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Review

Prolylcarboxypeptidase (PRCP) as a new target for obesity treatment

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Pages 67-78 | Published online: 27 Sep 2022

Keep up to date with the latest research on this topic with citation updates for this article.

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Thomas H. Graham. (2017) Prolylcarboxypeptidase (PrCP) inhibitors and the therapeutic uses thereof: a patent review. Expert Opinion on Therapeutic Patents 27:10, pages 1077-1088.
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Articles from other publishers (10)

Sandrine Mignon-Grasteau, Nicole Rideau, Irène Gabriel, Céline Chantry-Darmon, Marie-Yvonne Boscher, Nadine Sellier, Marie Chabault, Elisabeth Le Bihan-Duval & Agnès Narcy. (2015) Detection of QTL controlling feed efficiency and excretion in chickens fed a wheat-based diet. Genetics Selection Evolution 47:1.
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Thomas H. Graham, Min Shu, Andreas Verras, Qing Chen, Margarita Garcia-Calvo, Xiaohua Li, JeanMarie Lisnock, Xinchun Tong, Elaine C. Tung, Judyann Wiltsie, Jeffrey J. Hale, Shirly Pinto & Dong-Ming Shen. (2014) Pyrazoles as non-classical bioisosteres in prolylcarboxypeptidase (PrCP) inhibitors. Bioorganic & Medicinal Chemistry Letters 24:7, pages 1657-1660.
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Irina A. Goptar, Dmitry A. Shagin, Irina A. Shagina, Elena S. Mudrik, Yulia A. Smirnova, Dmitry P. Zhuzhikov, Mikhail A. Belozersky, Yakov E. Dunaevsky, Brenda Oppert, Irina Yu. Filippova & Elena N. Elpidina. (2013) A digestive prolyl carboxypeptidase in Tenebrio molitor larvae. Insect Biochemistry and Molecular Biology 43:6, pages 501-509.
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Jin Kwon Jeong & Sabrina Diano. (2013) Prolyl carboxypeptidase and its inhibitors in metabolism. Trends in Endocrinology & Metabolism 24:2, pages 61-67.
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Sarah Chajkowski Scarry & John M. Rimoldi. 2013. 91 103 .
Thomas H. Graham, Wensheng Liu, Andreas Verras, Mikhail Reibarkh, Kelly Bleasby, Urmi R. Bhatt, Qing Chen, Margarita Garcia-Calvo, Wayne M. Geissler, Judith N. Gorski, Huaibing He, Michael E. Lassman, JeanMarie Lisnock, Xiaohua Li, Zhu Shen, Xinchun Tong, Elaine C. Tung, Judyann Wiltsie, Dan Xie, Suoyu Xu, Jianying Xiao, Jeffrey J. Hale, Shirly Pinto & Dong-Ming Shen. (2012) A new class of prolylcarboxypeptidase inhibitors, Part 2: The aminocyclopentanes. Bioorganic & Medicinal Chemistry Letters 22:8, pages 2818-2822.
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Thomas H. Graham, Wensheng Liu, Andreas Verras, Iyassu K. Sebhat, Yusheng Xiong, Kelly Bleasby, Urmi R. Bhatt, Qing Chen, Margarita Garcia-Calvo, Wayne M. Geissler, Judith N. Gorski, Huaibing He, Michael E. Lassman, JeanMarie Lisnock, Xiaohua Li, Zhu Shen, Xinchun Tong, Elaine C. Tung, Judyann Wiltsie, Jianying Xiao, Dan Xie, Suoyu Xu, Jeffrey J. Hale, Shirly Pinto & Dong-Ming Shen. (2012) A new class of prolylcarboxypeptidase inhibitors, Part 1: Discovery and evaluation. Bioorganic & Medicinal Chemistry Letters 22:8, pages 2811-2817.
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Zhicai Wu, Cangming Yang, Thomas H. Graham, Andreas Verras, Renee M. Chabin, Suoyu Xu, Xinchun Tong, Dan Xie, Mike E. Lassman, Urmi R. Bhatt, Margarita M. Garcia-Calvo, Zhu Shen, Qing Chen, Kelly Bleasby, Ranabir Sinharoy, Jeffrey J. Hale, James R. Tata, Shirly Pinto, Steven L. Colletti & Dong-Ming Shen. (2012) Discovery of aminoheterocycles as potent and brain penetrant prolylcarboxypeptidase inhibitors. Bioorganic & Medicinal Chemistry Letters 22:4, pages 1727-1730.
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Zhicai Wu, Cangming Yang, Yusheng Xiong, Zhe Feng, Matthew Lombardo, Andreas Verras, Renee M. Chabin, Suoyu Xu, Xinchun Tong, Dan Xie, Mike E. Lassman, Urmi R. Bhatt, Margarita M. Garcia-Calvo, Wayne Geissler, Zhu Shen, Qing Chen, Ranabir Sinharoy, Jeffrey J. Hale, James R. Tata, Shirly Pinto, Dong-Ming Shen & Steven L. Colletti. (2012) Discovery of a new class of potent prolylcarboxypeptidase inhibitors derived from alanine. Bioorganic & Medicinal Chemistry Letters 22:4, pages 1774-1778.
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Thomas H. Graham, Hong C. Shen, Wensheng Liu, Yusheng Xiong, Andreas Verras, Kelly Bleasby, Urmi R. Bhatt, Renee M. Chabin, Dunlu Chen, Qing Chen, Margarita Garcia-Calvo, Wayne M. Geissler, Huaibing He, Michael E. Lassman, Zhu Shen, Xinchun Tong, Elaine C. Tung, Dan Xie, Suoyu Xu, Steven L. Colletti, James R. Tata, Jeffrey J. Hale, Shirly Pinto & Dong-Ming Shen. (2012) The discovery of non-benzimidazole and brain-penetrant prolylcarboxypeptidase inhibitors. Bioorganic & Medicinal Chemistry Letters 22:1, pages 658-665.
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