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DNA methyltransferase inhibitors in cancer: a chemical and therapeutic patent overview and selected clinical studies

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Pages 1427-1442 | Published online: 03 Oct 2012

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Guoliang Cui, Can Wang, Zhenyan Lin, Xiaoke Feng, Muxin Wei, Zhengyue Miao, Zhiguang Sun & Fei Wei. (2021) Prognostic and immunological role of Ras-related protein Rap1b in pan-cancer. Bioengineered 12:1, pages 4828-4840.
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Inkyung Jung, Jungeun An & Myunggon Ko. (2023) Epigenetic Regulators of DNA Cytosine Modification: Promising Targets for Cancer Therapy. Biomedicines 11:3, pages 654.
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Zongliang Zhang, Guoqing Wang, Kunhong Zhong, Yongdong Chen, Nian Yang, Qizhong Lu, Boyang Yuan, Zeng Wang, Hexian Li, Liping Guo, Ruyuan Zhang, Zhiguo Wu, Meijun Zheng, Shasha Zhao, Xin Tang, Bin Shao & Aiping Tong. (2023) A drug screening to identify novel combinatorial strategies for boosting cancer immunotherapy efficacy. Journal of Translational Medicine 21:1.
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Sook Ho Kim, Hae Jun Jung & Seok-Cheol Hong. (2021) Z-DNA as a Tool for Nuclease-Free DNA Methyltransferase Assay. International Journal of Molecular Sciences 22:21, pages 11990.
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Wenjing Xiao, Qiaodan Zhou, Xudong Wen, Rui Wang, Ruijie Liu, Tingting Wang, Jianyou Shi, Yonghe Hu & Jun Hou. (2021) Small-Molecule Inhibitors Overcome Epigenetic Reprogramming for Cancer Therapy. Frontiers in Pharmacology 12.
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