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Targeting topoisomerase I: molecular mechanisms and cellular determinants of response to topoisomerase I inhibitors

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Pages 1243-1256 | Published online: 09 Sep 2008

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Moustafa M. Madkour, Wafaa S. Ramadan, Ekram Saleh & Raafat El-Awady. (2023) Epigenetic modulations in cancer: predictive biomarkers and potential targets for overcoming the resistance to topoisomerase I inhibitors. Annals of Medicine 55:1.
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Doddabasappa Talimarada, Akanksha Sharma & Harish Holla. (2023) Identification of dual binding mode of Orthodiffenes towards human topoisomerase-I and α-tubulin: exploring the potential role in anti-cancer activity via in silico study. Journal of Biomolecular Structure and Dynamics 41:7, pages 2789-2803.
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Eman R. El-Sharkawy & Khaled Mahmoud. (2016) Cytotoxity of two new coumarin derivatives isolated from Launaea mucronata. Natural Product Research 30:4, pages 394-398.
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Serena Basili & Stefano Moro. (2009) Novel camptothecin derivatives as topoisomerase I inhibitors. Expert Opinion on Therapeutic Patents 19:5, pages 555-574.
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