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Histone modification enzymes: novel targets for cancer drugs

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Pages 135-154 | Published online: 02 Mar 2005

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Laura Vanagas, Victoria Jeffers, Silvina S Bogado, Maria C Dalmasso, William J Sullivan$suffix/text()$suffix/text() & Sergio O Angel. (2012) Toxoplasma histone acetylation remodelers as novel drug targets. Expert Review of Anti-infective Therapy 10:10, pages 1189-1201.
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Sutapa Mukherjee, Ruma Sarkar, Jaydip Biswas & Madhumita Roy. (2012) Curcumin Inhibits Histone Deacetylase Leading to Cell Cycle Arrest and Apoptosis via Upregulation of p21 in Breast Cancer Cell Lines. International Journal of Green Nanotechnology 4:2, pages 183-197.
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Rodney F Minchin & Shu Yang. (2010) Endosomal disruptors in non-viral gene delivery. Expert Opinion on Drug Delivery 7:3, pages 331-339.
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Steve Price & Hazel J Dyke. (2007) Histone deacetylase inhibitors. Expert Opinion on Therapeutic Patents 17:7, pages 745-765.
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P. Workman. (2004) Drug Discovery Strategies: Technologies to Accelerate Translation from Target to Drug. Journal of Chemotherapy 16:sup4, pages 13-15.
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Articles from other publishers (64)

Joanna Szczepanek & Andrzej Tretyn. (2023) MicroRNA-Mediated Regulation of Histone-Modifying Enzymes in Cancer: Mechanisms and Therapeutic Implications. Biomolecules 13:11, pages 1590.
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Ying Li, Lei Ding, Shuang Ren, Wen Zhang & Guo-Wu Rao. (2023) Protein Lysine Methyltransferases Inhibitors. Current Medicinal Chemistry 30:27, pages 3060-3089.
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Muhammad Nabeel Asim, Muhammad Ali Ibrahim, Muhammad Imran Malik, Imran Razzak, Andreas Dengel & Sheraz Ahmed. (2022) Histone-Net: a multi-paradigm computational framework for histone occupancy and modification prediction. Complex & Intelligent Systems 9:1, pages 399-419.
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Michela Giuliano, Claudia Pellerito, Adriana Celesia, Tiziana Fiore & Sonia Emanuele. (2021) Tributyltin(IV) Butyrate: A Novel Epigenetic Modifier with ER Stress- and Apoptosis-Inducing Properties in Colon Cancer Cells. Molecules 26:16, pages 5010.
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Skye Hsin-Hsien Yeh, Ming Hsien Lin, I. I. Leo Garcia Flores, Uday Mukhopadhyay, Danial Young, Kazuma Ogawa, Jeong-Hwan Jeong, William Tong, Juri G. Gelovani & Nobuyoshi Fukumitsu. (2021) In Vivo Evaluation of the Combined Anticancer Effects of Cisplatin and SAHA in Nonsmall Cell Lung Carcinoma Using [18F]FAHA and [18F]FDG PET/CT Imaging. Molecular Imaging 2021, pages 1-11.
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Mohsin Nawaz, Irfan Malik, Mudassar Hameed, Zulfiqar Hussain Kuthu & Jinlin Zhou. (2020) Modifications of histones in parasites as drug targets. Veterinary Parasitology 278, pages 109029.
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Kathryn Hill & Tania L. Roth. 2016. Developmental Psychopathology. Developmental Psychopathology 1 26 .
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Yang Cai, Xiang Yan, Guoqing Zhang, Weihong Zhao & Shunchang Jiao. (2015) The predictive value of ERCC1 and p53 for the effect of panobinostat and cisplatin combination treatment in NSCLC. Oncotarget 6:22, pages 18997-19005.
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Martin Lübke, Manfred Jung & Günter Haufe. (2013) New histone deacetylase inhibitors based on 4-fluoro-2-amino acid esters: Synthesis and activity. Journal of Fluorine Chemistry 152, pages 144-156.
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Santosh Kumar & Souvik Maiti. (2013) Effect of different arginine methylations on the thermodynamics of Tat peptide binding to HIV-1 TAR RNA. Biochimie 95:7, pages 1422-1431.
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Jatinder Goyal & Ronald Rodriguez. (2013) Evidence from clinical trials for the use of valproic acid in solid tumors: focus on prostate cancer. Clinical Investigation 3:5, pages 467-478.
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Giuseppe GianniniWalter Cabri, Caterina Fattorusso & Manuela Rodriquez. (2012) Histone deacetylase inhibitors in the treatment of cancer: overview and perspectives. Future Medicinal Chemistry 4:11, pages 1439-1460.
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Paul V. Licciardi & Tom C. Karagiannis. (2012) Regulation of Immune Responses by Histone Deacetylase Inhibitors. ISRN Hematology 2012, pages 1-10.
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