Citations (40)
Keep up to date with the latest research on this topic with citation updates for this article.
Read on this site (4)
Mohamed Moussaoui, Mouna Baassi, Soukayna Baammi, Hatim Soufi, Mohammed Salah, Rachid Daoud, Achraf EL Allali, M.E. Belghiti & Said Belaaouad. (2023) In silico design of novel CDK2 inhibitors through QSAR, ADMET, molecular docking and molecular dynamics simulation studies. Journal of Biomolecular Structure and Dynamics 0:0, pages 1-17.
Read now
Read now
Vincent A. Obakachi, Idowu Kehinde, Narva Deshwar Kushwaha, Olayinka I. Akinpelu, Babita Kushwaha, Srinivas Reddy Merugu, Francis Kayamba, Hezekiel M. Kumalo & Rajshekhar Karpoormath. (2022) Structural based investigation of novel pyrazole-thiazole Hybrids as dual CDK-1 and CDK-2 inhibitors for cancer chemotherapy. Molecular Simulation 48:8, pages 687-701.
Read now
Read now
Ahmed Kamal, Syed Mohammed Ali Hussaini, Abdul Rahim & Syed Riyaz. (2015) Podophyllotoxin derivatives: a patent review (2012 – 2014). Expert Opinion on Therapeutic Patents 25:9, pages 1025-1034.
Read now
Read now
Alberto Leoni, Alessandra Locatelli, Rita Morigi & Mirella Rambaldi. (2014) Novel thiazole derivatives: a patent review (2008 – 2012. Part 2). Expert Opinion on Therapeutic Patents 24:7, pages 759-777.
Read now
Read now
Articles from other publishers (36)
Burak Kuzu, Ali Ergüç, Fuat Karakuş & Ege Arzuk. (2023) Design, synthesis, and antiproliferative activities of novel thiazolyl-pyrazole hybrid derivatives. Medicinal Chemistry Research 32:8, pages 1690-1700.
Crossref
Crossref
Merve Bardakkaya, Burcu Kilic, Rahsan Ilıkcı Sagkan, Fatma Aksakal, Shakila Shakila & Deniz S. Dogruer. (2023) Synthesis and evaluation of multitarget new 2‐aminothiazole derivatives as potential anti‐Alzheimer's agents. Archiv der Pharmazie 356:8.
Crossref
Crossref
Burcu Kilic, Merve Bardakkaya, Rahsan Ilıkcı Sagkan, Fatma Aksakal, Shakila Shakila & Deniz S. Dogruer. (2023) New thiourea and benzamide derivatives of 2-aminothiazole as multi-target agents against Alzheimer's disease: Design, synthesis, and biological evaluation. Bioorganic Chemistry 131, pages 106322.
Crossref
Crossref
Benson M. Kariuki, Bakr F. Abdel-Wahab, Hanan A. Mohamed, Mohamed S. Bekheit & Gamal A. El-Hiti. (2022) Synthesis and Characterization of Novel 2-(1,2,3-Triazol-4-yl)-4,5-dihydro-1H-pyrazol-1-yl)thiazoles and 2-(4,5-Dihydro-1H-pyrazol-1-yl)-4-(1H-1,2,3-triazol-4-yl)thiazoles. Molecules 27:24, pages 8904.
Crossref
Crossref
Gaofeng Yin, Xiaodong Wang, Yuqing Wang, Tao Shi, Yaofu Zeng, Yuying Wang, Xue Peng & Zhen Wang. (2022) Lawesson's reagent promoted deoxygenation of azlactones for the syntheses of 2,4-disubstituted thiazoles. Organic & Biomolecular Chemistry 20:48, pages 9589-9592.
Crossref
Crossref
Müjgan Yaman, Ezgi İpek Dirin, Gökhan Kaplan, Nurgül Seferoğlu & Zeynel Seferoğlu. (2022) The synthesis, photophysical properties, DFT study and textile applications of fluorescent azo dyes bearing coumarin-thiazole. Journal of Molecular Liquids 368, pages 120718.
Crossref
Crossref
Sajid Ali Channar, Pervaiz Ali Channar, Aamer Saeed, Aisha A. Alsfouk, Syeda Abida Ejaz, Rabail Ujan, Razia Noor, Muhammad Sajjad Bilal, Qamar Abbas, Zahid Hussain, Bilal Ahmad Khan, Hussain Raza, Hafiz Abdul Bari Indher & Parvez Ali Mahesar. (2022) Exploring thiazole-linked thioureas using alkaline phosphatase assay, biochemical evaluation, computational analysis and structure–activity relationship (SAR) studies. Medicinal Chemistry Research 31:10, pages 1792-1802.
Crossref
Crossref
Prajakta Shamrao Sadavarte, Bhaskar Hari Zaware & Sushama Jayawant Takate. (2022) Kinetics of Thiazole Formation Using α-Halo Ketones and Thioamides. Oriental Journal Of Chemistry 38:4, pages 1031-1036.
Crossref
Crossref
Thoraya A. Farghaly, Eman M.H. Abbas, Amerah M. Al-Soliemy, Rehab Sabour & Mohamed R. Shaaban. (2022) Novel sulfonyl thiazolyl-hydrazone derivatives as EGFR inhibitors: Design, synthesis, biological evaluation and molecular docking studies. Bioorganic Chemistry 121, pages 105684.
Crossref
Crossref
A. V. Lozynskyi, I. M. Yushyn, Yu. T. Konechnyi, O. M. Roman, O. V. Matiykiv, O. V. Smaliukh, L. M. Mosula, S. V. Polovkovych & R. B. Lesyk. (2021) Synthesis and evaluation of biological activity of 1-[2-amino-4-methylthiazol-5-yl]-3-arylpropenones. Biopolymers and Cell 37:5, pages 389-399.
Crossref
Crossref
Kamal M. Dawood, Mohamed A. Raslan, Ashraf A. Abbas, Belal E. Mohamed, Magda H. Abdellattif, Mohamed S. Nafie & Mohamed K. Hassan. (2021) Novel Bis-Thiazole Derivatives: Synthesis and Potential Cytotoxic Activity Through Apoptosis With Molecular Docking Approaches. Frontiers in Chemistry 9.
Crossref
Crossref
Dinesh Kumar, Vamsi Krishna Kommalapati, Mahesh Kumar Jerald & Anjana Devi Tangutur. (2021) Fluorinated thiazolidinol drives autophagic cell death in pancreatic cancer cells via AMPK activation and perturbation of critical sentinels of oncogenic signaling. Chemico-Biological Interactions 343, pages 109433.
Crossref
Crossref
Ebru Zeytün, Mehlika D. Altıntop, Belgin Sever, Ahmet Özdemir, Doha E. Ellakwa, Zeynep Ocak, Halil I. Ciftci, Masami Otsuka, Mikako Fujita & Mohamed O. Radwan. (2021) A New Series of Antileukemic Agents: Design, Synthesis, In Vitro and In Silico Evaluation of Thiazole-Based ABL1 Kinase Inhibitors. Anti-Cancer Agents in Medicinal Chemistry 21:9, pages 1099-1109.
Crossref
Crossref
Rebaz Omar, Pelin Koparir & Metin Koparir. (2021) SYNTHESIS OF 1,3-THIAZOLE DERIVATIVES. INDIAN DRUGS 58:01, pages 7-19.
Crossref
Crossref
Rizk E. Khidre & Ibrahim Ali M. Radini. (2021) Design, synthesis and docking studies of novel thiazole derivatives incorporating pyridine moiety and assessment as antimicrobial agents. Scientific Reports 11:1.
Crossref
Crossref
Anca-Maria Borcea, Ioana Ionuț, Ovidiu Crișan & Ovidiu Oniga. (2021) An Overview of the Synthesis and Antimicrobial, Antiprotozoal, and Antitumor Activity of Thiazole and Bisthiazole Derivatives. Molecules 26:3, pages 624.
Crossref
Crossref
Mohd Adil Shareef, Irfan Khan, Bathini Nagendra Babu & Ahmed Kamal. (2020) A Comprehensive Review on the Therapeutic Versatility of Imidazo [2,1-b]thiazoles. Current Medicinal Chemistry 27:40, pages 6864-6887.
Crossref
Crossref
Huda K. Mahmoud, Thoraya A. Farghaly, Hanan G. Abdulwahab, Nadia T. Al-Qurashi & Mohamed R. Shaaban. (2020) Novel 2-indolinone thiazole hybrids as sunitinib analogues: Design, synthesis, and potent VEGFR-2 inhibition with potential anti-renal cancer activity. European Journal of Medicinal Chemistry 208, pages 112752.
Crossref
Crossref
Belgin Sever, Cüneyt Türkeş, Mehlika Dilek Altıntop, Yeliz Demir & Şükrü Beydemir. (2020) Thiazolyl-pyrazoline derivatives: In vitro and in silico evaluation as potential acetylcholinesterase and carbonic anhydrase inhibitors. International Journal of Biological Macromolecules 163, pages 1970-1988.
Crossref
Crossref
Emanuela Pesce, Nicoletta Pedemonte, Alberto Leoni, Alessandra Locatelli & Rita Morigi. (2020) Synthesis and biological evaluation of thiazole derivatives on basic defects underlying cystic fibrosis. Bioorganic & Medicinal Chemistry Letters 30:21, pages 127473.
Crossref
Crossref
Ahmed S. M. Al‐Janabi, Rania Zaky, Tarak A. Yousef, Bashar S. Nomi & Saad Shaaban. (2020) Synthesis, characterization, computational simulation, biological and anticancer evaluation of Pd(II), Pt(II), Zn(II), Cd(II), and Hg(II) complexes with 2‐amino‐4‐phenyl‐5‐selenocyanatothiazol ligand. Journal of the Chinese Chemical Society 67:6, pages 1032-1044.
Crossref
Crossref
Serpil Eryılmaz, Emine Türk Çelikoğlu, Önder İdil, Ersin İnkaya, Zehra Kozak, Ender Mısır & Melek Gül. (2020) Derivatives of pyridine and thiazole hybrid: Synthesis, DFT, biological evaluation via antimicrobial and DNA cleavage activity. Bioorganic Chemistry 95, pages 103476.
Crossref
Crossref
Georgios Charitos, Dimitrios T. Trafalis, Panayiotis Dalezis, Constantinos Potamitis, Vasiliki Sarli, Panagiotis Zoumpoulakis & Charalambos Camoutsis. (2019) Synthesis and anticancer activity of novel 3,6-disubstituted 1,2,4-triazolo-[3,4-b]-1,3,4-thiadiazole derivatives. Arabian Journal of Chemistry 12:8, pages 4784-4794.
Crossref
Crossref
Pedro Brandão, Marta Pineiro & Teresa M. V. D. Pinho e Melo. (2019) Flow Chemistry: Towards A More Sustainable Heterocyclic Synthesis. European Journal of Organic Chemistry 2019:43, pages 7188-7217.
Crossref
Crossref
Belgin Sever, Mehlika Dilek Altıntop, Mohamed O. Radwan, Ahmet Özdemir, Masami Otsuka, Mikako Fujita & Halil I. Ciftci. (2019) Design, synthesis and biological evaluation of a new series of thiazolyl-pyrazolines as dual EGFR and HER2 inhibitors. European Journal of Medicinal Chemistry 182, pages 111648.
Crossref
Crossref
Adileh Ayati, Saeed Emami, Setareh Moghimi & Alireza Foroumadi. (2019) Thiazole in the targeted anticancer drug discovery. Future Medicinal Chemistry 11:15, pages 1929-1952.
Crossref
Crossref
Anuradha, Sagarkumar Patel, Rajkumar Patle, Preethi Parameswaran, Alok Jain & Amit Shard. (2019) Design, computational studies, synthesis and biological evaluation of thiazole-based molecules as anticancer agents. European Journal of Pharmaceutical Sciences 134, pages 20-30.
Crossref
Crossref
Ismail Althagafi, Nashwa El-Metwaly & Thoraya A. Farghaly. (2019) New Series of Thiazole Derivatives: Synthesis, Structural Elucidation, Antimicrobial Activity, Molecular Modeling and MOE Docking. Molecules 24:9, pages 1741.
Crossref
Crossref
Runjhun Tandon, Iqubal Singh, Vijay Luxami, Nitin Tandon & Kamaldeep Paul. (2018)
Recent Advances and Developments of
in vitro
Evaluation of Heterocyclic Moieties on Cancer Cell Lines
. The Chemical Record 19:2-3, pages 362-393.
Crossref
Crossref
Swarnagowri Nayak & Santhosh L. Gaonkar. (2019) A Review on Recent Synthetic Strategies and Pharmacological Importance of 1,3-Thiazole Derivatives. Mini-Reviews in Medicinal Chemistry 19:3, pages 215-238.
Crossref
Crossref
Murtaza Madni, Muhammad Naeem Ahmed, Shahid Hameed, Syed Wadood Ali Shah, Umer Rashid, Khurshid Ayub, M.Nawaz Tahir & Tariq Mahmood. (2018) Synthesis, quantum chemical, in vitro acetyl cholinesterase inhibition and molecular docking studies of four new coumarin based pyrazolylthiazole nuclei. Journal of Molecular Structure 1168, pages 175-186.
Crossref
Crossref
Marta Reig, Ramón Bosque, Mercè Font-Bardía, Carme Calvis, Ramon Messeguer, Laura Baldomà, Josefa Badía, Dolores Velasco & Concepción López. (2018) A study of the properties, reactivity and anticancer activity of novel N-methylated-3-thiazolyl or 3-thienyl carbazoles and their Pd(II) and Pt(II) complexes. Journal of Inorganic Biochemistry 184, pages 134-145.
Crossref
Crossref
Mehlika Altıntop, Belgin Sever, Gülşen Akalın Çiftçi & Ahmet Özdemir. (2018) Design, Synthesis, and Evaluation of a New Series of Thiazole-Based Anticancer Agents as Potent Akt Inhibitors. Molecules 23:6, pages 1318.
Crossref
Crossref
Mohd. Imran Ansari & Suroor Ahmad Khan. (2017) Synthesis and antimicrobial activity of some novel quinoline-pyrazoline-based coumarinyl thiazole derivatives. Medicinal Chemistry Research 26:7, pages 1481-1496.
Crossref
Crossref
S. R. K. Battula, V. P. Rama Kishore Putta, G. V. Subbareddy, I. E. Chakravarthy & V. Saravanan. (2017) A divergent and metal free synthesis of sulfoximine tethered imidazoles, imidazopyridines, imidazothiazoles, imidazobenzothiazines, thiazoles and selenazoles. Organic & Biomolecular Chemistry 15:17, pages 3742-3755.
Crossref
Crossref
Jeffrey Y. W. Mak, Weijun Xu & David P. Fairlie. 2017. Peptidomimetics I. Peptidomimetics I
235
266
.