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Tyrosine kinase inhibitors as modulators of ATP binding cassette multidrug transporters: substrates, chemosensitizers or inducers of acquired multidrug resistance?

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Pages 623-642 | Published online: 17 Mar 2011

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Piyush Bugde, Riya Biswas, Fabrice Merien, Jun Lu, Dong-Xu Liu, Mingwei Chen, Shufeng Zhou & Yan Li. (2017) The therapeutic potential of targeting ABC transporters to combat multi-drug resistance. Expert Opinion on Therapeutic Targets 21:5, pages 511-530.
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Claudia Maria Hattinger, Marilù Fanelli, Elisa Tavanti, Serena Vella, Stefano Ferrari, Piero Picci & Massimo Serra. (2015) Advances in emerging drugs for osteosarcoma. Expert Opinion on Emerging Drugs 20:3, pages 495-514.
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Camille Tlemsani, Olivier Huillard, Jennifer Arrondeau, Pascaline Boudou-Rouquette, Anatole Cessot, Benoit Blanchet, Audrey Thomas-Schoemann, Romain Coriat, Jean-Philippe Durand, Julie Giroux, Jérôme Alexandre & François Goldwasser. (2015) Effect of glucuronidation on transport and tissue accumulation of tyrosine kinase inhibitors: consequences for the clinical management of sorafenib and regorafenib. Expert Opinion on Drug Metabolism & Toxicology 11:5, pages 785-794.
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