rosanna Tedesco, Luke W. Ashcraft, Bing Yao, Hong Jiang, Jennifer K. Huang, Melchor V. Marin, Carrie E. Aroyan, Jianchao Wang, Seyed Ahmed, Joelle L. Burgess, Amita M. Chaudhari, Carla A. Donatelli, Michael G. Darcy, Lance H. Ridgers, Ken A. Newlander, Stanley J. Schmidt, Deping Chai, Mariela Colón, Michael N. Zimmerman, Latesh Lad, Roman Sakowicz, Stephen Schauer, Lisa Belmont, Ramesh Baliga, Daniel W. Pierce, Jeffrey T. Finer, Zhengping Wang, Bradley P. Morgan, David J. MorgansJr.Jr., Kurt R. Auger, Chiu-Mei Sung, Jeff D. Carson, Lusong Luo, Erin D. Hugger, Robert A. Copeland, David Sutton, John D. Elliott, Jeffrey R. Jackson, Kenneth W. Wood, Dashyant Dhanak, Gustave Bergnes & Steven D. Knight. (2010) Discovery of the First Potent and Selective Inhibitor of Centromere-Associated Protein E: GSK923295. ACS Medicinal Chemistry Letters 1:1, pages 30-34.
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Makiko Shimizu, Hirosuke Ishii, Naohisa Ogo, Kenji Matsuno & Akira Asai. (2010) Biochemical analysis of cellular target of S-trityl-l-cysteine derivatives using affinity matrix. Bioorganic & Medicinal Chemistry Letters 20:5, pages 1578-1580.
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Patricia A. McDonnell, Joseph Yanchunas, John A. Newitt, Li Tao, Susan E. Kiefer, Marie Ortega, Stephanie Kut, Neil Burford, Valentina Goldfarb, Gerald J. Duke, Henry Shen, William Metzler, Michael Doyle, Zhong Chen, Christine Tarby, Robert Borzilleri, Wayne Vaccaro, Marco Gottardis, Songfeng Lu, Donald Crews, Kyoung Kim, Louis Lombardo & Deborah L. Roussell. (2009) Assessing compound binding to the Eg5 motor domain using a thermal shift assay. Analytical Biochemistry 392:1, pages 59-69.
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Kenji Matsuno, Jun-ichi Sawada, Mina Sugimoto, Naohisa Ogo & Akira Asai. (2009) Bis(hetero)aryl derivatives as unique kinesin spindle protein inhibitors. Bioorganic & Medicinal Chemistry Letters 19:4, pages 1058-1061.
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