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Corticotropin-releasing factor 1 receptor antagonists: a patent review

Pages 1057-1068 | Published online: 04 May 2013

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Mishra Shashank Shekhar, T. Venkatachalam, Chandra Shekhar Sharma, Hemendra Pratap Singh, Sourav Kalra & Neeraj Kumar. (2019) Computational investigation of binding mechanism of substituted pyrazinones targeting corticotropin releasing factor-1 receptor deliberated for anti-depressant drug design. Journal of Biomolecular Structure and Dynamics 37:12, pages 3226-3244.
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Neeraj Kumar, Shashank Shekhar Mishra, Chandra Shekhar Sharma, Hamendra Pratap Singh & Sourav Kalra. (2018) In silico binding mechanism prediction of benzimidazole based corticotropin releasing factor-1 receptor antagonists by quantitative structure activity relationship, molecular docking and pharmacokinetic parameters calculation. Journal of Biomolecular Structure and Dynamics 36:7, pages 1691-1712.
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Articles from other publishers (11)

Muriel Larauche, Judit Erchegyi, Charleen Miller, Myung Shin Sim, Jean Rivier, Dominic Behan & Yvette Taché. (2022) Peripheral CRF-R1/CRF-R2 antagonist, astressin C, induces a long-lasting blockade of acute stress-related visceral pain in male and female rats. Peptides 157, pages 170881.
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Yuanxia Lv, Jing Wen, Yingying Fang, Haoyuan Zhang & Jianwu Zhang. (2022) Corticotropin-releasing factor receptor 1 (CRF-R1) antagonists: Promising agents to prevent visceral hypersensitivity in irritable bowel syndrome. Peptides 147, pages 170705.
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Takuto Kojima, Michiyo Mochizuki, Takafumi Takai, Yasutaka Hoashi, Sachie Morimoto, Masaki Seto, Minoru Nakamura, Katsumi Kobayashi, Yuu Sako, Maiko Tanaka, Naoyuki Kanzaki, Yohei Kosugi, Takahiko Yano & Kazuyoshi Aso. (2018) Discovery of 1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazoles as novel class of corticotropin releasing factor 1 receptor antagonists. Bioorganic & Medicinal Chemistry 26:9, pages 2229-2250.
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Michiyo Mochizuki, Takuto Kojima, Katsumi Kobayashi, Etsuo Kotani, Yuji Ishichi, Naoyuki Kanzaki, Hideyuki Nakagawa, Teruaki Okuda, Yohei Kosugi, Takahiko Yano, Yuu Sako, Maiko Tanaka & Kazuyoshi Aso. (2017) Discovery of 4-chloro-2-(2,4-dichloro-6-methylphenoxy)-1-methyl-7-(pentan-3-yl)-1H-benzimidazole, a novel CRF1 receptor antagonist. Bioorganic & Medicinal Chemistry 25:5, pages 1556-1570.
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Yasuhiro Sawai, Osamu Yabe, Keiichiro Nakaoka & Tomomi Ikemoto. (2017) Process Development of a CRF 1 Receptor Antagonist Based on the Selective Chlorination of a Benzimidazolone via Chlorine Migration . Organic Process Research & Development 21:2, pages 222-230.
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Michiyo Mochizuki, Masakuni Kori, Mitsunori Kono, Takahiko Yano, Yuu Sako, Maiko Tanaka, Naoyuki Kanzaki, Albert C. Gyorkos, Christopher P. Corrette & Kazuyoshi Aso. (2016) Discovery of a 7-arylaminobenzimidazole series as novel CRF1 receptor antagonists. Bioorganic & Medicinal Chemistry 24:19, pages 4675-4691.
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Michiyo Mochizuki, Masakuni Kori, Katsumi Kobayashi, Takahiko Yano, Yuu Sako, Maiko Tanaka, Naoyuki Kanzaki, Albert C. Gyorkos, Christopher P. Corrette, Suk Young Cho, Scott A. Pratt & Kazuyoshi Aso. (2016) Design and Synthesis of Benzimidazoles As Novel Corticotropin-Releasing Factor 1 Receptor Antagonists. Journal of Medicinal Chemistry 59:6, pages 2551-2566.
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Jinmei Yu, Rengong Zhuo, Peng Peng, Xiaoyan Liu, Haitao Yan, Shuzhuo Zhang, Jianquan Zheng, Xiaoli Wei & Xiaoyun Ma. (2015) P7, a novel antagonist of corticotropin releasing factor receptor type 1 (CRFR1) screened from phage display library. Biochemical and Biophysical Research Communications 463:3, pages 200-204.
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Yvette Taché & Mulugeta Million. (2015) Role of Corticotropin-releasing Factor Signaling in Stress-related Alterations of Colonic Motility and Hyperalgesia. Journal of Neurogastroenterology and Motility 21:1, pages 008-024.
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Felix Hausch. (2013) Structures of Class B G Protein‐Coupled Receptors: Prospects for Drug Discovery. Angewandte Chemie International Edition 52:49, pages 12783-12785.
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Felix Hausch. (2013) Strukturen der G-Protein-gekoppelten Rezeptoren der Klasse B: Perspektiven für die Arzneimittelforschung. Angewandte Chemie 125:49, pages 13017-13019.
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