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Expert Opinion on Therapeutic Patents Volume 23, 2013 - Issue 2
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Falcipain inhibitors as potential therapeutics for resistant strains of malaria: a patent review

Uttam Rajaram ManeThe M. S. University of Baroda, Pharmacy Department, Faculty of Tech. and Engg, Vadodara, 390001, Gujarat, India+91 265 2434187; +91 265 2418927; [email protected];Torrent Research Centre, Village Bhat, Dist. Gandhinagar, 382421, Gujarat, India
,
Ramesh C GuptaTorrent Research Centre, Village Bhat, Dist. Gandhinagar, 382421, Gujarat, India
,
Sunil Sadanand NadkarniTorrent Research Centre, Village Bhat, Dist. Gandhinagar, 382421, Gujarat, India
,
Rajani R GiridharThe M. S. University of Baroda, Pharmacy Department, Faculty of Tech. and Engg, Vadodara, 390001, Gujarat, India+91 265 2434187; +91 265 2418927; [email protected]
,
Prashant Prakash NaikThe M. S. University of Baroda, Pharmacy Department, Faculty of Tech. and Engg, Vadodara, 390001, Gujarat, India+91 265 2434187; +91 265 2418927; [email protected]
&
Mange R YadavThe M. S. University of Baroda, Pharmacy Department, Faculty of Tech. and Engg, Vadodara, 390001, Gujarat, India+91 265 2434187; +91 265 2418927; [email protected]
Pages 165-187 | Published online: 11 Dec 2012

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Thommas M. Musyoka, Aquillah M. Kanzi, Kevin A. Lobb & Özlem Tastan Bishop. (2016) Analysis of non-peptidic compounds as potential malarial inhibitors against Plasmodial cysteine proteases via integrated virtual screening workflow. Journal of Biomolecular Structure and Dynamics 34:10, pages 2084-2101.
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Erick Tavares Marcelino Alves, Filipe Gomes Pernichelle, Lucas Adriano Nascimento, Glaucio Monteiro Ferreira & Elizabeth Igne Ferreira. (2023) Covalent Inhibitors for Neglected Diseases: An Exploration of Novel Therapeutic Options. Pharmaceuticals 16:7, pages 1028.
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Lik Tong Tan & Ma Yadanar Phyo. (2020) Marine Cyanobacteria: A Source of Lead Compounds and their Clinically-Relevant Molecular Targets. Molecules 25:9, pages 2197.
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Thommas Mutemi Musyoka, Joyce Njoki Njuguna & Özlem Tastan Bishop. (2019) Comparing sequence and structure of falcipains and human homologs at prodomain and catalytic active site for malarial peptide based inhibitor design. Malaria Journal 18:1.
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Rafael Pinto Vieira, Viviane Corrêa Santos & Rafaela Salgado Ferreira. (2019) Structure-based Approaches Targeting Parasite Cysteine Proteases. Current Medicinal Chemistry 26:23, pages 4435-4453.
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Mohd Asad, Azhar Muneer, Pradeep Kumar, Vandana Thakur, Sumit Rathore, Pawan Malhotra & Asif Mohmmed. 2019. Pathogenicity and Drug Resistance of Human Pathogens. Pathogenicity and Drug Resistance of Human Pathogens 181 211 .
Ayodeji A. Agbowuro, Wilhelmina M. Huston, Allan B. Gamble & Joel D. A. Tyndall. (2018) Proteases and protease inhibitors in infectious diseases. Medicinal Research Reviews 38:4, pages 1295-1331.
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Lik Tong Tan. 2017. Natural Products Targeting Clinically Relevant Enzymes. Natural Products Targeting Clinically Relevant Enzymes 19 43 .
Emir Salas-Sarduy, Yasel Guerra, Giovanni Covaleda Cortés, Francesc Avilés & María Chávez Planes. (2017) Identification of Tight-Binding Plasmepsin II and Falcipain 2 Inhibitors in Aqueous Extracts of Marine Invertebrates by the Combination of Enzymatic and Interaction-Based Assays. Marine Drugs 15:4, pages 123.
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Vasanthanathan Poongavanam & Jacob Kongsted. (2016) Binding affinity models for Falcipain inhibition based on the Linear Interaction Energy method. Journal of Molecular Graphics and Modelling 70, pages 236-245.
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Rudi Oliveira, Daniela Miranda, Joana Magalhães, Rita Capela, Maria J. Perry, Paul M. O’Neill, Rui Moreira & Francisca Lopes. (2015) From hybrid compounds to targeted drug delivery in antimalarial therapy. Bioorganic & Medicinal Chemistry 23:16, pages 5120-5130.
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Sai Kumar Chakka, Mohammad Kalamuddin, Srividhya Sundararaman, Lianhu Wei, Sourabh Mundra, Radhakrishnan Mahesh, Pawan Malhotra, Asif Mohmmed & Lakshmi P. Kotra. (2015) Identification of novel class of falcipain-2 inhibitors as potential antimalarial agents. Bioorganic & Medicinal Chemistry 23:9, pages 2221-2240.
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Elke Persch, Oliver Dumele & François Diederich. (2015) Molecular Recognition in Chemical and Biological Systems. Angewandte Chemie International Edition 54:11, pages 3290-3327.
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Elke Persch, Oliver Dumele & François Diederich. (2015) Molekulare Erkennung in chemischen und biologischen Systemen. Angewandte Chemie 127:11, pages 3341-3382.
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Jinghui Wang, Feng Li, Yan Li, Yinfeng Yang, Shuwei Zhang & Ling Yang. (2013) Structural features of falcipain-3 inhibitors: an in silico study. Molecular BioSystems 9:9, pages 2296.
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Sumit Rathore, Shaifali Jain, MohD Asad, Gaurav Datta, Pawan Malhotra & Asif Mohmmed. 2013. Proteases in Health and Disease. Proteases in Health and Disease 215 242 .

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