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Drug Evaluation

Efavirenz: a review

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Pages 851-871 | Published online: 11 Apr 2007

Keep up to date with the latest research on this topic with citation updates for this article.

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Rohini Kharwade, Nilesh Mahajan, Sachin More, Amol Warokar, Sachin Mendhi, Akshay Dhobley & Devendra Palve. (2023) Effect of PEGylation on drug uptake, biodistribution, and tissue toxicity of efavirenz–ritonavir loaded PAMAM G4 dendrimers. Pharmaceutical Development and Technology 28:2, pages 200-218.
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Chang Hoon Lee, Francesco Franchi & Dominick J. Angiolillo. (2020) Clopidogrel drug interactions: a review of the evidence and clinical implications. Expert Opinion on Drug Metabolism & Toxicology 16:11, pages 1079-1096.
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Liting Yan, Fengting Yu, Huimin Zhang, Hongxin Zhao, Linghang Wang, Zaiyan Liang, Xia Zhang, Liang Wu, Hongyuan Liang, Siyuan Yang, Yunxia Tang & Fujie Zhang. (2020) Transmitted and Acquired HIV-1 Drug Resistance from a Family: A Case Study. Infection and Drug Resistance 13, pages 3763-3770.
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Yali Wang, Erik De Clercq & Guangdi Li. (2019) Current and emerging non-nucleoside reverse transcriptase inhibitors (NNRTIs) for HIV-1 treatment. Expert Opinion on Drug Metabolism & Toxicology 15:10, pages 813-829.
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Tomohiko Ichikawa, Hirofumi Tsujino, Takahiro Miki, Masaya Kobayashi, Chiaki Matsubara, Sara Miyata, Taku Yamashita, Kohei Takeshita, Yasushige Yonezawa & Tadayuki Uno. (2018) Allosteric activation of cytochrome P450 3A4 by efavirenz facilitates midazolam binding. Xenobiotica 48:12, pages 1227-1236.
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Evelyn Rodríguez-Estrada, Mónica Fernández-Sánchez, Jairo Muñoz-Delgado, Ana Fresan-Orellana & Gustavo Reyes-Terán. (2016) Sleep and rest activity measured by wrist actigraphy in an HIV-infected patient with Steven–Johnson syndrome. Biological Rhythm Research 47:1, pages 1-6.
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Beatriz Larru, Jessica Eby & Elizabeth D Lowenthal. (2014) Antiretroviral treatment in HIV-1 infected pediatric patients: focus on efavirenz. Pediatric Health, Medicine and Therapeutics 5, pages 29-42.
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Peter Derek Christian Leutscher, Chalotte Stecher, Merete Storgaard & Carsten Schade Larsen. (2013) Discontinuation of efavirenz therapy in HIV patients due to neuropsychiatric adverse effects. Scandinavian Journal of Infectious Diseases 45:8, pages 645-651.
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Brookie M Best & Miguel Goicoechea. (2008) Efavirenz – Still First-line King?. Expert Opinion on Drug Metabolism & Toxicology 4:7, pages 965-972.
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