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Review Article

Hepatic OATP and OCT uptake transporters: their role for drug-drug interactions and pharmacogenetic aspects

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Pages 380-401 | Accepted 17 Nov 2009, Published online: 25 Jan 2010

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Mustafa Modiwala, Tarang Jadav, Amit Kumar Sahu, Rakesh K. Tekade & Pinaki Sengupta. (2022) A Critical Review on Advancement in Analytical Strategies for the Quantification of Clinically Relevant Biological Transporters. Critical Reviews in Analytical Chemistry 52:7, pages 1557-1571.
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Rui-Feng Liang, Wen-Jing Ge, Xian-Mei Song, Jun-Ping Zhang, Wei-Feng Cui, She-Feng Zhang & Geng-Sheng Li. (2020) Involvement of organic anion-transporting polypeptides and organic cation transporter in the hepatic uptake of jatrorrhizine. Xenobiotica 50:4, pages 479-487.
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Manuela de Lima Toccafondo Vieira & Carlos Alberto Tagliati. (2014) Hepatobiliary transporters in drug-induced cholestasis: a perspective on the current identifying tools. Expert Opinion on Drug Metabolism & Toxicology 10:4, pages 581-597.
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William J. Chiou, Sonia M. de Morais, Ryota Kikuchi, Richard L. Voorman, Xiaofeng Li & Daniel A. J. Bow. (2014) In vitro OATP1B1 and OATP1B3 inhibition is associated with observations of benign clinical unconjugated hyperbilirubinemia. Xenobiotica 44:3, pages 276-282.
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David A Powell. (2014) An overview of patented small molecule stearoyl coenzyme-A desaturase inhibitors (2009 – 2013). Expert Opinion on Therapeutic Patents 24:2, pages 155-175.
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Hugh A Barton, Yurong Lai, Theunis C Goosen, Hannah M Jones, Ayman F El-Kattan, James R Gosset, Jian Lin & Manthena V Varma. (2013) Model-based approaches to predict drug–drug interactions associated with hepatic uptake transporters: preclinical, clinical and beyond. Expert Opinion on Drug Metabolism & Toxicology 9:4, pages 459-472.
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Alexander M Cressman, Vanja Petrovic & Micheline Piquette-Miller. (2012) Inflammation-mediated changes in drug transporter expression/activity: implications for therapeutic drug response. Expert Review of Clinical Pharmacology 5:1, pages 69-89.
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