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Expert Opinion on Therapeutic Patents Volume 22, 2012 - Issue 8
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5HT6 receptor antagonists: a patent update. Part 1. Sulfonyl derivatives

Alexandre V IvachtchenkoChemDiv, Inc., 6605 Nancy Ridge Drive, San Diego, CA 92121, USA+1 858 794 4860; +1 858 794 4931; [email protected];Chemical Diversity Research Institute, Department of Organic Chemistry, 114401 Khimki, Moscow Reg, Russia
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Yan A IvanenkovChemDiv, Inc., 6605 Nancy Ridge Drive, San Diego, CA 92121, USA+1 858 794 4860; +1 858 794 4931; [email protected];Chemical Diversity Research Institute, Department of Computational Medicinal Chemistry, 114401 Khimki, Moscow Reg, Russia
Pages 917-964 | Published online: 20 Jul 2012

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Alberto Leoni, Alessandra Locatelli, Rita Morigi & Mirella Rambaldi. (2014) Novel thiazole derivatives: a patent review (2008 – 2012. Part 2). Expert Opinion on Therapeutic Patents 24:7, pages 759-777.
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Alexandre V Ivachtchenko, Yan A Ivanenkov & Andrey V Skorenko. (2012) 5-HT6 receptor modulators: a patent update. Part 2. Diversity in heterocyclic scaffolds. Expert Opinion on Therapeutic Patents 22:10, pages 1123-1168.
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Articles from other publishers (12)

Galal H. Elgemeie, Rasha A. Azzam, Wafaa A. Zaghary, Ashraf A. Aly, Nadia H. Metwally, Mona O. Sarhan, Elshimaa M. Abdelhafez & Rasha E. Elsayed. 2022. N-Sulfonated-N-Heterocycles. N-Sulfonated-N-Heterocycles 383 415 .
Noriko Nakano, Satoru Matsuda, Mayuko Ichimura, Akari Minami, Mako Ogino, Toshiyuki Murai & Yasuko Kitagishi. (2017) PI3K/AKT signaling mediated by G protein-coupled receptors is involved in neurodegenerative Parkinson's disease (Review). International Journal of Molecular Medicine 39:2, pages 253-260.
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Hilda Ferrero, Maite Solas, Paul T. Francis & Maria J. Ramirez. (2016) Serotonin 5-HT6 Receptor Antagonists in Alzheimer’s Disease: Therapeutic Rationale and Current Development Status. CNS Drugs 31:1, pages 19-32.
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Alexandre V. Ivachtchenko, Yan Lavrovsky & Ilya Okun. (2016) AVN-101: A Multi-Target Drug Candidate for the Treatment of CNS Disorders. Journal of Alzheimer's Disease 53:2, pages 583-620.
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Dmitrii A. Vasilevskii, Vladimir S. Yashchenko & Vyacheslav K. Ol’khovik. (2016) Synthesis of heterofunctional 3,3'-sulfonyldibenzoic acid derivatives. Chemistry of Heterocyclic Compounds 52:2, pages 128-132.
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Vittorio Canale, Rafał Kurczab, Anna Partyka, Grzegorz Satała, Karolina Słoczyńska, Tomasz Kos, Magdalena Jastrzębska-Więsek, Agata Siwek, Elżbieta Pękala, Andrzej J. Bojarski, Anna Wesołowska, Piotr Popik & Paweł Zajdel. (2016) N-Alkylated arylsulfonamides of (aryloxy)ethyl piperidines: 5-HT7 receptor selectivity versus multireceptor profile. Bioorganic & Medicinal Chemistry 24:2, pages 130-139.
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A. V. Ivachtchenko, E. S. Golovina, M. G. Kadieva, O. D. Mitkin & I. M. Okun. (2015) Antagonists of Serotonin 5-HT6 Receptors. VI. Substituted 3-(Phenylsulfonyl)Quinolines, Synthesis and Structure–Activity Relationships. Pharmaceutical Chemistry Journal 48:10, pages 646-660.
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Bellinda Benhamú, Mar Martín-Fontecha, Henar Vázquez-Villa, Leonardo Pardo & María L. López-Rodríguez. (2014) Serotonin 5-HT 6 Receptor Antagonists for the Treatment of Cognitive Deficiency in Alzheimer’s Disease . Journal of Medicinal Chemistry 57:17, pages 7160-7181.
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A V Ivachtchenko. (2014) Sulfonyl-containing modulators of serotonin 5-HT 6 receptors and their pharmacophore models . Russian Chemical Reviews 83:5, pages 439-473.
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. 2014. The Role of 5-HT Systems on Memory and Dysfunctional Memory. The Role of 5-HT Systems on Memory and Dysfunctional Memory 67 84 .
Alfredo Meneses. 2014. Identification of Neural Markers Accompanying Memory. Identification of Neural Markers Accompanying Memory 5 45 .
Alexandre Ivachtchenko, Elena Golovina, Madina Kadieva, Oleg Mitkin, Sergei Tkachenko & Ilya Okun. (2013) Synthesis of substituted diphenyl sulfones and their structure–activity relationship with the antagonism of 5-НТ6 receptors. Bioorganic & Medicinal Chemistry 21:15, pages 4614-4627.
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