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Xenobiotica
the fate of foreign compounds in biological systems
Volume 36, 2006 - Issue 1
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Original

Role of P-glycoprotein in the hepatic metabolism of tacrolimus

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Pages 1-13 | Received 23 Sep 2005, Published online: 12 Jul 2010

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Xixi Huang, Rui Zhang, Tingyu Yang, Ye Wei, Chunxiao Yang, Jiani Zhou, Yani Liu & Shaojun Shi. (2021) Inhibition effect of epigallocatechin-3-gallate on the pharmacokinetics of calcineurin inhibitors, tacrolimus, and cyclosporine A, in rats. Expert Opinion on Drug Metabolism & Toxicology 17:1, pages 121-134.
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Ling Pei, Run Li, Hong Zhou, Wenxin Du, Yajie Gu, Yingshuo Jiang, Yongqing Wang, Xin Chen, Jianguo Sun & Junrong Zhu. (2023) A Physiologically Based Pharmacokinetic Approach to Recommend an Individual Dose of Tacrolimus in Adult Heart Transplant Recipients. Pharmaceutics 15:11, pages 2580.
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Fahadul Islam, Md. Rezaul Islam, Mohamed H. Nafady, Md. Faysal, Sharuk L. Khan, Mehrukh Zehravi, Talha Bin Emran & Md. Habibur Rahman. 2023. Pharmacogenomics. Pharmacogenomics 323 344 .
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Zulcaif Ahmad, Muhammad Imran Khan, Muhammad Irfan Siddique, Hafiz Shoaib Sarwar, Gul Shahnaz, Syed Zajif Hussain, Nadeem Irfan Bukhari, Irshad Hussain & Muhammad Farhan Sohail. (2020) Fabrication and Characterization of Thiolated Chitosan Microneedle Patch for Transdermal Delivery of Tacrolimus. AAPS PharmSciTech 21:2.
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Divya Dheer, Jyoti, Prem N. Gupta & Ravi Shankar. (2018) Tacrolimus: An updated review on delivering strategies for multifarious diseases. European Journal of Pharmaceutical Sciences 114, pages 217-227.
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K Sanghavi, R C Brundage, M B Miller, D P Schladt, A K Israni, W Guan, W S Oetting, R B Mannon, R P Remmel, A J Matas & P A Jacobson. (2015) Genotype-guided tacrolimus dosing in African-American kidney transplant recipients. The Pharmacogenomics Journal 17:1, pages 61-68.
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Niraj S. Trasi, Hitesh S. Purohit, Hong Wen, Dajun D. Sun & Lynne S. Taylor. (2017) Non-Sink Dissolution Behavior and Solubility Limit of Commercial Tacrolimus Amorphous Formulations. Journal of Pharmaceutical Sciences 106:1, pages 264-272.
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Vijaykumar Nekkanti, Javier Rueda, Zhijun Wang & Guru V Betageri. (2015) Design, Characterization, and In Vivo Pharmacokinetics of Tacrolimus Proliposomes. AAPS PharmSciTech 17:5, pages 1019-1029.
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Bojana Golubović, Katarina Vučićević, Dragana Radivojević, Sandra Vezmar Kovačević, Milica Prostran & Branislava Miljković. (2014) Total plasma protein effect on tacrolimus elimination in kidney transplant patients – Population pharmacokinetic approach. European Journal of Pharmaceutical Sciences 52, pages 34-40.
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Xiao Ling Qin, Xiao Chen, Ying Wang, Xin Ping Xue, Ying Wang, Jia Li Li, Xue Ding Wang, Guo Ping Zhong, Chang Xi Wang, Hui Yang, Min Huang & Hui Chang Bi. (2014) In Vivo to In Vitro Effects of Six Bioactive Lignans of Wuzhi Tablet ( Schisandra Sphenanthera Extract ) on the CYP3A/P-glycoprotein–Mediated Absorption and Metabolism of Tacrolimus . Drug Metabolism and Disposition 42:1, pages 193-199.
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Hyun Lee, Tian Zhu, Kavankumar Patel, Yan-Yan Zhang, Lena Truong, Kirk E. Hevener, Joseph L. Gatuz, Gitanjali Subramanya, Hyun-Young Jeong, Susan L. Uprichard & Michael E. Johnson. (2013) High-Throughput Screening (HTS) and Hit Validation to Identify Small Molecule Inhibitors with Activity against NS3/4A proteases from Multiple Hepatitis C Virus Genotypes. PLoS ONE 8:10, pages e75144.
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Hua Wei, Xia Tao, Peng Di, Yingbo Yang, Jingxian Li, Xiaofeng Qian, Jin Feng & Wansheng Chen. (2013) Effects of Traditional Chinese Medicine Wuzhi Capsule on Pharmacokinetics of Tacrolimus in Rats . Drug Metabolism and Disposition 41:7, pages 1398-1403.
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Xiao-Ling Qin, Tao Yu, Ling-Jue Li, Ying Wang, Hao-Min Gu, Yong-Tao Wang, Min Huang & Hui-Chang Bi. (2013) Effect of long-term co-administration of Wuzhi tablet (Schisandra sphenanthera extract) and prednisone on the pharmacokinetics of tacrolimus. Phytomedicine 20:3-4, pages 375-379.
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Nicolas Picard & Pierre Marquet. 2012. Pharmacogenomics in Clinical Therapeutics. Pharmacogenomics in Clinical Therapeutics 70 97 .
Su-Young Choi, Liam Fischer, Kyunghee Yang, Hyejin Chung & Hyunyoung Jeong. (2011) Isoform-specific regulation of cytochrome P450 expression and activity by estradiol in female rats. Biochemical Pharmacology 81:6, pages 777-782.
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Xiao Ling Qin, Hui Chang Bi, Xue Ding Wang, Jia Li Li, Ying Wang, Xin Ping Xue, Xiao Chen, Chang Xi Wang, Le Jia Xu, Yi Tao Wang & Min Huang. (2010) Mechanistic understanding of the different effects of Wuzhi Tablet (Schisandra sphenanthera extract) on the absorption and first-pass intestinal and hepatic metabolism of Tacrolimus (FK506). International Journal of Pharmaceutics 389:1-2, pages 114-121.
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K. Sandy Pang, Han-Joo Maeng & Jianghong Fan. (2009) Interplay of Transporters and Enzymes in Drug and Metabolite Processing. Molecular Pharmaceutics 6:6, pages 1734-1755.
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Xiao-ling Qin, Hui-chang Bi, Chang-xi Wang, Jia-li Li, Xue-ding Wang, Long-shan Liu, Xiao Chen & Min Huang. (2009) Study of the effect of Wuzhi tablet ( Schisandra sphenanthera extract) on tacrolimus tissue distribution in rat by liquid chromatography tandem mass spectrometry method . Biomedical Chromatography, pages n/a-n/a.
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Johnny Moretto, Germain Bessard & Françoise Stanke-Labesque. (2007) Médicaments immunosuppresseurs et antirétroviraux : une association riche en interactions. Therapies 62:4, pages 327-335.
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