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Research Article

Flocculated amorphous itraconazole nanoparticles for enhanced in vitro supersaturation and in vivo bioavailability

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Pages 557-570 | Received 19 Jan 2011, Accepted 16 Aug 2011, Published online: 01 Oct 2011

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Neeraj Kumar, Shishu, Gulshan Bansal, Sandeep Kumar & Asim Kumar Jana. (2013) Preparation and cyclodextrin assisted dissolution rate enhancement of itraconazolium dinitrate salt. Drug Development and Industrial Pharmacy 39:2, pages 342-351.
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Naila A. Mugheirbi & Lidia Tajber. (2015) Mesophase and size manipulation of itraconazole liquid crystalline nanoparticles produced via quasi nanoemulsion precipitation. European Journal of Pharmaceutics and Biopharmaceutics 96, pages 226-236.
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Lindsay A. Wegiel, Laura I. Mosquera-Giraldo, Lisa J. Mauer, Kevin J. Edgar & Lynne S. Taylor. (2015) Phase Behavior of Resveratrol Solid Dispersions Upon Addition to Aqueous media. Pharmaceutical Research 32:10, pages 3324-3337.
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Hong Yu & Kunn Hadinoto. (2015) Mitigating the adverse effect of spray drying on the supersaturation generation capability of amorphous nanopharmaceutical powders. Powder Technology 277, pages 97-104.
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Naila A. Mugheirbi, Krzysztof J. Paluch & Lidia Tajber. (2014) Heat induced evaporative antisolvent nanoprecipitation (HIEAN) of itraconazole. International Journal of Pharmaceutics 471:1-2, pages 400-411.
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Wean Sin Cheow, Tie Yi Kiew, Yue Yang & Kunn Hadinoto. (2014) Amorphization Strategy Affects the Stability and Supersaturation Profile of Amorphous Drug Nanoparticles. Molecular Pharmaceutics 11:5, pages 1611-1620.
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K. Gilani, Z. Daman, E. Moazeni, A. Ghaffari, M. Pourasgari & M.A. Barghi. (2014) Preparation and characterization of various solid dispersion formulations of itraconazole to enhance the drug dissolution profile. Journal of Drug Delivery Science and Technology 24:6, pages 659-664.
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Raman Iyer, Navnit Shah, Harpreet Sandhu, Duk Soon Choi, Hitesh Chokshi & A.Waseem Malick. 2014. Amorphous Solid Dispersions. Amorphous Solid Dispersions 373 394 .
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Stephanie Bosselmann, Masao Nagao, Keat T. Chow & Robert O. Williams. (2012) Influence of Formulation and Processing Variables on Properties of Itraconazole Nanoparticles Made by Advanced Evaporative Precipitation into Aqueous Solution. AAPS PharmSciTech 13:3, pages 949-960.
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Xue-Zhong Zhang, Xin-En Huang, Yan-Li Xu, Xiu-Qun Zhang, Ai-ling Su & Zheng-Shan Shen. (2012) Phase II Study on Voriconazole for Treatment of Chinese Patients with Malignant Hematological Disorders and Invasive Aspergillosis. Asian Pacific Journal of Cancer Prevention 13:5, pages 2415-2418.
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