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Xenobiotica
the fate of foreign compounds in biological systems
Volume 40, 2010 - Issue 3
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General Xenobiochemistry

Interaction of HIV protease inhibitors with OATP1B1, 1B3, and 2B1

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Pages 163-176 | Received 20 Sep 2009, Accepted 24 Nov 2009, Published online: 27 Jan 2010

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Aishwarya Jala, Srikanth Ponneganti, Devi Swetha Vishnubhatla, Gayathri Bhuvanam, Prithvi Raju Mekala, Bincy Varghese, Pullapanthula Radhakrishnanand, Ramu Adela, Upadhyayula Suryanarayana Murty & Roshan M. Borkar. (2021) Transporter-mediated drug–drug interactions: advancement in models, analytical tools, and regulatory perspective. Drug Metabolism Reviews 53:3, pages 285-320.
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Sumathy Mathialagan, Chester Costales, Laurie Tylaska, Emi Kimoto, Anna Vildhede, Jillian Johnson, Nathaniel Johnson, Takami Sarashina, Kenta Hashizume, Caleb D. Isringhausen, Lydia M. M. Vermeer, Andrea R. Wolff & A. David Rodrigues. (2018) In vitro studies with two human organic anion transporters: OAT2 and OAT7. Xenobiotica 48:10, pages 1037-1049.
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. (2016) Abstract. Drug Metabolism Reviews 48:sup1, pages 28-157.
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Melinda J. Reese, Gary D. Bowers, Joan E. Humphreys, Elizabeth P. Gould, Susan L. Ford, Lindsey O. Webster & Joseph W. Polli. (2016) Drug interaction profile of the HIV integrase inhibitor cabotegravir: assessment from in vitro studies and a clinical investigation with midazolam. Xenobiotica 46:5, pages 445-456.
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Jef Stappaerts, Sarinj Fattah, Pieter Annaert & Patrick Augustijns. (2014) Hepatobiliary and intestinal elimination of darunavir in an integrated preclinical rat model. Xenobiotica 44:6, pages 489-497.
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William J. Chiou, Sonia M. de Morais, Ryota Kikuchi, Richard L. Voorman, Xiaofeng Li & Daniel A. J. Bow. (2014) In vitro OATP1B1 and OATP1B3 inhibition is associated with observations of benign clinical unconjugated hyperbilirubinemia. Xenobiotica 44:3, pages 276-282.
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Roberto Lozano, Nieves Domeque & Alberto-Fermin Apesteguia. (2013) Atazanavir–bilirubin interaction: a pharmacokinetic–pharmacodynamic model. Clinical Pharmacology: Advances and Applications 5, pages 153-159.
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Nicolas Picard, Laure Levoir, Fabien Lamoureux, Sook Wah Yee, Kathleen M. Giacomini & Pierre Marquet. (2011) Interaction of sirolimus and everolimus with hepatic and intestinal organic anion-transporting polypeptide transporters. Xenobiotica 41:9, pages 752-757.
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Grant T. Generaux, Fiorenza M. Bonomo, Marta Johnson & Kelly M. Mahar Doan. (2011) Impact of SLCO1B1 (OATP1B1) and ABCG2 (BCRP) genetic polymorphisms and inhibition on LDL-C lowering and myopathy of statins. Xenobiotica 41:8, pages 639-651.
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. (2010) Invited Speakers. Drug Metabolism Reviews 42:sup1, pages 1-323.
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