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Xenobiotica
the fate of foreign compounds in biological systems
Volume 22, 1992 - Issue 8
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Research Article

Hep G2 cell line as a human model for sulphate conjugation of drugs

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Pages 973-982 | Received 01 May 1991, Accepted 01 Feb 1992, Published online: 22 Sep 2008

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Lijun Luo, Chunyang Zhou, Katsuhisa Kurogi, Yoichi Sakakibara, Masahito Suiko & Ming-Cheh Liu. (2016) Sulfation of 6-hydroxymelatonin, N-acetylserotonin and 4-hydroxyramelteon by the human cytosolic sulfotransferases (SULTs). Xenobiotica 46:7, pages 612-619.
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Articles from other publishers (25)

Chaojun Jia, Lijun Luo, Katsuhisa Kurogi, Juming Yu, Chunyang Zhou & Ming-Cheh Liu. (2016) Identification of the Human SULT Enzymes Involved in the Metabolism of Rotigotine. The Journal of Clinical Pharmacology 56:6, pages 754-760.
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Katsuhisa Kurogi, Andriy Chepak, Michael T. Hanrahan, Ming-Yih Liu, Yoichi Sakakibara, Masahito Suiko & Ming-Cheh Liu. (2014) Sulfation of opioid drugs by human cytosolic sulfotransferases: Metabolic labeling study and enzymatic analysis. European Journal of Pharmaceutical Sciences 62, pages 40-48.
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Yue Chen, Shunfen Zhang, Tianyan Zhou, Chaoqun Huang, Alicia McLaughlin & Guangping Chen. (2013) Liver X receptor alpha mediated genistein induction of human dehydroepiandrosterone sulfotransferase (hSULT2A1) in Hep G2 cells. Toxicology and Applied Pharmacology 268:2, pages 106-112.
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K. Ko, K. Kurogi, G. Davidson, M.-Y. Liu, Y. Sakakibara, M. Suiko & M.-C. Liu. (2012) Sulfation of ractopamine and salbutamol by the human cytosolic sulfotransferases. Journal of Biochemistry 152:3, pages 275-283.
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Tsung-Ho Ying, Shun-Fa Yang, Su-Ju Tsai, Shu-Ching Hsieh, Yi-Chang Huang, Da-Tian Bau & Yi-Hsien Hsieh. (2011) Fisetin induces apoptosis in human cervical cancer HeLa cells through ERK1/2-mediated activation of caspase-8-/caspase-3-dependent pathway. Archives of Toxicology 86:2, pages 263-273.
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Jorge Raul Pasqualini. (2009) Estrogen Sulfotransferases in Breast and Endometrial Cancers. Annals of the New York Academy of Sciences 1155:1, pages 88-98.
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Hao Sheng Bian, Sherry Yan Yan Ngo, Weiqi Tan, Chang Hua Wong, Urs A. Boelsterli & Theresa May Chin Tan. (2007) Induction of human sulfotransferase 1A3 (SULT1A3) by glucocorticoids. Life Sciences 81:25-26, pages 1659-1667.
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Jorge Pasqualini & Gerard Chetrite. 2005. Human Cytosolic Sulfotransferases. Human Cytosolic Sulfotransferases 135 156 .
Chi-Tai Yeh, Shang-Ming Huang & Gow-Chin Yen. (2005) Induction of Phenolsulfotransferase Expression by Phenolic Acids in Human Hepatoma HepG 2 Cells . Journal of Agricultural and Food Chemistry 53:12, pages 4766-4773.
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Junko Miyano, Shigeo Yamamoto, Nobumitsu Hanioka, Shizuo Narimatsu, Tsutomu Ishikawa, Kenichiro Ogura, Tadashi Watabe, Masuhiro Nishimura, Nobuhiko Ueda & Shinsaku Naito. (2005) Involvement of SULT1A3 in elevated sulfation of 4-hydroxypropranolol in Hep G2 cells pretreated with β-naphthoflavone. Biochemical Pharmacology 69:6, pages 941-950.
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David W. Boulton & J. Paul Fawcett. (2001) The Pharmacokinetics of Levosalbutamol. Clinical Pharmacokinetics 40:1, pages 23-40.
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Shizuo Narimatsu, Naoko Kobayashi, Kazuo Asaoka, Yasuhiro Masubuchi, Toshiharu Horie, Masakiyo Hosokawa, Tsutomu Ishikawa, Shigeru Ohmori, Mitsukazu Kitada, Junko Miyano, Hiroyuki Kataoka & Shigeo Yamamoto. (2001) High-performance liquid chromatographic analysis of the sulfation of 4-hydroxypropranolol enantiomers by monkey liver cytosol. Chirality 13:3, pages 140-147.
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Yoko Otake, Amy L Nolan, U.Kristina Walle & Thomas Walle. (2000) Quercetin and resveratrol potently reduce estrogen sulfotransferase activity in normal human mammary epithelial cells. The Journal of Steroid Biochemistry and Molecular Biology 73:5, pages 265-270.
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U.Kristina Walle, Alema Galijatovic & Thomas Walle. (1999) Transport of the flavonoid chrysin and its conjugated metabolites by the human intestinal cell line Caco-2. Biochemical Pharmacology 58:3, pages 431-438.
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A.G Schuur, Å Bergman, A Brouwer & T.J Visser. (1999) Effects of Pentachlorophenol and Hydroxylated Polychlorinated Biphenyls on Thyroid Hormone Conjugation in a Rat and a Human Hepatoma Cell Line. Toxicology in Vitro 13:3, pages 417-425.
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T.J Schrader. (1999) Comparison of HepG2 feeder cells generated by exposure to γ-rays, X-rays, UV-C light or mitomycin C for ability to activate 7,12-dimethylbenz[a]anthracene in a cell-mediated Chinese hamster V79/HGPRT mutation assay. Mutation Research/Fundamental and Molecular Mechanisms of Mutagenesis 423:1-2, pages 137-148.
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M. Jurima-romet, H.S. Huang, D.J. Beck & A.P. Li. (1996) Evaluation of drug interactions in intact hepatocytes: Inhibitors of terfenadine metabolism. Toxicology in Vitro 10:6, pages 655-663.
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E. ALISON EATON, U. KRISTINA WALLE, HUGH M. WILSON, GUNNAR ABERG & THOMAS WALLE. (2008) Stereoselective sulphate conjugation of salbutamol by human lung and bronchial epithelial cells. British Journal of Clinical Pharmacology 41:3, pages 201-206.
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Thomas Walle, E. Alison Eaton, U. Kristina Walle & Gene R. Pesola. (1996) Stereoselective metabolism ofRS-albuterol in humans. Clinical Reviews in Allergy & Immunology 14:1, pages 101-113.
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Thomas Walle, E.Alison Eaton & U.Kristina Walle. (1995) Quercetin, a potent and specific inhibitor of the human P-form phenolsulfotransferase. Biochemical Pharmacology 50:5, pages 731-734.
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Yoichi Sakakibara, Masahito Suiko & Ming‐Cheh Liu. (2008) De novo Sulfation of l ‐Tyrosine in HepG2 Human Hepatoma Cells and Its Possible Functional Implication . European Journal of Biochemistry 226:2, pages 293-301.
Crossref
Thomas Walle, U.Kristina Walle, Jill A. Shwed, Kelly R. Thornburg, Chad E. Mathis & Gene R. Pesola. (1994) Human phenolsulfotransferases: chiral substrates and expression in Hep G2 cells. Chemico-Biological Interactions 92:1-3, pages 47-55.
Crossref
UK Walle, GR Pesola & T Walle. (2012) Stereoselective sulphate conjugation of salbutamol in humans: comparison of hepatic, intestinal and platelet activity.. British Journal of Clinical Pharmacology 35:4, pages 413-418.
Crossref
Thomas D. Eller, U.Kristina Walle & Thomas Walle. (1993) Immunoaffinity isolation of the sulfate conjugate of 4'-hydroxypropranolol from plasma. Journal of Chromatography B: Biomedical Sciences and Applications 612:2, pages 320-325.
Crossref
Gene R. Pesola & Thomas Walle. (1993) Stereoselective sulfate conjugation of isoproterenol in humans: Comparison of hepatic, intestinal, and platelet activity. Chirality 5:8, pages 602-609.
Crossref

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