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Review Article

Fetoprotective activity of breast cancer resistance protein (BCRP, ABCG2): expression and function throughout pregnancy

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Pages 53-68 | Received 24 Mar 2010, Accepted 09 Jul 2010, Published online: 20 Sep 2010

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Jakub Hofman, Radim Kučera, Zuzana Neumanova, Jiri Klimes, Martina Ceckova & Frantisek Staud. (2016) Placental passage of olomoucine II, but not purvalanol A, is affected by p-glycoprotein (ABCB1), breast cancer resistance protein (ABCG2) and multidrug resistance-associated proteins (ABCCs). Xenobiotica 46:5, pages 416-423.
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Frantisek Staud & Martina Ceckova. (2015) Regulation of drug transporter expression and function in the placenta. Expert Opinion on Drug Metabolism & Toxicology 11:4, pages 533-555.
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Frantisek Staud, Lukas Cerveny & Martina Ceckova. (2012) Pharmacotherapy in pregnancy; effect of ABC and SLC transporters on drug transport across the placenta and fetal drug exposure. Journal of Drug Targeting 20:9, pages 736-763.
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Aizati NA Daud, Jorieke EH Bergman, Marian K Bakker, Hao Wang, Hermien EK de Walle, Torsten Plösch & Bob Wilffert. (2014) Pharmacogenetics of drug-induced birth defects: the role of polymorphisms of placental transporter proteins. Pharmacogenomics 15:7, pages 1029-1041.
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D. Beghin. (2014) Le passage placentaire des médicamentsPlacental transfer of drugs. Revue de médecine périnatale 6:1, pages 12-20.
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G Moreno-Sanz, O Sasso, A Guijarro, O Oluyemi, R Bertorelli, A Reggiani & D Piomelli. (2012) Pharmacological characterization of the peripheral FAAH inhibitor URB937 in female rodents: interaction with the Abcg2 transporter in the blood-placenta barrier. British Journal of Pharmacology 167:8, pages 1620-1628.
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Adeniyi Olagunju, Andrew Owen & Tim R Cressey. (2012) Potential effect of pharmacogenetics on maternal, fetal and infant antiretroviral drug exposure during pregnancy and breastfeeding. Pharmacogenomics 13:13, pages 1501-1522.
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Sarabjit S. Gahir & Micheline Piquette-Miller. (2011) Gestational and Pregnane X Receptor-Mediated Regulation of Placental ATP-Binding Cassette Drug Transporters in Mice. Drug Metabolism and Disposition 39:3, pages 465-471.
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