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Journal of Receptor Research Volume 11, 1991 - Issue 1-4
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Research Article

Biologically Active Monoiodinated α-MSH Derivatives for Receptor Binding Studies Using Human Melanoma Cells

Alex N. Eberle Laboratory of Endocrinology, Department of Research (ZLF), University Hospital and University Children's Hospital, CH-4031, Basel, Switzerland
,
Vreni Jäggin Verin Laboratory of Endocrinology, Department of Research (ZLF), University Hospital and University Children's Hospital, CH-4031, Basel, Switzerland
,
Flavio Solca Laboratory of Endocrinology, Department of Research (ZLF), University Hospital and University Children's Hospital, CH-4031, Basel, Switzerland
,
Walter Siegrist Laboratory of Endocrinology, Department of Research (ZLF), University Hospital and University Children's Hospital, CH-4031, Basel, Switzerland
,
Caroline Küenlin Laboratory of Endocrinology, Department of Research (ZLF), University Hospital and University Children's Hospital, CH-4031, Basel, Switzerland
,
Claudia Bagutti Laboratory of Endocrinology, Department of Research (ZLF), University Hospital and University Children's Hospital, CH-4031, Basel, Switzerland
,
Sibylla Stutz Laboratory of Endocrinology, Department of Research (ZLF), University Hospital and University Children's Hospital, CH-4031, Basel, Switzerland
&
Jürg Girard Laboratory of Endocrinology, Department of Research (ZLF), University Hospital and University Children's Hospital, CH-4031, Basel, Switzerland
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Pages 311-322 | Published online: 26 Sep 2008

Citations (33)

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Read on this site (12)

Alex N. Eberle & Gabriele Mild. (2009) Receptor-mediated tumor targeting with radiopeptides. Journal of Receptors and Signal Transduction 29:1, pages 1-37.
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Jarl ES Wikberg. (2001) Melanocortin receptors: new opportunities in drug discovery. Expert Opinion on Therapeutic Patents 11:1, pages 61-76.
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Edith Hintermann, Heidi Tanner, Christiane Talke-Messerer, Sophie Schlumberger, Urs Zumsteg & Alex N. Eberle. (2001) INTERACTION OF MELANIN-CONCENTRATING HORMONE (MCH), NEUROPEPTIDE E-I (NEI), NEUROPEPTIDE G-E (NGE), AND α-MSH WITH MELANOCORTIN AND MCH RECEPTORS ON MOUSE B16 MELANOMA CELLS. Journal of Receptors and Signal Transduction 21:1, pages 93-116.
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Alex N. Eberle, Jószef Bódi, György Orosz, Helga Süli-Vargha, Verena Jäggin & Urs Zumsteg. (2001) ANTAGONIST AND AGONIST ACTIVITIES OF THE MOUSE AGOUTI PROTEIN FRAGMENT (91–131) AT THE MELANOCORTIN-1 RECEPTOR. Journal of Receptors and Signal Transduction 21:1, pages 25-45.
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Yves Brandenburger, Keith Rose, Claudia Bagutti & Alex N. Eberle. (1999) Synthesis and Receptor Binding Analysis of Thirteen Oligomeric α-MSH Analogs. Journal of Receptors and Signal Transduction 19:1-4, pages 467-480.
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G. Heizmann, P. Hildebrand, H. Tanner, S. Ketterer, A. Pansky, S. Froidevaux, C. Beglinger & A. N. Eberle. (1999) A Combinatorial Peptoid Library for the Identification of Novel MSH and GRP / Bombesin Receptor Ligands. Journal of Receptors and Signal Transduction 19:1-4, pages 449-466.
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E. Hintermann, R. Drozdz, H. Tanner & A. N. Eberle. (1999) Synthesis and Characterization of New Radioligands for the Mammalian Melanin-Concentrating Hormone (MCH) Receptor. Journal of Receptors and Signal Transduction 19:1-4, pages 411-422.
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S. Froidevaux, M. Meier, M. Häusler, H. Mäcke, C. Beglinger & A. N. Eberle. (1999) A Microplate Binding Assay for the Somatostatin Type-2 Receptor (SSTR2). Journal of Receptors and Signal Transduction 19:1-4, pages 167-180.
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Walter Siegrist, Roma Drozdz, Renato Cotti, Derril H. Willard, William O. Wilkison & Alex N. Eberle. (1997) Interactions of α-Melanotropin and Agouti on B16 Melanoma Cells: Evidence for Inverse Agonism of Agouti. Journal of Receptors and Signal Transduction 17:1-3, pages 75-98.
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Claudia Bagutti, Marc Oestreicher, Walter Siegrist, Martin Oberholzer & Alex N. Eberle. (1995) α-MSH Receptor Autoradiography on Mouse and Human Melanoma Tissue Sections and Biopsies. Journal of Receptors and Signal Transduction 15:1-4, pages 427-442.
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Walter Siegrist & Alex N. Eberle. (1993) Homologous Regulation of the MSH Receptor in Melanoma Cells. Journal of Receptor Research 13:1-4, pages 263-281.
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Claudia Bagutti & Alex N. Eberle. (1993) Synthesis and Biological Properties of a Biotinylated Derivative of Acth1-17 for MSH Receptor Studies. Journal of Receptor Research 13:1-4, pages 229-244.
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Articles from other publishers (21)

Maria Cristina Oliveira & João D.G. Correia. (2019) Biomedical applications of radioiodinated peptides. European Journal of Medicinal Chemistry 179, pages 56-77.
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Feng Gao, Wiebke Sihver, Ralf Bergmann, Martin Walther, Holger Stephan, Birgit Belter, Christin Neuber, Cathleen Haase-Kohn, Cristina Bolzati, Jens Pietzsch & Hans-Jürgen Pietzsch. (2019) Radiochemical and radiopharmacological characterization of a 64 Cu-labeled α-MSH analog conjugated with different chelators . Journal of Labelled Compounds and Radiopharmaceuticals 62:8, pages 495-509.
Crossref
Feng Gao, Wiebke Sihver, Ralf Bergmann, Birgit Belter, Cristina Bolzati, Nicola Salvarese, Jörg Steinbach, Jens Pietzsch & Hans-Jürgen Pietzsch. (2018) Synthesis, Characterization, and Initial Biological Evaluation of [ 99m Tc]Tc-Tricarbonyl-labeled DPA-α-MSH Peptide Derivatives for Potential Melanoma Imaging . ChemMedChem 13:11, pages 1146-1158.
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Feng Gao, Wiebke Sihver, Christoph Jurischka, Ralf Bergmann, Cathleen Haase-Kohn, Birgit Mosch, Jörg Steinbach, Davide Carta, Cristina Bolzati, Andrea Calderan, Jens Pietzsch & Hans-Jürgen Pietzsch. (2015) Radiopharmacological characterization of 64Cu-labeled α-MSH analogs for potential use in imaging of malignant melanoma. Amino Acids 48:3, pages 833-847.
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Molly E. Martin, M. Sue O’Dorisio, Whitney M. Leverich, Kyle C. Kloepping, Susan A. Walsh & Michael K. Schultz. 2013. Theranostics, Gallium-68, and Other Radionuclides. Theranostics, Gallium-68, and Other Radionuclides 149 175 .
Nicholas J. Baumhover, Molly E. Martin, Sharavathi G. Parameswarappa, Kyle C. Kloepping, M. Sue O’Dorisio, F. Christopher Pigge & Michael K. Schultz. (2011) Improved synthesis and biological evaluation of chelator-modified α-MSH analogs prepared by copper-free click chemistry. Bioorganic & Medicinal Chemistry Letters 21:19, pages 5757-5761.
Crossref
Yubin Miao & Thomas P. Quinn. (2008) Peptide-targeted radionuclide therapy for melanoma. Critical Reviews in Oncology/Hematology 67:3, pages 213-228.
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Alex N. Eberle & Sylvie Froidevaux. (2003) Radiolabeled ?-melanocyte-stimulating hormone analogs for receptor-mediated targeting of melanoma: from tritium to indium. Journal of Molecular Recognition 16:5, pages 248-254.
Crossref
Alex N. Eberle. 2000. The Melanocortin Receptors. The Melanocortin Receptors 3 67 .
Roma Drozdz, Edith Hintermann, Heidi Tanner, Urs Zumsteg & Alex N. Eberle. (1999) [D-(p-Benzoylphenylalanine)13, tyrosine19]-melanin-concentrating hormone, a potent analogue for MCH receptor crosslinking. Journal of Peptide Science 5:5, pages 234-242.
Crossref
Mauro Vallarino, Michele Trabucchi, Nicolas Chartrel, Verena J�ggin, Alex N. Eberle & Hubert Vaudry. (1998) Melanin-concentrating hormone system in the brain of the lungfishProtopterus annectens. The Journal of Comparative Neurology 390:1, pages 41-51.
Crossref
Ganesan Vaidyanathan & Michael R. Zalutsky. (1997) Fluorine-18-labeled [Nle4,d-Phe7]-α-MSH, an α-melanocyte stimulating hormone analogue. Nuclear Medicine and Biology 24:2, pages 171-178.
Crossref
Johanna Chluba-de Tapia, Claudia Bagutt, Renato Cotti & Alex N. Eberle. (1996) Induction of constitutive melanogenesis in amelanotic mouse melanoma cells by transfection of the human melanocortin-1 receptor gene. Journal of Cell Science 109:8, pages 2023-2030.
Crossref
Walter Lichtensteiger, Beatrice Hanimann, Walter Siegrist & Alex N. Eberle. (1996) Region- and stage-specific patterns of melanocortin receptor ontogeny in rat central nervous system, cranial nerve ganglia and sympathetic ganglia. Developmental Brain Research 91:1, pages 93-110.
Crossref
Roma Drozdz, Walter Siegrist, Bridget I. Baker, Johanna Chluba-de Tapia & Alex N. Eberle. (1995) Melanin-concentrating hormone binding to mouse melanoma cells in vitro. FEBS Letters 359:2-3, pages 199-202.
Crossref
R. Drozdz, B. I. Baker & A. N. Eberle. 1995. Peptides 1994. Peptides 1994 785 786 .
Roma Drozdz & Alex N. Eberle. (2004) Synthesis and lodination of human (phenylalanine 13 , tyrosine 19 ) melanin‐concentrating hormone for radioreceptor assay . Journal of Peptide Science 1:1, pages 58-65.
Crossref
J.B. Dietrich, P. Hildebrand, L.Baselgia Jeker, A. Pansky, A.N. Eberle & C. Beglinger. (1994) Effects of BIM26226, a potent and specific bombesin receptor antagonist, on amylase release and binding of bombesin-like peptides to AR4-2J cells. Regulatory Peptides 53:3, pages 165-173.
Crossref
Claudia Bagutti, Barbara Stolz, Rainer Albert, Christian Bruns, Janos Pless & Alex N. Eberle. (1994) [111In]-DTPA-labeled analogues of α-melanocyte-stimulating hormone for melanoma targeting: Receptor bindingin vitro andin vivo. International Journal of Cancer 58:5, pages 749-755.
Crossref
ALEX N. EBERLE, WALTER SIEGRIST, CLAUDIA BAGUTTI, JOHANNA CHLUBA-DE TAPIA, FLAVIO SOLCA, JARL E. S. WIKBERG & VIJAY CHHAJLANI. (1993) Receptors for Melanocyte-Stimulating Hormone on Melanoma Cells. Annals of the New York Academy of Sciences 680:1 The Melanotro, pages 320-341.
Crossref
W. Siegrist, C. Bagutti, F. Solca, J. Girard & A.N. Eberle. (1992) 3.5 MSH receptors on mouse and human melanoma cells: receptor identification, analysis and quantification. Progress in Histochemistry and Cytochemistry 26:1-4, pages 110-118.
Crossref

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