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Xenobiotica
the fate of foreign compounds in biological systems
Volume 19, 1989 - Issue 6
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Research Article

Pharmacokinetics of the Antidepressant Rolipram in Healthy Volunteers

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Pages 683-692 | Received 22 Sep 1988, Accepted 12 Feb 1989, Published online: 22 Sep 2008

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Ajaib S. Paintlia, Manjeet K. Paintlia, Inderjit Singh & Avtar K. Singh. (2008) Combined medication of lovastatin with rolipram suppresses severity of experimental autoimmune encephalomyelitis. Experimental Neurology 214:2, pages 168-180.
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David R. Sprague, Masahiro Fujita, Yong Hoon Ryu, Jeih-San Liow, Victor W. Pike & Robert B. Innis. (2008) Whole-body biodistribution and radiation dosimetry in monkeys and humans of the phosphodiesterase 4 radioligand [11C](R)-rolipram: comparison of two-dimensional planar, bisected and quadrisected image analyses. Nuclear Medicine and Biology 35:4, pages 493-500.
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Bradley Newhouse, Shelley Allen, Benjamin Fauber, Aaron S. Anderson, C. Todd Eary, Joshua D. Hansen, Justin Schiro, John J. Gaudino, Ellen Laird, David Chantry, Christine Eberhardt & Laurence E. Burgess. (2004) Racemic and chiral lactams as potent, selective and functionally active CCR4 antagonists. Bioorganic & Medicinal Chemistry Letters 14:22, pages 5537-5542.
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Gail W. Sullivan, Holliday T. Carper & Gerald L. Mandell. (1995) The specific type IV phosphodiesterase inhibitor rolipram combined with adenosine reduces tumor necrosis factor-α-primed neutrophil oxidative activity. International Journal of Immunopharmacology 17:10, pages 793-803.
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N. Sommer, P.-A. Löschmann, G.H. Northoff, M. Weller, A. Steinbrecher, J.P. Steinbach, R. Lichtenfels, R. Meyermann, A. Riethmüller, A. Fontana, J. Dichgans & R. Martin. (1995) The antidepressant rolipram suppresses cytokine production and prevents autoimmune encephalomyelitis. Nature Medicine 1:3, pages 244-248.
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Claudia C.S. Chini, Eduardo N. Chini, Josie M. Williams, Karel Matoušovic & Thomas P. Dousa. (1994) Formation of reactive oxygen metabolites in glomeruli is suppressed by inhibition of cAMP phosphodiesterase isozyme type IV. Kidney International 46:1, pages 28-36.
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J. Semmler, H. Wachtell & S. Endres. (1993) The specific type IV phosphodiesterase inhibitor rolipram suppresses tumor necrosis factor-α production by human mononuclear cells. International Journal of Immunopharmacology 15:3, pages 409-413.
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G. Laux, A. Delini-Stula, U. Breyer-Pfaff, J. Demling, D. Ebert, W. Pöldinger, S. Kasper, M. Osterheider, O. Dietmaier, H.-J. Möller & J. Fuger. 1993. Neuro-Psychopharmaka. Neuro-Psychopharmaka 105 268 .
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Anton J. M. Loonen. (1992) Dealing with sadness, madness and hostility. Pharmaceutisch Weekblad Scientific Edition 14:4, pages 206-220.
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W. Krause & G. Kühne. (1992) High-performance liquid chromatographic procedure for specificity testing of radioimmunoassays: rolipram. Journal of Chromatography B: Biomedical Sciences and Applications 573:2, pages 303-308.
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W. Krause, G. K�hne & N. Sauerbrey. (1990) Pharmacokinetics of (+)-rolipram and (?)-rolipram in healthy volunteers. European Journal of Clinical Pharmacology 38:1, pages 71-75.
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