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Expert Opinion on Therapeutic Patents Volume 22, 2012 - Issue 10
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5-HT6 receptor modulators: a patent update. Part 2. Diversity in heterocyclic scaffolds

Alexandre V IvachtchenkoChemDiv, Inc., 6605 Nancy Ridge Drive, San Diego, CA 92121, USA;Chemical Diversity Research Institute, Department of Computational Medicinal Chemistry, 114401 Khimki, Moscow Reg, Russia+858 794 4860; +858 794 4931; [email protected]
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Yan A IvanenkovChemDiv, Inc., 6605 Nancy Ridge Drive, San Diego, CA 92121, USA;Chemical Diversity Research Institute, Department of Computational Medicinal Chemistry, 114401 Khimki, Moscow Reg, Russia+858 794 4860; +858 794 4931; [email protected]
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Andrey V SkorenkoChemical Diversity Research Institute, Department of Computational Medicinal Chemistry, 114401 Khimki, Moscow Reg, Russia+858 794 4860; +858 794 4931; [email protected]
Pages 1123-1168 | Published online: 07 Sep 2012

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Alberto Leoni, Alessandra Locatelli, Rita Morigi & Mirella Rambaldi. (2014) Novel thiazole derivatives: a patent review (2008 – 2012. Part 2). Expert Opinion on Therapeutic Patents 24:7, pages 759-777.
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Articles from other publishers (12)

Shuwirda Boon Seen, Yu Gong & Mark Ashton. 2023. 1 85 .
Galal H. Elgemeie, Rasha A. Azzam, Wafaa A. Zaghary, Ashraf A. Aly, Nadia H. Metwally, Mona O. Sarhan, Elshimaa M. Abdelhafez & Rasha E. Elsayed. 2022. N-Sulfonated-N-Heterocycles. N-Sulfonated-N-Heterocycles 383 415 .
Hilda Ferrero, Maite Solas, Paul T. Francis & Maria J. Ramirez. (2016) Serotonin 5-HT6 Receptor Antagonists in Alzheimer’s Disease: Therapeutic Rationale and Current Development Status. CNS Drugs 31:1, pages 19-32.
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Alexandre V. Ivachtchenko, Yan Lavrovsky & Ilya Okun. (2016) AVN-101: A Multi-Target Drug Candidate for the Treatment of CNS Disorders. Journal of Alzheimer's Disease 53:2, pages 583-620.
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Paweł Zajdel, Krzysztof Marciniec, Grzegorz Satała, Vittorio Canale, Tomasz Kos, Anna Partyka, Magdalena Jastrzębska-Więsek, Anna Wesołowska, Agnieszka Basińska-Ziobroń, Jacek Wójcikowski, Władysława A. Daniel, Andrzej J. Bojarski & Piotr Popik. (2016) N 1-Azinylsulfonyl-1 H -indoles: 5-HT6 Receptor Antagonists with Procognitive and Antidepressant-Like Properties . ACS Medicinal Chemistry Letters 7:6, pages 618-622.
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Jakub Staroń, Dawid Warszycki, Justyna Kalinowska-Tłuścik, Grzegorz Satała & Andrzej J. Bojarski. (2015) Rational design of 5-HT 6 R ligands using a bioisosteric strategy: synthesis, biological evaluation and molecular modelling . RSC Advances 5:33, pages 25806-25815.
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Leonid I. Belen'kii & Yu B. Evdokimenkova. 2015. 193 363 .
A. V. Ivachtchenko, E. S. Golovina, M. G. Kadieva, O. D. Mitkin & I. M. Okun. (2015) Antagonists of Serotonin 5-HT6 Receptors. VI. Substituted 3-(Phenylsulfonyl)Quinolines, Synthesis and Structure–Activity Relationships. Pharmaceutical Chemistry Journal 48:10, pages 646-660.
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A V Ivachtchenko. (2014) Sulfonyl-containing modulators of serotonin 5-HT 6 receptors and their pharmacophore models . Russian Chemical Reviews 83:5, pages 439-473.
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. 2014. The Role of 5-HT Systems on Memory and Dysfunctional Memory. The Role of 5-HT Systems on Memory and Dysfunctional Memory 67 84 .
Alfredo Meneses. 2014. Identification of Neural Markers Accompanying Memory. Identification of Neural Markers Accompanying Memory 5 45 .
Alexandre Ivachtchenko, Elena Golovina, Madina Kadieva, Oleg Mitkin, Sergei Tkachenko & Ilya Okun. (2013) Synthesis of substituted diphenyl sulfones and their structure–activity relationship with the antagonism of 5-НТ6 receptors. Bioorganic & Medicinal Chemistry 21:15, pages 4614-4627.
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