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Original Research

Nanoparticulate formulations of mithramycin analogs for enhanced cytotoxicity

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Pages 2757-2767 | Published online: 08 Nov 2011

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Óscar Estupiñán, Enrique Niza, Iván Bravo, Verónica Rey, Juan Tornín, Borja Gallego, Pilar Clemente-Casares, Francisco Moris, Alberto Ocaña, Verónica Blanco-Lorenzo, Mar Rodríguez-Santamaría, Aitana Vallina-Álvarez, M. Victoria González, Aida Rodríguez, Daniel Hermida-Merino, Carlos Alonso-Moreno & René Rodríguez. (2021) Mithramycin delivery systems to develop effective therapies in sarcomas. Journal of Nanobiotechnology 19:1.
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Óscar Estupiñán, Claudia Rendueles, Paula Suárez, Verónica Rey, Dzohara Murillo, Francisco Morís, Gemma Gutiérrez, María del Carmen Blanco-López, María Matos & René Rodríguez. (2021) Nano-Encapsulation of Mithramycin in Transfersomes and Polymeric Micelles for the Treatment of Sarcomas. Journal of Clinical Medicine 10:7, pages 1358.
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David Schweer, J. Robert McCorkle, Jurgen Rohr, Oleg V. Tsodikov, Frederick Ueland & Jill Kolesar. (2021) Mithramycin and Analogs for Overcoming Cisplatin Resistance in Ovarian Cancer. Biomedicines 9:1, pages 70.
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Yang Liu, Joseph M. Eckenrode, Yinan Zhang, Jianjun Zhang, Reiya C. Hayden, Annet Kyomuhangi, Larissa V. Ponomareva, Zheng Cui, Jürgen Rohr, Oleg V. Tsodikov, Steven G. Van Lanen, Khaled A. Shaaban, Markos Leggas & Jon S. Thorson. (2020) Mithramycin 2′-Oximes with Improved Selectivity, Pharmacokinetics, and Ewing Sarcoma Antitumor Efficacy. Journal of Medicinal Chemistry 63:22, pages 14067-14086.
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Stevi Weidenbach, Caixia Hou, Jhong-Min Chen, Oleg V. Tsodikov & Jürgen Rohr. (2016) Dimerization and DNA recognition rules of mithramycin and its analogues. Journal of Inorganic Biochemistry 156, pages 40-47.
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Tsz Chung Lai, Hyunah Cho & Glen S. Kwon. (2014) Reversibly core cross-linked polymeric micelles with pH- and reduction-sensitivities: effects of cross-linking degree on particle stability, drug release kinetics, and anti-tumor efficacy. Polym. Chem. 5:5, pages 1650-1661.
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Daniel Scott, Jhong-Min Chen, Younsoo Bae & Jürgen Rohr. (2013) Semi-Synthetic Mithramycin SA Derivatives with Improved AntiCancer Activity. Chemical Biology & Drug Design 81:5, pages 615-624.
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Mo Dan, Daniel F. Scott, Peter A. Hardy, Robert J. Wydra, J. Zach Hilt, Robert A. Yokel & Younsoo Bae. (2012) Block Copolymer Cross-Linked Nanoassemblies Improve Particle Stability and Biocompatibility of Superparamagnetic Iron Oxide Nanoparticles. Pharmaceutical Research 30:2, pages 552-561.
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Hyun Jin Lee & Younsoo Bae. (2012) Pharmaceutical Differences Between Block Copolymer Self-Assembled and Cross-Linked Nanoassemblies as Carriers for Tunable Drug Release. Pharmaceutical Research 30:2, pages 478-488.
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