1,023
Views
26
CrossRef citations to date
0
Altmetric
Original Articles

Synthesis and evaluation of antimicrobial, antitubercular and anticancer activities of benzimidazole derivatives

, , , , , & show all
Pages 100-109 | Received 08 Jul 2017, Accepted 05 Nov 2017, Published online: 06 Mar 2019

References

  • S.S.MorseFactors in the emergence of infectious diseasesEmerg Infect Dis11995715
  • Kent MM, Yin S. Controlling infectious diseases. Popul Bull 2006; 61: 1–20.
  • N.GautamA.GargA.K.BishnoiS.AgarwalD.C.GautamAntioxidant and antimicrobial assessment of synthesized and spectrally characterized new nitrophenothiazines and their sulfone analoguesPhosphorus Sulfur Silicon Relat Elem1902015528536
  • H.W.HethcoteThe mathematics of infectious diseasesSIAM Rev422000599653
  • J.CamachoA.BarazarteN.GamboaJ.RodriguesR.RojasA.Vaisberget al.Synthesis and biological evaluation of benzimidazole-5-carbohydrazide derivatives as antimalarial cytotoxic and antitubercular agentsBioorg Med Chem19201120232029
  • P.PrakashB.ArunaA.A.SardesaiS.E.HasnainPurified recombinant hypothetical protein coded by open reading frame Rv1885c of Mycobacterium tuberculosis exhibits a monofunctional aroq class of periplasmic chorismate mutase activityJ Biol Chem28020051964119648
  • H.AgarwalA.KumarN.C.BalM.I.SiddiqiA.AroraLigand based virtual screening and biological evaluation of inhibitors of chorismate mutase (Rv1885c) from Mycobacterium tuberculosis H37RvBioorg Med Chem Lett17200730533058
  • A.AroraN.R.ChandraA.DasB.GopalS.C.MandeB.Prakashet al.Structural biology of Mycobacterium tuberculosis proteins: the Indian effortsTuberculosis912011456468
  • H.GuoN.RaoChorismate-mutase catalysed Claisen rearrangementU.NubbemeyerM.HiersemannThe Claisen Rearrangement- Methods and applications2007Wiley-VCH Verlag GmbH & Co. KGaAWeinheim123
  • J.M.LiN.LiD.Y.ZhuL.G.WanY.L.HeC.YangIsocitrate lyase from Mycobacterium Tuberculosis promotes survival of Mycobacterium Smegmatis within macrophage by suppressing cell apoptosisChin Med J121200811141119
  • V.C.C.UyJ.B.BillonesTowards antituberculosis drugs: virtual screening for potential inhibitors of pantothenate synthetase of Mycobacterium tuberculosisPhilipp Sci Lett52012122130
  • American Cancer SocietyBreast Cancer Facts & Figures 2015–20162015American Cancer Society, Inc.Atlanta138
  • J.B.WrightThe chemistry of the benzimidazolesChem Rev481951397541
  • C.H.SrideviK.BalajiA.NaiduR.SudhakaranSynthesis of some phenylpyrazolo benzimidazolo quinoxaline derivatives as potent antihistaminic agentsE- J Chem (online)72010234238
  • P.K.RanjithP.RajeeshK.R.HaridasN.K.SusantaT.N.RowR.Rishikesanet al.Design and synthesis of positional isomers of 5 and 6-bromo-1-[(phenyl)sulfonyl]-2-[(4-nitrophenoxy)methyl]-1H-benzimidazoles as possible antimicrobial and antitubercular agentsBioorg Med Chem Lett23201352285234
  • R.K.AroraN.KaurY.BansalG.BansalNovel coumarin-benzimidazole derivatives as antioxidants and safer anti-inflammatory agentsActa Pharm Sin B42014368375
  • T.PanX.HeB.ChenH.ChenG.GengH.Luoet al.Development of benzimidazole derivatives to inhibit HIV-1 replication through protecting APOBEC3G proteinEur J Med Chem952015500513
  • K.VasanthaG.BasavarajaswamyM.V.RaiP.BojaV.R.PaiN.Shruthiet al.Rapid ‘one-pot’ synthesis of a novel benzimidazole-5-carboxylate and its hydrazone derivatives as potential anti-inflammatory and antimicrobial agentsBioorg Med Chem Lett25201514201426
  • M.GabaP.GabaD.UppalN.DhingraM.S.BahiaO.Silakariet al.Benzimidazole derivatives: search for GI-friendly anti-inflammatory analgesic agentsActa Pharm Sin B52015337342
  • J.WenY.LuoH.ZhangH.ZhaoC.ZhouG.CaiA green and convenient approach toward benzimidazole derivatives and their antimicrobial activityChin Chem Lett272016391394
  • R.S.KeriA.HiremathadS.BudagumpiB.M.NagarajaComprehensive review in current developments of benzimidazole-based medicinal chemistryChem Biol Drug Des862015196510.1111/cbdd.12462
  • Y.BansalO.SilakariThe therapeutic journey of benzimidazoles: a reviewBioorg Med Chem20201262086236
  • S.YadavB.NarasimhanH.KaurPerspectives of benzimidazole derivatives as anticancer agents in the new eraAnticancer Agents Med Chem16201614031425
  • R.A.HaqueS.BudagumpiS.Y.ChooM.K.ChoongB.E.LokeshK.SudeshNitrile-functionalized Hg(II)- and Ag(I)-N-heterocyclic carbene complexes: synthesis, crystal structures, nuclease and DNA binding activitiesAppl Organometal Chem262012689700
  • K.F.AnsariC.LalSynthesis physicochemical properties and antimicrobial activity of some new benzimidazole derivativesEur J Med Chem44200940284033
  • S.YadavP.KumarE.D.ClercqJ.BalzariniC.PannecouqueS.K.Dewanet al.4-[1-(Substituted aryl/alkyl carbonyl)-benzoimidazol-2-yl]-benzenesulfonic acids: synthesis, antimicrobial activity, QSAR studies, and antiviral evaluationEur J Med Chem45201059855997
  • J.G.CappucinoN.ShermanMicrobiology: a laboratory mannual1999Addison Wesley Longman IncCalifornia263
  • Pharmacopoeia of India, vol. II. Ministry of Health Department New Delhi: Govt. of India; 1996; p. A-88.
  • M.C.Rodriguez-ArguellesE.C.Lopez-SilvaJ.SanmartinP.PelagattiF.ZaniCopper complexes of imidazole-2-pyrrole-2- and indol-3-carbaldehyde thiosemicarbazones: inhibitory activity against fungi and bacteriaJ Inorg Biochem99200522312239
  • Parish T, Stroker NG. Mycobacteria Protocols: Methods in molecular Biology. (Vol. 101) Totowa NJ: Humana Press Totowa; 1998, p. 395–422.
  • L.A.CollinsS.G.FranzblauMicroplate alamar blue assay versus BACTEC 460 system for high-throughput screening of compounds against Mycobacterium tuberculosis and Mycobacterium aviumAntimicrob Agents Chemother41199710041009
  • C.KirimuhuzyaP.WaakoM.JolobaO.OdyekThe antimycobacterial activity of Lantana camara a plant traditionally used to treat symptoms of tuberculosis in South-western UgandaAfr Health Sci920094045
  • C.PerezC.AnesiniIn vitro antimicrobial activity of Argentine folk medicinal plants against Salmonella typhiiJ Ethnopharmacol4419944146
  • M.J.SanjayNatural products: an important source for antitubercular drugsCRISP520041
  • L.TonaK.KambuN.NgimbiK.CimangaA.J.VlietinckAntiamoebic and phytochemical screening of some Congolese medicinal plantsJ Ethnopharmacol6119985765
  • G.H.DixonH.L.KornbergAssay methods for key enzymes of the glyoxylate cycleBiochem J7219593P
  • M.KratkyJ.VinaovaN.G.RodriguezJ.StolarikovaAntimycobacterial activity of salicylanilide benzenesulfonatesMolecules172013492503
  • S.SamalaP.B.DeviR.NallangiP.YogeeswariD.SriramDevelopment of 3-phenyl-4,5,6,7-tetrahydro-1??-pyrazolo[4,3-c]pyridine derivatives as novel Mycobacterium tuberculosis pantothenate synthetase inhibitorsEur J Med Chem692013356364
  • S.WangD.EisenbergCrystal structures of a pantothenate synthetase from M. tuberculosis and its complexes with substrates and a reaction intermediateProtein Sci12200310971108
  • R.AdepuK.Shiva KumarS.SandraD.RambabuG.Rama KrishnaC.Malla Reddyet al.C-N bond formation under Cu-catalysis: synthesis and in vitro evaluation of N-aryl substituted thieno[2,3-d]pyrimidin-4-(3H)-ones against chorismate mutaseBioorg Med Chem20201251275138
  • P.SkehanR.StorengD.ScudieroA.MonksJ.McMahonD.Visticaet al.New colorimetric cytotoxicity assay for anticancer-drug screeningJ Natl Cancer Inst82199011071112
  • K.M.HosamaniR.V.ShingalapurSynthesis of 2-mercaptobenzimidazole derivatives as potential anti-microbial and cytotoxic agentsArch Pharm (Weinheim)3442011311319
  • A.K.ZainabSynthesis of some new 1, 2, 4-triazoles derived from 2-mercaptobenzimidazoleUm-Salama Sci J62009200208
  • Budeanu CH, Rusu G, Cojocaru Z, Nistor, C. Investigations on a series of five-membered nitrogen heterocycles. Synthesis of some new benzimidazolyl-2-mercaptoacetohydrazidehydrazones and testing of their cytostatic action on experimental tumors. Revista Medico-Chirurgicala 1976; 80: 605–9.
  • S.EmamiM.FalhatiA.BanifafemiA.ShafieeStereoselective synthesis and antifungal activity of (Z)-trans-3-azolyl-2-methylchromanone oxime ethersBioorg Med Chem12200458815889