Abstract
The synthesis of 4‐alkyl‐2‐arylmorpholin‐2‐ol hydrochlorides by diastereoselective reaction of 2‐bromoacetophenones with β‐aminoalcohols has been accomplished.
Acknowledgments
The authors wish to thank to “Consejo Nacional de Ciencia y Tecnologìa” (Conacyt, México) for financial support and scholarship to Luis S. Zamudio‐Rivera. We thank Dr. Rosa Luisa Santillan for reading the manuscript and for her helpful comments.