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Expert Opinion on Drug Discovery Volume 10, 2015 - Issue 11
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Drug Discovery Case History

The preclinical discovery and development of dolutegravir for the treatment of HIV

Fabrice BaillyUniversite de lille, Pharmaceutical and Biological Sciences, 3, rue du Pr Laguesse, BP83, Lille 59006, France+33 0 3 62 28 36 94; [email protected];Jean-Pierre Aubert Research Center UMR-S1172 INSERM, Onco and Neurochemistry team, 3, rue du Pr Laguesse, BP83, Lille 59006, France
(Faculty of Pharmaceutical and Biological Sciences) &
Philippe CotelleUniversite de lille, Pharmaceutical and Biological Sciences, 3, rue du Pr Laguesse, BP83, Lille 59006, France+33 0 3 62 28 36 94; [email protected];Jean-Pierre Aubert Research Center UMR-S1172 INSERM, Onco and Neurochemistry team, 3, rue du Pr Laguesse, BP83, Lille 59006, France
(Faculty of Pharmaceutical and Biological Sciences)
Pages 1243-1253 | Published online: 07 Sep 2015

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Yoshiyuki Taoda, Shuichi Sugiyama & Takahiro Seki. (2023) New designs for HIV-1 integrase inhibitors: a patent review (2018-present). Expert Opinion on Therapeutic Patents 33:1, pages 51-66.
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Articles from other publishers (9)

Ila M. Sarode & Anil B. Jindal. (2022) Current status of dolutegravir delivery systems for the treatment of HIV-1 infection. Journal of Drug Delivery Science and Technology 76, pages 103802.
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Sanjay Kumar, Geethu S Kumar, Subhrangsu Sundar Maitra, Petr Malý, Shiv Bharadwaj, Pradeep Sharma & Vivek Dhar Dwivedi. (2022) Viral informatics: bioinformatics-based solution for managing viral infections. Briefings in Bioinformatics 23:5.
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Nadia M. Ikumi, Dilly Anumba & Mushi Matjila. (2022) Pharmacokinetics and placental transfer of dolutegravir in pregnancy. Journal of Antimicrobial Chemotherapy 77:2, pages 283-289.
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Victor T. Sabe, Thandokuhle Ntombela, Lindiwe A. Jhamba, Glenn E.M. Maguire, Thavendran Govender, Tricia Naicker & Hendrik G. Kruger. (2021) Current trends in computer aided drug design and a highlight of drugs discovered via computational techniques: A review. European Journal of Medicinal Chemistry 224, pages 113705.
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Lei Wang, Tiffany C. Edwards, Rajkumar Lalji Sahani, Jiashu Xie, Hideki Aihara, Robert J. Geraghty & Zhengqiang Wang. (2021) Metal binding 6-arylthio-3-hydroxypyrimidine-2,4-diones inhibited human cytomegalovirus by targeting the pUL89 endonuclease of the terminase complex. European Journal of Medicinal Chemistry 222, pages 113640.
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Benjamin E. Blass. 2021. Basic Principles of Drug Discovery and Development. Basic Principles of Drug Discovery and Development 1 41 .
Joseph M. Fortunak, Ji Zhang, Frederick E. NytkoIIIIII & Tiffany N. Ellison. 2018. Green Techniques for Organic Synthesis and Medicinal Chemistry. Green Techniques for Organic Synthesis and Medicinal Chemistry 621 647 .
Pratiq A. Patel, Nina Kvaratskhelia, Yara Mansour, Janet Antwi, Lei Feng, Pratibha Koneru, Mathew J. Kobe, Nivedita Jena, Guqin Shi, Mosaad S. Mohamed, Chenglong Li, Jacques J. Kessl & James R. Fuchs. (2016) Indole-based allosteric inhibitors of HIV-1 integrase. Bioorganic & Medicinal Chemistry Letters 26:19, pages 4748-4752.
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Muriel Billamboz, Virginie Suchaud, Fabrice Bailly, Cedric Lion, Marie-Line Andréola, Frauke Christ, Zeger Debyser & Philippe Cotelle. (2016) 2-hydroxyisoquinoline-1,3(2 H ,4 H )-diones (HIDs) as human immunodeficiency virus type 1 integrase inhibitors: Influence of the alkylcarboxamide substitution of position 4. European Journal of Medicinal Chemistry 117, pages 256-268.
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