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Sphingosine 1-phosphate receptor 1 agonists: a patent review (2013-2015)

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Pages 455-470 | Received 15 Dec 2015, Accepted 18 Feb 2016, Published online: 15 Mar 2016

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Élise Pépin, Tim Jalinier, Guillaume L. Lemieux, Guy Massicotte & Michel Cyr. (2020) Sphingosine-1-Phosphate Receptors Modulators Decrease Signs of Neuroinflammation and Prevent Parkinson’s Disease Symptoms in the 1-Methyl-4-Phenyl-1,2,3,6-Tetrahydropyridine Mouse Model. Frontiers in Pharmacology 11.
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Junfei Jin, Zhongyang Lu, Yanchun Li, Ji Hyun Ru, Maria F Lopes-Virella & Yan Huang. (2018) LPS and palmitate synergistically stimulate sphingosine kinase 1 and increase sphingosine 1 phosphate in RAW264.7 macrophages. Journal of Leukocyte Biology 104:4, pages 843-853.
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Giancarlo Comi, Hans-Peter Hartung, Rajesh Bakshi, Ian M. Williams & Heinz Wiendl. (2017) Benefit–Risk Profile of Sphingosine-1-Phosphate Receptor Modulators in Relapsing and Secondary Progressive Multiple Sclerosis. Drugs 77:16, pages 1755-1768.
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Ambra Vestri, Federica Pierucci, Alessia Frati, Lucia Monaco & Elisabetta Meacci. (2017) Sphingosine 1-Phosphate Receptors: Do They Have a Therapeutic Potential in Cardiac Fibrosis?. Frontiers in Pharmacology 8.
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Frédéric St-Cyr Giguère, Suzanne Attiori Essis, Laure Chagniel, Marc Germain, Michel Cyr & Guy Massicotte. (2017) The sphingosine-1-phosphate receptor 1 agonist SEW2871 reduces Tau-Ser262 phosphorylation in rat hippocampal slices. Brain Research 1658, pages 51-59.
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Linda Bendall. (2016) Extracellular molecules in hematopoietic stem cell mobilisation. International Journal of Hematology 105:2, pages 118-128.
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