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The therapeutic potential of GPR119 agonists for type 2 diabetes

, PhD & , PhD
Pages 321-328 | Published online: 03 Feb 2012

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Huilan Li, Yuanying Fang, Shuchun Guo & Zunhua Yang. (2021) GPR119 agonists for the treatment of type 2 diabetes: an updated patent review (2014-present). Expert Opinion on Therapeutic Patents 31:9, pages 795-808.
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André J. Scheen. (2016) Investigational insulin secretagogues for type 2 diabetes. Expert Opinion on Investigational Drugs 25:4, pages 405-422.
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Joseph W. Polli, Elizabeth Hussey, Mark Bush, Grant Generaux, Glenn Smith, David Collins, Susan McMullen, Nancy Turner & Derek J. Nunez. (2013) Evaluation of drug interactions of GSK1292263 (a GPR119 agonist) with statins: from in vitro data to clinical study design. Xenobiotica 43:6, pages 498-508.
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Lauren M Cornall, Michael L Mathai, Deanne H Hryciw & Andrew J McAinch. (2013) Is GPR119 agonism an appropriate treatment modality for the safe amelioration of metabolic diseases?. Expert Opinion on Investigational Drugs 22:4, pages 487-498.
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Anders Tengholm. (2012) Cyclic AMP dynamics in the pancreatic β-cell. Upsala Journal of Medical Sciences 117:4, pages 355-369.
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Anuradha Mehra, Rekha Sangwan, Aryan Mehra, Shivani Sharma, Pankaj Wadhwa & Amit Mittal. (2023) Therapeutic charisma of imidazo [2,1-b] [1,3,4]-thiadiazole analogues: a patent review. Pharmaceutical Patent Analyst.
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Zekun Lyu, Min Zhao, Patricio Atanes & Shanta Jean Persaud. (2022) Quantification of changes in human islet G protein‐coupled receptor mRNA expression in obesity. Diabetic Medicine 39:12.
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Jianan Zhao, Yu Zhao, Yiyang Hu & Jinghua Peng. (2021) Targeting the GPR119/incretin axis: a promising new therapy for metabolic-associated fatty liver disease. Cellular & Molecular Biology Letters 26:1.
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Silvano Paternoster, Peter V. Simpson, Elena Kokh, Hüsün Sheyma Kizilkaya, Mette Marie Rosenkilde, Ricardo L. Mancera, Damien J. Keating, Massimiliano Massi & Marco Falasca. (2021) Pharmacological and structure-activity relationship studies of oleoyl-lysophosphatidylinositol synthetic mimetics. Pharmacological Research 172, pages 105822.
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Ajay Manaithiya, Ozair Alam, Vrinda Sharma, Mohd. Javed Naim, Shruti Mittal & Imran A Khan. (2021) GPR119 agonists: Novel therapeutic agents for type 2 diabetes mellitus. Bioorganic Chemistry 113, pages 104998.
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Prateek Sharma, Sukhbir Singh, Vinay Thakur, Neelam Sharma & Ajmer Singh Grewal. (2021) Novel and emerging therapeutic drug targets for management of type 2 Diabetes Mellitus. Obesity Medicine 23, pages 100329.
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Amit Gupta, Tapan Behl, Aayush Sehgal, Shaveta Bhardwaj, Sukhbir Singh, Neelam Sharma & Abdul Hafeez. (2021) Exploring the recent molecular targets for diabetes and associated complications. Molecular Biology Reports 48:3, pages 2863-2879.
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Alain Veilleux, Vincenzo Di Marzo & Cristoforo Silvestri. (2019) The Expanded Endocannabinoid System/Endocannabinoidome as a Potential Target for Treating Diabetes Mellitus. Current Diabetes Reports 19:11.
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