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D. McKILLOP*C. J. BUTTERS, S. J. HILL, P. J. SIMONS, T. L. EDWARDS & S. E. DOUGHTY. (1998) Enzyme-inducing effects of bicalutamide in mouse, rat and dog. Xenobiotica 28:5, pages 465-478.
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P. J. Simons, I. D. Cockshott, E. J. Douglas, E. A. Gordon, S. Knott & R. J. Ruane. (1991) Distribution in female rats of an anaesthetic intravenous dose of 14C-propofol. Xenobiotica 21:10, pages 1325-1335.
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P. J. Simons, I. D. Cockshott, E. J. Douglas, E. A. Gordon, S. Knott & R. J. Ruane. (1991) Species differences in blood profiles, metabolism and excretion of 14C-propofol after intravenous dosing to rat, dog and rabbit. Xenobiotica 21:10, pages 1243-1256.
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Articles from other publishers (19)
Yoshiyuki Akiyama, Naoya Matsumura, Asami Ono, Shun Hayashi, Satoko Funaki, Naomi Tamura, Takahiro Kimoto, Maiko Jiko, Yuka Haruna, Akiko Sarashina, Masahiro Ishida, Kotaro Nishiyama, Masahiro Fushimi, Yukiko Kojima, Takuya Fujita & Kiyohiko Sugano. (2022) Prediction of Oral Drug Absorption in Rats from In Vitro Data. Pharmaceutical Research 40:2, pages 359-373.
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Wenjing Shi, Haixiao Di, Bo Pang, Huixin Jin, Hongtao Liu, Bo Qiu, Bingnan Ren & Guoxun Pang. (2022) Comparative pharmacokinetic study of bicalutamide administration alone and in combination with vitamin D in rats. Acta Chromatographica 34:4, pages 453-460.
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Salvatore Ferla, Marcella Bassetto, Fabrizio Pertusati, Sahar Kandil, Andrew D. Westwell, Andrea Brancale & Christopher McGuigan. (2016) Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety. Bioorganic & Medicinal Chemistry Letters 26:15, pages 3636-3640.
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Suresh P. S., S. Vijay Kumar, Avinash Kumar & Ramesh Mullangi. (2015) Development of an LC-MS/MS method for determination of bicalutamide on dried blood spots: application to pharmacokinetic study in mice. Biomedical Chromatography 29:2, pages 254-260.
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Juhyun Kim, Christopher C. Coss & James T. Dalton. (2013) Effect of para halogen modification of S-3-(phenoxy)-2-hydroxy-2-methyl-N-(4-nitro-3-trifluoromethyl-phenyl)-propionamides on metabolism and clearance. Archives of Pharmacal Research 37:11, pages 1464-1476.
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Kuldeep Sharma, Gopal V. Pawar, Sanjeev Giri, Sriram Rajagopal & Ramesh Mullangi. (2012) Development and validation of a highly sensitive LC‐MS/MS‐ESI method for the determination of bicalutamide in mouse plasma: application to a pharmacokinetic study. Biomedical Chromatography 26:12, pages 1589-1595.
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Minoli A. Perera, Donghua Yin, Di Wu, Kenneth K. Chan, Duane D. Miller & James Dalton. (2006) In Vivo Metabolism and Final Disposition of a Novel Nonsteroidal Androgen in Rats and Dogs. Drug Metabolism and Disposition 34:10, pages 1713-1721.
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Wenqing Gao, Juhyun Kim & James T. Dalton. (2006) Pharmacokinetics and Pharmacodynamics of Nonsteroidal Androgen Receptor Ligands. Pharmaceutical Research 23:8, pages 1641-1658.
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Di Wu, Zengru Wu, Jun Yang, Vipin A. Nair, Duane D. Miller & James T. Dalton. (2006) PHARMACOKINETICS AND METABOLISM OF A SELECTIVE ANDROGEN RECEPTOR MODULATOR IN RATS: IMPLICATION OF MOLECULAR PROPERTIES AND INTENSIVE METABOLIC PROFILE TO INVESTIGATE IDEAL PHARMACOKINETIC CHARACTERISTICS OF A PROPANAMIDE IN PRECLINICAL STUDY. Drug Metabolism and Disposition 34:3, pages 483-494.
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Juhyun Kim, Di Wu, Dong Jin Hwang, Duane D. Miller & James T. Dalton. (2005)
The
Para
Substituent of
S
-3-(Phenoxy)-2-hydroxy-2-methyl-
N
-(4-nitro-3-trifluoromethyl-phenyl)-propionamides Is a Major Structural Determinant of in Vivo Disposition and Activity of Selective Androgen Receptor Modulators
. Journal of Pharmacology and Experimental Therapeutics 315:1, pages 230-239.
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Ian D Cockshott. (2004) Bicalutamide. Clinical Pharmacokinetics 43:13, pages 855-878.
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Donghua Yin, Huiping Xu, Yali He, Leonid I. Kirkovsky, Duane D. Miller & James T. Dalton. (2003) Pharmacology, Pharmacokinetics, and Metabolism of Acetothiolutamide, a Novel Nonsteroidal Agonist for the Androgen Receptor. Journal of Pharmacology and Experimental Therapeutics 304:3, pages 1323-1333.
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Yali He, Donghua Yin, Minoli Perera, Leonid Kirkovsky, Nina Stourman, Wei Li, James T Dalton & Duane D Miller. (2002) Novel nonsteroidal ligands with high binding affinity and potent functional activity for the androgen receptor. European Journal of Medicinal Chemistry 37:8, pages 619-634.
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Tara Nickerson & Michael Pollak. (1999) Bicalutamide (Casodex)-induced prostate regression involves increased expression of genes encoding insulin-like growth factor binding proteins. Urology 54:6, pages 1120-1125.
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Geert J.C.M. Kolvenbag & Anthony Nash. (1999) Bicalutamide dosages used in the treatment of prostate cancer. The Prostate 39:1, pages 47-53.
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James T. Dalton, Arnab Mukherjee, Zixin Zhu, Leonid Kirkovsky & Duane D. Miller. (1998) Discovery of Nonsteroidal Androgens. Biochemical and Biophysical Research Communications 244:1, pages 1-4.
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B.J.A. Furr & H. Tucker. (1996) The preclinical development of bicalutamide: pharmacodynamics and mechanism of action. Urology 47:1, pages 13-25.
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Mark S. Soloway, Paul F. Schellhammer, Joseph A. Smith, Gerald W. Chodak, Nicholas J. Vogelzang & Gerard T. Kennealey. (1995) Bicalutamide in the Treatment of Advanced Prostatic Carcinoma. The Journal of Urology, pages 2110-2114.
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Mark S. Soloway, Paul F. Schellhammer, Joseph A. Jr. Smith, Gerald W. Chodak, Nicholas J. Vogelzang & Gerard T. Kennealey. (1995) Bicalutamide in the Treatment of Advanced Prostatic Carcinoma: A Phase II Noncomparative Multicenter Trial Evaluating Safety, Efficacy and Long-Term Endocrine Effects of Monotherapy. Journal of Urology 154:6, pages 2110-2114.
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