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Haytham O. Tawfik, Amany Belal, Mohammed A. S. Abourehab, Andrea Angeli, Alessandro Bonardi, Claudiu T. Supuran & Mervat H. El-Hamamsy. (2022) Dependence on linkers’ flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 2765-2785.
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Claudiu T. Supuran. (2018) Carbonic anhydrase inhibitors as emerging agents for the treatment and imaging of hypoxic tumors. Expert Opinion on Investigational Drugs 27:12, pages 963-970.
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Ahmed Fekri & Eman M. Keshk. (2016) Utility involving thioacetoacetanilides as precursors for synthesis of new thiazole, thiadiazole and thiophene derivatives with antimicrobial activity. Journal of Sulfur Chemistry 37:2, pages 148-161.
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Salwa M. I. Morsy, Abdelfattah M. Badawi, Alessandro Cecchi, Andrea Scozzafava & Claudiu T. Supuran. (2009) Carbonic anhydrase inhibitors. Biphenylsulfonamides with inhibitory action towards the transmembrane, tumor-associated isozymes IX possess cytotoxic activity against human colon, lung and breast cancer cell lines. Journal of Enzyme Inhibition and Medicinal Chemistry 24:2, pages 499-505.
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Arabinda Das, Naren L. Banik & Swapan K. Ray. (2008) Modulatory Effects of Acetazolomide and Dexamethasone on Temozolomide Mediated Apoptosis in Human Glioblastoma T98G and U87MG Cells. Cancer Investigation 26:4, pages 352-358.
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Muhammad Zareef, Rashid Iqbal, NajimA. Al-Masoudi, JavidH. Zaidi, Muhammad Arfan & SohailA. Shahzad. (2007) Synthesis, Anti–HIV, and Antifungal Activity of New Benzensulfonamides Bearing the 2,5-Disubstituted-1,3,4-Oxadiazole Moiety. Phosphorus, Sulfur, and Silicon and the Related Elements 182:2, pages 281-298.
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Muhammad Zareef, Alessio Innocenti, Rashid Iqbal, Javid H. Zaidi, Muhammad Arfan, Andrea Scozzafava & Claudiu T. Supuran. (2006) Carbonic anhydrase inhibitors. Inhibition of human tumor-associated isozymes IX and cytosolic isozymes I and II with some 1,3,4-oxadiazole-thiols. Journal of Enzyme Inhibition and Medicinal Chemistry 21:4, pages 351-359.
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. (2004) Carbonic anhydrase/COX-2 inhibitors in the treatment of various diseases. Expert Opinion on Therapeutic Patents 14:12, pages 1803-1806.
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Silvia Pastorekova, Seppo Parkkila, Jaromir Pastorek & Claudiu T. Supuran. (2004) Review Article. Journal of Enzyme Inhibition and Medicinal Chemistry 19:3, pages 199-229.
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Marco Franchi, Daniela Vullo, Enzo Gallori, Jaromir Pastorek, Antonella Russo, Andrea Scozzafava, Silvia Pastorekova & Claudiu T. Supuran. (2003) Carbonic Anhydrase Inhibitors. Inhibition of Cytosolic Isozymes I and II and Transmembrane, Cancer-associated Isozyme IX with Lipophilic Sulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 18:4, pages 333-338.
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Carsten Uhd Nielsen, Birger Brodin, Flemming Steen Jørgensen, Sven Frokjaer & Bente Steffansen. (2002) Human peptide transporters: therapeutic applications. Expert Opinion on Therapeutic Patents 12:9, pages 1329-1350.
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Claudiu T Supuran & Andrea Scozzafava. (2002) Applications of carbonic anhydrase inhibitors and activators in therapy. Expert Opinion on Therapeutic Patents 12:2, pages 217-242.
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Haytham O. Tawfik, Andrea Petreni, Claudiu T. Supuran & Mervat H. El-Hamamsy. (2022) Discovery of new carbonic anhydrase IX inhibitors as anticancer agents by toning the hydrophobic and hydrophilic rims of the active site to encounter the dual-tail approach. European Journal of Medicinal Chemistry 232, pages 114190.
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Nathaniel H. Boyd, Kiera Walker, Joshua Fried, James R. Hackney, Paul C. McDonald, Gloria A. Benavides, Raffaella Spina, Alessandra Audia, Sarah E. Scott, Catherine J. Libby, Anh Nhat Tran, Mark O. Bevensee, Corinne Griguer, Susan Nozell, G. Yancey Gillespie, Burt Nabors, Krishna P. Bhat, Eli E. Bar, Victor Darley-Usmar, Bo Xu, Emily Gordon, Sara J. Cooper, Shoukat Dedhar & Anita B. Hjelmeland. (2017) Addition of carbonic anhydrase 9 inhibitor SLC-0111 to temozolomide treatment delays glioblastoma growth in vivo. JCI Insight 2:24.
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Mohamad Yusuf & Payal Jain. (2014) Synthesis and biological significances of 1,3,4-thiadiazolines and related heterocyclic compounds. Arabian Journal of Chemistry 7:5, pages 525-552.
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Diego M. Gil, Oscar E. Piro, Gustavo A. Echeverría, María E. Tuttolomondo & Aída Ben Altabef. (2013) Layered crystal structure, conformational and vibrational properties of 2,2,2-trichloroethoxysulfonamide: An experimental and theoretical study. Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy 116, pages 122-131.
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Harun M. Said, Carsten Hagemann, Fabrizio Carta, Astrid Katzer, Bülent Polat, Adrian Staab, Andrea Scozzafava, Jelena Anacker, Giles H. Vince, Michael Flentje & Claudiu T. Supuran. (2013) Hypoxia induced CA9 inhibitory targeting by two different sulfonamide derivatives including Acetazolamide in human Glioblastoma. Bioorganic & Medicinal Chemistry 21:13, pages 3949-3957.
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K. Sarojini, H. Krishnan, Charles C. Kanagam & S. Muthu. (2013) Molecular Structure, Vibrational Spectroscopy and Homo, Lumo Studies of 4-methyl-N-(2-methylphenyl) Benzene Sulfonamide Using DFT Method. Advanced Materials Research 665, pages 101-111.
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K. Sarojini, H. Krishnan, Charles C. Kanakam & S. Muthu. (2012) Synthesis, X-ray structural, characterization, NBO and HOMO–LUMO analysis using DFT study of 4-methyl-N-(naphthalene-1-yl)benzene sulfonamide. Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy 96, pages 657-667.
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Paul C. McDonald, Jean-Yves Winum, Claudiu T. Supuran & Shoukat Dedhar. (2012) Recent Developments in Targeting Carbonic Anhydrase IX for Cancer Therapeutics. Oncotarget 3:1, pages 84-97.
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Narges K. Tafreshi, Marilyn M. Bui, Kellsey Bishop, Mark C. Lloyd, Steven A. Enkemann, Alexis S. Lopez, Dominique Abrahams, Bradford W. Carter, Josef Vagner, Stephen R. Grobmyer, Robert J. Gillies & David L. Morse. (2012) Noninvasive Detection of Breast Cancer Lymph Node Metastasis Using Carbonic Anhydrases IX and XII Targeted Imaging Probes. Clinical Cancer Research 18:1, pages 207-219.
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Gilles MeesChristel VangestelRudi DierckxPatrick PauwelsJan Van MeerbeeckChristophe Van de Wiele. (2010) Carbonic Anhydrase IX Expression Correlates with FDG Uptake by Primary Non–Small Cell Lung Cancer. Cancer Biotherapy and Radiopharmaceuticals 25:2, pages 149-154.
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Islam Ullah Khan, Ghulam Mustafa, Muhammad Nadeem Arshad, Muhammad Shafiq & Shahzad Sharif. (2009) 4-(4-Bromobenzenesulfonamido)benzoic acid. Acta Crystallographica Section E Structure Reports Online 65:5, pages o1073-o1073.
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Steven Blake, Ricardo Capone, Michael Mayer & Jerry Yang. (2008) Chemically Reactive Derivatives of Gramicidin A for Developing Ion Channel-Based Nanoprobes. Bioconjugate Chemistry 19:8, pages 1614-1624.
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Anne Thiry, Claudiu T. Supuran, Bernard Masereel & Jean-Michel Dogné. (2008) Recent Developments of Carbonic Anhydrase Inhibitors as Potential Anticancer Drugs. Journal of Medicinal Chemistry 51:11, pages 3051-3056.
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Claudiu T Supuran. (2007) Therapeutic applications of the carbonic anhydrase inhibitors. Therapy 4:3, pages 355-378.
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Alexander Hillebrecht, Claudiu T. Supuran & Gerhard Klebe. (2006) Integrated Approach Using Protein and Ligand Information to Analyze Selectivity- and Affinity-Determining Features of Carbonic Anhydrase Isozymes. ChemMedChem 1:8, pages 839-853.
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R. Iqbal, M. Zareef, S. Ahmed, J. H. Zaidi, M. Arfan, M. Shafique & N. A. Al-Masoudi. (2006) Synthesis, Antimicrobial and Anti-HIV Activity of Some Novel Benzenesulfonamides Bearing 2,5-Disubstituted-1,3,4-Oxadiazole Moiety. Journal of the Chinese Chemical Society 53:3, pages 689-696.
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Daniel Edmund Bryan Swinson & Kenneth John O'Byrne. (2006) Interactions Between Hypoxia and Epidermal Growth Factor Receptor in Non–Small-Cell Lung Cancer. Clinical Lung Cancer 7:4, pages 250-256.
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Sally-Ann Poulsen, Laurent F. Bornaghi & Peter C. Healy. (2005) Synthesis and structure–activity relationships of novel benzene sulfonamides with potent binding affinity for bovine carbonic anhydrase II. Bioorganic & Medicinal Chemistry Letters 15:24, pages 5429-5433.
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Özen Özensoy, Luca Puccetti, Giuseppe Fasolis, Oktay Arslan, Andrea Scozzafava & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors: Inhibition of the tumor-associated isozymes IX and XII with a library of aromatic and heteroaromatic sulfonamides. Bioorganic & Medicinal Chemistry Letters 15:21, pages 4862-4866.
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Alessio Innocenti, Raquel Villar, Victor Martinez-Merino, María J. Gil, Andrea Scozzafava, Daniela Vullo & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors: Inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with benzo[b]thiophene 1,1-dioxide sulfonamides. Bioorganic & Medicinal Chemistry Letters 15:21, pages 4872-4876.
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Alexandru T. Balaban, Padmakar V. Khadikar, Claudiu T. Supuran, Abhilash Thakur & Mamta Thakur. (2005) Study on supramolecular complexing ability vis-à-vis estimation of pKa of substituted sulfonamides: Dominating role of Balaban index (J). Bioorganic & Medicinal Chemistry Letters 15:17, pages 3966-3973.
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Jean-Yves Winum, Alessio Innocenti, Jihane Nasr, Jean-Louis Montero, Andrea Scozzafava, Daniela Vullo & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with N-hydroxysulfamides—a new zinc-binding function in the design of inhibitors. Bioorganic & Medicinal Chemistry Letters 15:9, pages 2353-2358.
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Yun-Hee Kim, Kum-Joo Shin, Taehoon G. Lee, Euikyung Kim, Myoung-Shik Lee, Sung Ho Ryu & Pann-Ghill Suh. (2005) G2 arrest and apoptosis by 2-amino-N-quinoline-8-yl-benzenesulfonamide (QBS), a novel cytotoxic compound. Biochemical Pharmacology 69:9, pages 1333-1341.
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Hasan Turkmen, Mustafa Durgun, Serpil Yilmaztekin, Mahmut Emul, Alessio Innocenti, Daniela Vullo, Andrea Scozzafava & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors. Novel sulfanilamide/acetazolamide derivatives obtained by the tail approach and their interaction with the cytosolic isozymes I and II, and the tumor-associated isozyme IX. Bioorganic & Medicinal Chemistry Letters 15:2, pages 367-372.
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Daniela Vullo, Marco Franchi, Enzo Gallori, Jaromir Pastorek, Andrea Scozzafava, Silvia Pastorekova & Claudiu T Supuran. (2003) Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with aromatic and heterocyclic sulfonamides. Bioorganic & Medicinal Chemistry Letters 13:6, pages 1005-1009.
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Claudiu T. Supuran, Andrea Scozzafava & Angela Casini. (2002) Carbonic anhydrase inhibitors. Medicinal Research Reviews 23:2, pages 146-189.
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Leon Margolin. (2003) Severe Psoriasis Palmaris et Plantaris Associated with Topical Use of Dorzolamide. Clinical Drug Investigation 23:7, pages 487-489.
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K.J O'Byrne, G Cox, D Swinson, D Richardson, J.G Edwards, J Lolljee, A Andi, M.I Koukourakis, A Giatromanolaki, K Gatter, A.L Harris, D Waller & J.L Jones. (2001) Towards a biological staging model for operable non-small cell lung cancer. Lung Cancer 34, pages S83-S89.
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Sofia Svedhem, Karin Enander, Martin Karlsson, Hans Sjöbom, Bo Liedberg, Stefan Löfås, Lars-Göran Mårtensson, Sven Erik Sjöstrand, Stefan Svensson, Uno Carlsson & Ingemar Lundström. (2001) Subtle Differences in Dissociation Rates of Interactions between Destabilized Human Carbonic Anhydrase II Mutants and Immobilized Benzenesulfonamide Inhibitors Probed by a Surface Plasmon Resonance Biosensor. Analytical Biochemistry 296:2, pages 188-196.
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