Figures & data
Scheme 1. Preparation of 2,4-dioxothiazolidinyl acetic acids 3a–3g.
Table 1. CA inhibitory activity of carboxylates 3a–3g and standard sulphonamide inhibitor acetazolamide AAZ, by a stopped-flow CO2 hydrase assayCitation45.
Journal of Enzyme Inhibition and Medicinal Chemistry
Volume 35, 2020 - Issue 1
Short Communication
A class of carbonic anhydrase IX/XII – selective carboxylate inhibitors
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Claudiu T. Supuranb Dipartimento Neurofarba, Sezione di Scienze Farmaceutiche e Nutraceutiche, Università degli Studi di Firenze, Florence, ItalyCorrespondence[email protected]
https://orcid.org/0000-0003-4262-0323
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