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Xenobiotica
the fate of foreign compounds in biological systems
Volume 14, 1984 - Issue 5
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Original Article

Inhibition of mono-oxygenase and oxidase activity of rat-hepatic cytochrome P-450 by H2-receptor blockers

A. Bast Department of Pharmacology and Pharmacotherapy, Faculty of Pharmacy, State University of Utrecht, Catharijnesingel 60, 3511 GH, Utrecht, The Netherlands
,
K. M. Savenije-chapel Department of Pharmacology and Pharmacotherapy, Faculty of Pharmacy, State University of Utrecht, Catharijnesingel 60, 3511 GH, Utrecht, The Netherlands
&
B. H. Kroes Department of Pharmacology and Pharmacotherapy, Faculty of Pharmacy, State University of Utrecht, Catharijnesingel 60, 3511 GH, Utrecht, The Netherlands
Pages 399-408 | Received 03 Jan 1984, Published online: 30 Sep 2009

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Arnold R. Goeptar, Heleen Scheerens & Nico P. E. Vermeulen. (1995) Oxygen and Xenobiotic Reductase Activities of Cytochrome P450. Critical Reviews in Toxicology 25:1, pages 25-65.
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M. Paolini, R. Mesirca, L. Pozzetti, A. Sapone, G. L. Biagi, N. M. Trieff & G. Cantelli‐Forti. (1994) Correlation between murine liver cytochrome p450 2b1 induction by halogenated hydrocarbons and toxicity. Toxicological & Environmental Chemistry 44:1-2, pages 55-64.
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M. Paolini, R. Mesirca, L. Pozzetti, A. Sapone, E. Sapigni, G. L. Biagi, N. M. Trieff & G. Cantelli‐Forti. (1994) Correlation between cytochrome p450 2b1 induction by barbiturates and toxicity in the chick embryo in ovo . Toxicological & Environmental Chemistry 44:1-2, pages 43-53.
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E. Tanaka, Z. Daling, K. Abe, T. Nakamura & T. Horie. (1994) Dual effects of a novel thienodiazepine platelet-activating factor antagonist, on drug-oxidizing enzymes in beagle dog. Xenobiotica 24:4, pages 293-300.
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M. Stefek. (1993) I n vitvo studies on the interaction of the pyridoindole antioxidant stobadine with rat liver microsomal P450. Xenobiotica 23:9, pages 983-993.
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J. O. Persson, Y. Terelius & M. Ingelman-sundberg. (1990) Cytochrome P-450-dependent formation of reactive oxygen radicals: isozyme-specific inhibition of P-450-mediated reduction of oxygen and carbon tetrachloride. Xenobiotica 20:9, pages 887-900.
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W. Gristwood & K. Wilson. (1988) Kinetics of some benzothiazoles, benzoxazoles, and quinolines as substrates and inhibitors of rabbit liver aldehyde oxidase. Xenobiotica 18:8, pages 949-954.
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Michael Murray. (1987) Mechanisms of the Inhibition of Cytochrome P 450-Mediated Drug Oxidation by Therapeutic Agents. Drug Metabolism Reviews 18:1, pages 55-81.
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UrmilaM. Joshi & JohnE. Thornburg. (1986) Interactions between cimetidine, methylparathion, and parathion. Journal of Toxicology and Environmental Health 19:3, pages 337-344.
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Articles from other publishers (29)

R Leurs, D Donnell, H Timmerman & A Bast. (1989) Interaction of Nefopam and Orphenadrine with the Cytochrome P-450 and the Glutathione System in Rat Liver. Journal of Pharmacy and Pharmacology 41:6, pages 388-393.
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M. J. Eccles, T. C. Danbury, J. M. Ford & C. J. C. Roberts. (1997) The effect of velnacrine on the mixed function oxidase system. European Journal of Drug Metabolism and Pharmacokinetics 22:2, pages 121-125.
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Pekka Uotila. (1996) The role of cyclic AMP and oxygen intermediates in the inhibition of cellular immunity in cancer. Cancer Immunology, Immunotherapy 43:1, pages 1-9.
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Peter H. Roos & Axel Mahnke. (1996) Metabolite complex formation of orphenadrine with cytochrome P450. Biochemical Pharmacology 52:1, pages 73-84.
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M. Paolini, G. L. Biagi, C. Bauer & G. Cantelli‐Forti. (2013) Cocktail Strategy: Complications and Limitations. The Journal of Clinical Pharmacology 33:11, pages 1011-1012.
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Ron M. C. Herings, Bruno H. Ch. Stricker, Hubert G. M. Leufkens, Albert Bakker, Ferd Sturmans & John Urquhart. (1993) Public health problems and the rapid estimation of the size of the population at risk. Pharmacy World & Science 15:5, pages 212-218.
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Nevins W. Todd, Christine M. Hunt, Thomas P. Kennedy, Claude A. Piantadosi & A. Richard Whorton. (1992) Effects of Inhibition and Induction of Cytochrome P-450 Isozymes on Hyperoxic Lung Injury in Rats. American Journal of Respiratory Cell and Molecular Biology 7:2, pages 222-229.
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Arnold R. Goeptar, Johan M. Te Koppele, Etienne P.A. Neve & Nico P.E. Vermeulen. (1992) Reductase and oxidase activity of rat liver cytochrome P450 with 2,3,5,6-tetramethylbenzoquinone as substrate. Chemico-Biological Interactions 83:3, pages 249-269.
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C. Saunier, G. Audibert, D. Hartemann, A. Sautegeau, P. Amend, O. Bigard & C. Alvernhe. (2008) Preserved CO 2 response in cerebral and muscular blood vessels during cimetidine treatment . Clinical Physiology 11:4, pages 367-373.
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H. van der Goot, A. Bast & H. Timmerman. 1991. Histamine and Histamine Antagonists. Histamine and Histamine Antagonists 573 748 .
Kamlesh P. Vyas, Prasad H. Kari, Regina W. Wang & Anthony Y.H. Lu. (1990) Biotransformation of lovastatin—III. Biochemical Pharmacology 39:1, pages 67-73.
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Aalt Bast & Guido R. M. M. Haenen. 1990. Free Radicals, Lipoproteins, and Membrane Lipids. Free Radicals, Lipoproteins, and Membrane Lipids 359 370 .
Gunilla Ekström & Magnus Ingelman-Sundberg. (1989) Rat liver microsomal NADPH-supported oxidase activity and lipid peroxidation dependent on ethanol-inducible cytochrome P-450 (P-450IIE1). Biochemical Pharmacology 38:8, pages 1313-1319.
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A. Bast, P. A. L. Goossens & E. M. Savenije-Chapel. (1989) Dependence of hydrogen peroxide formation in rat liver microsomes on the molecular structure of cytochrome P-450 substrates: A study with barbiturates and β-adrenoceptor antagonists. European Journal of Drug Metabolism and Pharmacokinetics 14:2, pages 93-100.
Crossref
A. Bast, K. Smid & H. Timmerman. (1989) The effects of cimetidine, ranitidine and famotidine on rat hepatic microsomal cytochrome P-450 activities. Agents and Actions 27:1-2, pages 188-191.
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Sylvie Rolin, Hajar Souhaili-El Amri, Anne-Marie Batt, Michele Levy, Denyse Bagrel & Gerard Siest. (1989) Study of the in vitro bioactivation of albendazole in human liver microsomes and hepatoma cell lines. Cell Biology and Toxicology 5:1, pages 1-14.
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G. Ignesti, F. Buffoni, M. Perretti & A. Cintelli. (1988) Induction and quail liver diamine oxidase (histaminase). Part II: Different responses to the inducers. Agents and Actions 25:1-2, pages 43-47.
Crossref
Ylva Terelius & Magnus Ingelman-Sundberg. (1988) Cytochrome P-450-dependent oxidase activity and hydroxyl radical production in micellar and membranous types of reconstituted systems. Biochemical Pharmacology 37:7, pages 1383-1389.
Crossref
Ulrich Förstermann, Ute Alheid, Jürgen C. Frölich & Alexander Mülsch. (2012) Mechanisms of action of lipoxygenase and cytochrome P‐450‐mono‐oxygenase inhibitors in blocking endothelium‐dependent vasodilatation. British Journal of Pharmacology 93:3, pages 569-578.
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Hajar Souhaili-El Amri, Xavier Fargetton, Etienne Benoit, Muriel Totis & Anne-Marie Batt. (1988) Inducing effect of albendazole on rat liver drug-metabolizing enzymes and metabolite pharmacokinetics. Toxicology and Applied Pharmacology 92:1, pages 141-149.
Crossref
E. Rekka, G.J. Sterk, H. Timmerman & A. Bast. (1988) Identification of structural characteristics of some potential H2-receptor antagonists that determine the interaction with rat hepatic P-450. Chemico-Biological Interactions 67:1-2, pages 117-127.
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M. Mitchard, A. Harris & B.M. Mullinger. (1987) Ranitidine drug interactions—a literature review. Pharmacology & Therapeutics 32:3, pages 293-325.
Crossref
R. M. Lee & R. D. McDowall. (1986) RECENT ADVANCES IN PHARMACEUTICAL CHEMISTRY—REVIEW II HISTAMINE H 2 -RECEPTOR ANTAGONISTS . Journal of Clinical Pharmacy and Therapeutics 11:6, pages 389-408.
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Markku Pasanen, Pentti Arvela, Olavi Pelkonen, Eero Sotaniemi & Ulrich Klotz. (1986) Effect of five structurally diverse H2-receptor antagonists on drug metabolism. Biochemical Pharmacology 35:24, pages 4457-4461.
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Yasuharu Imai, Masami Inada, Shinji Tamura, Shuzo Noda, Sumio Kawata, Yuzo Minami & Seiichiro Tarui. (1986) Interaction of famotidine with rat liver microsomes, a study showing less inhibition of drug metabolism than with cimetidine. Pharmacological Research Communications 18:7, pages 629-638.
Crossref
Karel Lavrjusen, Jos Van Houdt, Dirk Thius, Willem Meuldermans & Jos Heykants. (1986) Induction potential of antifungals containing an imidazole or triazole moiety. Biochemical Pharmacology 35:11, pages 1867-1878.
Crossref
Aalt Bast. (1986) Is formation of reactive oxygen by cytochrome P-450 perilous and predictable?. Trends in Pharmacological Sciences 7, pages 266-270.
Crossref
Paul R. Ortiz de Montellano. 1986. Cytochrome P-450. Cytochrome P-450 217 271 .
Aalt Bast & Guido R.M.M. Haenen. (1984) Cytochrome P-450 and glutathione: what is the significance of their interrelationship in lipid peroxidation?. Trends in Biochemical Sciences 9:12, pages 510-513.
Crossref

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