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Autoradiography: high-resolution molecular imaging in pharmaceutical discovery and development

Pages 503-514 | Published online: 14 May 2007

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Mario Pellegatti. (2012) Preclinical in vivo ADME studies in drug development: a critical review. Expert Opinion on Drug Metabolism & Toxicology 8:2, pages 161-172.
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Eleanor Q. Blatherwick, Gary J. Van Berkel, Kathryn Pickup, Maria K. Johansson, Marie-Eve Beaudoin, Roderic O. Cole, Jennifer M. Day, Suzanne Iverson, Ian D. Wilson, James H. Scrivens & Daniel J. Weston. (2011) Utility of spatially-resolved atmospheric pressure surface sampling and ionization techniques as alternatives to mass spectrometric imaging (MSI) in drug metabolism. Xenobiotica 41:8, pages 720-734.
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Mario Pellegatti & Sabrina Pagliarusco. (2011) Drug and metabolite concentrations in tissues in relationship to tissue adverse findings: a review. Expert Opinion on Drug Metabolism & Toxicology 7:2, pages 137-146.
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Articles from other publishers (36)

Lu Peng, Benabdallah Nadia, Jiang Wen, Brian W. Simons, Zhang Hanwen, Robert F. Hobbs, Ulmert David, Brian C. Baumann, Russell K. Pachynski, Abhinav K. Jha & Daniel L.J. Thorek. (2022) Blind Image Restoration Enhances Digital Autoradiographic Imaging of Radiopharmaceutical Tissue Distribution. Journal of Nuclear Medicine 63:4, pages 591-597.
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Conor L. Evans, Maiko Hermsmeier, Akira Yamamoto & Kin F. Chan. (2020) Visualizing topical drug uptake with conventional fluorescence microscopy and deep learning. Biomedical Optics Express 11:12, pages 6864.
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Youssouf Djibril Soubaneh, Emilien Pelletier, Isabelle Desbiens & Claude Rouleau. (2019) Radiolabeling of amide functionalized multi-walled carbon nanotubes for bioaccumulation study in fish bone using whole-body autoradiography. Environmental Science and Pollution Research 27:4, pages 3756-3767.
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Caroline Bouter & Yvonne Bouter. (2019) 18F-FDG-PET in Mouse Models of Alzheimer's Disease. Frontiers in Medicine 6.
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Christopher A.G. Kalnins, Nigel A. Spooner, Michael J.P. Clarke & David Ottaway. (2019) Alpha particle autoradiography for high spatial resolution mapping of radionuclides. Journal of Environmental Radioactivity 197, pages 9-15.
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Jonathan Vigne, James Thackeray, Jeroen Essers, Marcus Makowski, Zoreh Varasteh, Adelina Curaj, Angelos Karlas, Emmanuel Canet-Soulas, Willem Mulder, Fabian Kiessling, Michael Schäfers, René Botnar, Moritz Wildgruber & Fabien Hyafil. (2018) Current and Emerging Preclinical Approaches for Imaging-Based Characterization of Atherosclerosis. Molecular Imaging and Biology 20:6, pages 869-887.
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Tashi Parsons-Davis, Kim Knight, Marc Fitzgerald, Gary Stone, Lee Caldeira, Christina Ramon & Michael Kristo. (2018) Application of modern autoradiography to nuclear forensic analysis. Forensic Science International 286, pages 223-232.
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Jens Atzrodt, Volker Derdau, William J. Kerr & Marc Reid. (2018) Deuterium- and Tritium-Labelled Compounds: Applications in the Life Sciences. Angewandte Chemie International Edition 57:7, pages 1758-1784.
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Jens Atzrodt, Volker Derdau, William J. Kerr & Marc Reid. (2018) Deuterium- und tritiummarkierte Verbindungen: Anwendungen in den modernen Biowissenschaften. Angewandte Chemie 130:7, pages 1774-1802.
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Yijun Ding, Luca Caucci & Harrison H. Barrett. (2017) Null functions in three-dimensional imaging of alpha and beta particles. Scientific Reports 7:1.
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Yong-il KimJin Chul PaengGi Jeong CheonKeon Wook KangDong Soo LeeJune-Key Chung. (2017) Discrepancy Between Tumor Antigen Distribution and Radiolabeled Antibody Binding in a Nude Mouse Xenograft Model of Human Melanoma. Cancer Biotherapy and Radiopharmaceuticals 32:3, pages 83-89.
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Randall W. Moreadith, Tacey X. Viegas, Michael D. Bentley, J. Milton Harris, Zhihao Fang, Kunsang Yoon, Bekir Dizman, Rebecca Weimer, Brendan P. Rae, Xiuling Li, Christoph Rader, David Standaert & Warren Olanow. (2017) Clinical development of a poly(2-oxazoline) (POZ) polymer therapeutic for the treatment of Parkinson’s disease – Proof of concept of POZ as a versatile polymer platform for drug development in multiple therapeutic indications. European Polymer Journal 88, pages 524-552.
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L. Gutiérrez, G. Stepien, L. Gutiérrez, M. Pérez-Hernández, J. Pardo, J. Pardo, V. Grazú & J.M. de la Fuente. 2017. Comprehensive Medicinal Chemistry III. Comprehensive Medicinal Chemistry III 264 295 .
Mônica Siqueira Ferreira, Diogo Noin de Oliveira, Caroline Costa Mesquita, Ana Paula de Lima Barbosa, Gabriel Forato Anhê & Rodrigo Ramos Catharino. (2016) MALDI-MSI: a fast and reliable method for direct melatonin quantification in biological fluids. Journal of Analytical Science and Technology 7:1.
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Gordon J. Dear & Angus N. R. Nedderman. 2016. Metabolite Safety in Drug Development. Metabolite Safety in Drug Development 17 43 .
Richard J.A. Goodwin, Anna Nilsson, C. Logan Mackay, John G. Swales, Maria K. Johansson, Martin Billger, Per E. Andrén & Suzanne L. Iverson. (2016) Exemplifying the Screening Power of Mass Spectrometry Imaging over Label-Based Technologies for Simultaneous Monitoring of Drug and Metabolite Distributions in Tissue Sections. SLAS Discovery 21:2, pages 187-193.
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Thierry Flandre, Sarah Taplin, Stewart Jones & Peter Lloyd. 2010. Pharmaceutical Sciences Encyclopedia. Pharmaceutical Sciences Encyclopedia 1 14 .
D F Cobice, R J A Goodwin, P E Andren, A Nilsson, C L Mackay & R Andrew. (2015) Future technology insight: mass spectrometry imaging as a tool in drug research and development. British Journal of Pharmacology 172:13, pages 3266-3283.
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Mônica Siqueira Ferreira, Rosimeire Nunes de Oliveira, Diogo Noin de Oliveira, Cibele Zanardi Esteves, Silmara Marques Allegretti & Rodrigo Ramos Catharino. (2015) Revealing praziquantel molecular targets using mass spectrometry imaging: an expeditious approach applied to Schistosoma mansoni. International Journal for Parasitology 45:6, pages 385-391.
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Eric G. Solon. (2015) Autoradiography techniques and quantification of drug distribution. Cell and Tissue Research 360:1, pages 87-107.
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Philipp Uhl, Gert Fricker, Uwe Haberkorn & Walter Mier. (2015) Radionuclides in drug development. Drug Discovery Today 20:2, pages 198-208.
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Mônica Siqueira Ferreira, Diogo Noin de Oliveira, Rosimeire Nunes de Oliveira, Silmara Marques Allegretti & Rodrigo Ramos Catharino. (2014) Screening the life cycle of Schistosoma mansoni using high-resolution mass spectrometry. Analytica Chimica Acta 845, pages 62-69.
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Achim Buck & Axel Walch. (2014) In situ drug and metabolite analysis in biological and clinical research by MALDI MS imaging . Bioanalysis 6:9, pages 1241-1253.
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Lívia Riberti Rodrigues, Diogo Noin de Oliveira, Mônica Siqueira Ferreira & Rodrigo Ramos Catharino. (2014) In situ assessment of atorvastatin impurity using MALDI mass spectrometry imaging (MALDI-MSI). Analytica Chimica Acta 818, pages 32-38.
Crossref
Eric G. Solon & Brian R. Moyer. 2014. Pharmaco-Imaging in Drug and Biologics Development. Pharmaco-Imaging in Drug and Biologics Development 133 185 .
Brian R. Moyer. 2014. Pharmaco-Imaging in Drug and Biologics Development. Pharmaco-Imaging in Drug and Biologics Development 1 43 .
Mônica Siqueira Ferreira, Diogo Noin de Oliveira, Rosimeire Nunes de Oliveira, Silmara Marques Allegretti, Aníbal Eugênio Vercesi & Rodrigo Ramos Catharino. (2014) Mass spectrometry imaging: a new vision in differentiating Schistosoma mansoni strains . Journal of Mass Spectrometry 49:1, pages 86-92.
Crossref
Diogo de Oliveira, Sabrina de Bona Sartor, Mônica Ferreira & Rodrigo Catharino. (2013) Cosmetic Analysis Using Matrix-Assisted Laser Desorption/Ionization Mass Spectrometry Imaging (MALDI-MSI). Materials 6:3, pages 1000-1010.
Crossref
Eric G. Solon. (2012) Use of Radioactive Compounds and Autoradiography to Determine Drug Tissue Distribution. Chemical Research in Toxicology 25:3, pages 543-555.
Crossref
Alexander V. LyubimovEric G. Solon. 2011. Encyclopedia of Drug Metabolism and Interactions. Encyclopedia of Drug Metabolism and Interactions 1 34 .
Stephen Castellino, M Reid Groseclose & David Wagner. (2011) MALDI imaging mass spectrometry: bridging biology and chemistry in drug development. Bioanalysis 3:21, pages 2427-2441.
Crossref
Xiao Ren, Tobias Paehler, Manfred Zimmer, Zuyu Guo, Patricia Zane & Gary T Emmons. (2010) Impact of various factors on radioactivity distribution in different DBS papers. Bioanalysis 2:8, pages 1469-1475.
Crossref
Eric G. Solon, Alain Schweitzer, Markus Stoeckli & Brendan Prideaux. (2009) Autoradiography, MALDI-MS, and SIMS-MS Imaging in Pharmaceutical Discovery and Development. The AAPS Journal 12:1, pages 11-26.
Crossref
Brendan Prideaux, Dieter Staab & Markus Stoeckli. 2010. Mass Spectrometry Imaging. Mass Spectrometry Imaging 405 413 .
Stefan Balaz. (2009) Modeling Kinetics of Subcellular Disposition of Chemicals. Chemical Reviews 109:5, pages 1793-1899.
Crossref
Brian R MoyerJohn A Barrett. (2009) Biomarkers and imaging: physics and chemistry for noninvasive analyses. Bioanalysis 1:2, pages 321-356.
Crossref

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