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Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 50, 2020 - Issue 19
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Articles

Synthesis and antibacterial activity of hydroxylated 2-arylbenzothiazole derivatives

Yordan Stremskia Department of Organic Chemistry, University of Plovdiv “Paisii Hilendarski”, Plovdiv, BulgariaCorrespondence[email protected] [email protected]
ORCID Iconhttps://orcid.org/0000-0001-8665-3130View further author information
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Desislava Kirkovaa Department of Organic Chemistry, University of Plovdiv “Paisii Hilendarski”, Plovdiv, Bulgaria;b Tobacco and Tobacco Products Institute, Chemistry of Tobacco and Tobacco Smoke, Markovo, Plovdiv, BulgariaORCID Iconhttps://orcid.org/0000-0001-5394-0109View further author information
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Stela Statkova-Abeghea Department of Organic Chemistry, University of Plovdiv “Paisii Hilendarski”, Plovdiv, BulgariaCorrespondence[email protected] [email protected]
ORCID Iconhttps://orcid.org/0000-0002-3833-6779View further author information
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Plamen Angelova Department of Organic Chemistry, University of Plovdiv “Paisii Hilendarski”, Plovdiv, BulgariaORCID Iconhttps://orcid.org/0000-0002-3625-9933View further author information
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Iliyan Ivanova Department of Organic Chemistry, University of Plovdiv “Paisii Hilendarski”, Plovdiv, BulgariaORCID Iconhttps://orcid.org/0000-0002-4662-3735View further author information
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Danail Georgievc Department of Biochemistry and Microbiology, University of Plovdiv “Paisii Hilendarski”, Plovdiv, BulgariaORCID Iconhttps://orcid.org/0000-0002-8518-611XView further author information
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Pages 3007-3015 | Received 07 Apr 2020, Published online: 14 Jul 2020
 
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Abstract

N-acyliminium reagents formed in situ from benzothiazole and alkyl chloroformates react with hydroxyarenes in a Friedel-Crafts manner, providing access to 2-(hydroxyaryl)-benzothiazolines with antibacterial properties.

Graphical Abstract

Acknowledgement

The authors are grateful to the Faculty of Biology, Department of Plant Physiology and Molecular Biology and Dr. Mladen Naydenov for carrying out high resolution mass spectral measurements on equipment provided under the EC FP7/REGPOT-2009-1/BioSupport project.

Additional information

Funding

This research was funded by the Bulgarian National Science Fund [Grant DN09/15‐2016] and the University of Plovdiv [Grant MU19-HF-012]. Yordan Stremski and Desislava Kirkova thank the Ministry of Education and Science for financial support under National Program “Young Scientists and Postdoctoral Researchers” [PMC 577/2018].

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