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Journal of Receptor Research Volume 6, 1986 - Issue 5-6
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Research Article

The Binding of Agonists and Antagonists to Rat Lung Beta-Adrenergic Receptors as Investigated by Thermodynamics and Structure-activity Relationships

Françoise Bree Département de Pharmacologie UER de Médecine, Université Paris XII, 8 rue du Général Sarrail, Creteil, F-94010, France
,
Nabil El Tayar Ecole de Pharmacie, Université de Lausanne, 3 place du Château, CH-1005, Lausanne, Suisse, France
,
Han Van de Waterbeemd Ecole de Pharmacie, Université de Lausanne, 3 place du Château, CH-1005, Lausanne, Suisse, France
,
Bernard Testa Ecole de Pharmacie, Université de Lausanne, 3 place du Château, CH-1005, Lausanne, Suisse, France
&
Jean-Paul Tillement Département de Pharmacologie UER de Médecine, Université Paris XII, 8 rue du Général Sarrail, Creteil, F-94010, France
Pages 381-409 | Published online: 26 Sep 2008

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V.N. Novoseletsky, T.V. Pyrkov & R.G. Efremov. (2010) Analysis of hydrophobic interactions of antagonists with the beta2-adrenergic receptor. SAR and QSAR in Environmental Research 21:1-2, pages 37-55.
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Susan E Northfield & David T Manallack. (2007) Lipophilicity of Beta‐Adrenocepter Antagonists: A New Classification Scheme for Clinical Use. Journal of Pharmacy Practice and Research 37:2, pages 98-101.
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Adolf Miklavc & Darko Kocjan. (2004) Entropic Trapping Binding Mechanism:  Its Likely Role in Receptor−Ligand and Other Biochemical Systems. Journal of Chemical Information and Computer Sciences 44:2, pages 422-426.
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Pier Andrea Borea, Alessandro Dalpiaz, Katia Varani, Laura Guerra & Gastone Gilli. (1995) Binding thermodynamics of adenosine A2a receptor ligands. Biochemical Pharmacology 49:4, pages 461-469.
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Robert B. Raffa, Kenneth D. Wild, Henry I. Mosberg & Frank Porreca. (1993) Thermodynamic parameters for [D-Pen2,5]enkephalin at δ-opioid receptors in the mouse isolated vas deferens. European Journal of Pharmacology: Molecular Pharmacology 244:3, pages 231-238.
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Pier Andrea Borea, Leda Montesi, Anna Muzzolini & Roberto Fantozzi. (1991) Temperature dependence of [3H]PAF binding to washed human platelets. Biochemical Pharmacology 41:4, pages 629-630.
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Frank Brady, Sajinder K. Luthra, Henri-J. Tochon-Danguy, Colin J. Steel, Stephen L. Waters, Malcolm J. Kensett, Patricia Landais, Farah Shah, Knut A. Jaeggi, Alex Drake, John C. Clark & Victor W. Pike. (1991) Asymmetric synthesis of a precursor for the automated radiosynthesis of as a preferred radioligand for β-adrenergic receptors. International Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes 42:7, pages 621-628.
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D. J. Prentice, V. J. Barrett, S. J. MacLennan & G. R. Martin. 1991. Serotonin: Molecular Biology, Receptors and Functional Effects. Serotonin: Molecular Biology, Receptors and Functional Effects 161 173 .
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Gábor Náray-SzabÓ. (2009) Electrostatics in computer-aided drug design. International Journal of Quantum Chemistry 36:S16, pages 87-99.
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Robert B. Raffa & Frank Porreca. (1989) Thermodynamic analysis of the drug-receptor interaction. Life Sciences 44:4, pages 245-258.
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Bernard Testa, Peter Jenner, Gavin J. Kilpatrick, Nabil El Tayar, Han Van de Waterbeemd & C.David Marsden. (1987) Do thermodynamic studies provide information on both the binding to and the activation of dopaminergic and other receptors?. Biochemical Pharmacology 36:23, pages 4041-4046.
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