Abstract
New water soluble 1-vinylsulfonyl-2-arylpyrrolidine derivatives were obtained through aza-Michael reaction of 4-chloro-6-[1-(vinylsulfonyl)pyrrolidin-2-yl]benzene-1,3-diol with secondary aminophosphonates in water-ethanol medium in the presence of triethylamine.
Graphical Abstract
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