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Original Article

Development of an oral formulation of omeprazole

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Pages 113-120 | Published online: 08 Jul 2009

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A. Riedel & C. S. Leopold. (2005) Degradation of Omeprazole Induced by Enteric Polymer Solutions and Aqueous Dispersions: HPLC Investigations. Drug Development and Industrial Pharmacy 31:2, pages 151-160.
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Chul Soon Yong, Jae-Hee Jung, Jong-Dal Rhee, Chong-Kook Kim & Han-Gon Choi. (2001) Physicochemical Characterization and Evaluation of Buccal Adhesive Tablets Containing Omeprazole. Drug Development and Industrial Pharmacy 27:5, pages 447-455.
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A. G. Davidson & A. McCallum. (1996) A Survey of the Stability of Omeprazole Products from 13 Countries. Drug Development and Industrial Pharmacy 22:12, pages 1173-1185.
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C. Cederberg, T. Andersson & I. Skånberg. (1989) Omeprazole: Pharmacokinetics and Metabolism in Man. Scandinavian Journal of Gastroenterology 24:sup166, pages 33-40.
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H. Larsson, H. Mattsson & E. Carlsson. (1988) Gastric Acid Antisecretory Effect of Two Different Dosage Forms of Omeprazole during Prolonged Oral Treatment in the Gastric Fistula Dog. Scandinavian Journal of Gastroenterology 23:8, pages 1013-1019.
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Articles from other publishers (62)

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Annika Elbe, Kathrin Isabelle Foerster, Antje Blank, Peter Rose, Jürgen Burhenne, Walter Emil Haefeli & Gerd Mikus. (2022) Evaluation of CYP2C19 activity using microdosed oral omeprazole in humans. European Journal of Clinical Pharmacology 78:6, pages 975-987.
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Ajinkya Trimukhe, Satish Rojekar, Pradeep R. Vavia & R.R. Deshmukh. (2021) Pulsed plasma surface modified omeprazole microparticles for delayed release application. Journal of Drug Delivery Science and Technology 66, pages 102905.
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Alireza Khatibi, Payam Zahedi, Hedayatollah Ghourchian & Atefe Sadeghi Lari. (2021) Development of microfluidic-based cellulose acetate phthalate nanoparticles containing omeprazole for antiulcer activity: In vitro and in vivo evaluations. European Polymer Journal 147, pages 110294.
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Federica Ronchi, Antonio Sereno, Maxime Paide, Pierre Sacré, George Guillaume, Vincent Stéphenne, Jonathan Goole & Karim Amighi. (2019) Development and evaluation of an omeprazole-based delayed-release liquid oral dosage form. International Journal of Pharmaceutics 567, pages 118416.
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Elena Puris, Markku Pasanen, Veli‐Pekka Ranta, Mikko Gynther, Aleksanteri Petsalo, Pirjo Käkelä, Ville Männistö & Jussi Pihlajamäki. (2019) Laparoscopic Roux‐en‐Y gastric bypass surgery influenced pharmacokinetics of several drugs given as a cocktail with the highest impact observed for CYP1A2, CYP2C8 and CYP2E1 substrates. Basic & Clinical Pharmacology & Toxicology.
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Andressa Veiga, Paulo R. Oliveira, Larissa S. Bernardi, Cassiana Mendes, Marcos A. S. Silva, Maximiliano S. Sangoi, Paulo R. Janissek & Fábio S. Murakami. (2017) Solid-state compatibility studies of a drug without melting point. Journal of Thermal Analysis and Calorimetry 131:3, pages 3201-3209.
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John Chung & Filippos Kesisoglou. (2018) Physiologically Based Oral Absorption Modelling to Study Gut-Level Drug Interactions. Journal of Pharmaceutical Sciences 107:1, pages 18-23.
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Mohammad Sofiqur Rahman, Naoko Yoshida, Hirohito Tsuboi, Tep Keila, Tey Sovannarith, Heng Bun Kiet, Eav Dararth, Theingi Zin, Tsuyoshi Tanimoto & Kazuko Kimura. (2017) Erroneous formulation of delayed-release omeprazole capsules: alert for importing countries. BMC Pharmacology and Toxicology 18:1.
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Ping Ren, Minglei Cui, Om Anand, Li Xia, Zhuojun J. Zhao, Dajun Sun, Trueman Sharp, Dale P. Conner, John Peters, Wenlei Jiang, Ethan Stier & Xiaojian Jiang. (2017) In vitro Approaches to Support Bioequivalence and Substitutability of Generic Proton Pump Inhibitors via Nasogastric Tube Administration. The AAPS Journal 19:6, pages 1593-1599.
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Jens Van Den Abeele, Jari Rubbens, Joachim Brouwers & Patrick Augustijns. (2017) The dynamic gastric environment and its impact on drug and formulation behaviour. European Journal of Pharmaceutical Sciences 96, pages 207-231.
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Ching Kim Tye, Zhanbin Wang, Randy C. Dockens, Blisse Vakkalagadda, Chunlei Wang, Yingru Zhang, Ching Chiang Su & Michael J. Hageman. (2016) Pre-absorption physicochemical compatibility assessment of 8-drug metabolic cocktail. International Journal of Pharmaceutics 514:2, pages 364-373.
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Yohei Kosugi, Syunsuke Yamamoto, Noriyasu Sano, Atsutoshi Furuta, Tomoko Igari, Yasushi Fujioka & Nobuyuki Amano. (2015) Evaluation of Acid Tolerance of Drugs Using Rats and Dogs Controlled for Gastric Acid Secretion. Journal of Pharmaceutical Sciences 104:9, pages 2887-2893.
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Vishnu Dutt Sharma, Suleyman Akocak, Marc A. Ilies & Reza Fassihi. (2015) Solid-State Interactions at the Core-Coat Interface: Physicochemical Characterization of Enteric-Coated Omeprazole Pellets Without a Protective Sub-Coat. AAPS PharmSciTech 16:4, pages 934-943.
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