Solubility of budesonide in {ethanol + water} mixtures from T = (293.2 to 313.2) K: Experimental measurement and mathematical modelling

References

• Johansson SÅ, Andersson KE, Brattsand R, et al. Topical and systemic glucocorticoid potencies of budesonide and beclomethasone dipropionate in man. Eur J Clin Pharmacol. 1982;22:523–529.
   PubMed Web of Science ®Google Scholar
• Juniper EF, Kline PA, Vanzieleghem MA, et al. Effect of long-term treatment with an inhaled corticosteroid (budesonide) on airway hyperresponsiveness and clinical asthma in nonsteroid-dependent asthmatics. Am Rev Respir Dis. 1990;142:832–836.
   PubMed Web of Science ®Google Scholar
• Hvizdos KM, Jarvis B. Budesonide inhalation suspension. Drugs. 2000;60:1141–1178.
   PubMed Web of Science ®Google Scholar
• Spencer CM, McTavish D. Budesonide. Drugs. 1995;50:854–872.
   PubMed Web of Science ®Google Scholar
• Dalby C, Polanowski T, Larsson T, et al. The bioavailability and airway clearance of the steroid component of budesonide/formoterol and salmeterol/fluticasone after inhaled administration in patients with COPD and healthy subjects: a randomized controlled trial. Respir Res. 2009;10:104–115.
   PubMed Web of Science ®Google Scholar
• Di L, Fish PV, Mano T. Bridging solubility between drug discovery and development. Drug Discov Today. 2012;17:486–495.
   PubMed Web of Science ®Google Scholar
• Strickley RG. Solubilizing excipients in oral and injectable formulations. Pharm Res. 2004;21:201–230.
   PubMed Web of Science ®Google Scholar
• Alsenz J, Kansy M. High throughput solubility measurement in drug discovery and development. Adv Drug Delivery Rev. 2007;59:546–567.
   PubMed Web of Science ®Google Scholar
• Khan AD, Singh L. Various techniques of bioavailability enhancement: a review. J Drug Deliv. 2016;6:34–41.
   Google Scholar
• Shayanfar A, Fakhree MAA, Acree WE Jr, et al. Solubility of lamotrigine, diazepam, and clonazepam in ethanol + water mixtures at 298.15 K. J Chem Eng Data. 2008;54:1107–1109.
   Web of Science ®Google Scholar
• Delgado DR, Rodríguez GA, Martínez F. Thermodynamic study of the solubility of sulfapyridine in some ethanol + water mixtures. J Mol Liq. 2013;177:156–161.
   Web of Science ®Google Scholar
• Jouyban A. Review of the cosolvency models for predicting solubility of drugs in water-cosolvent mixtures. J Pharm Pharm Sci. 2008;11:32−58.
   PubMed Web of Science ®Google Scholar
• Jouyban-Gharamaleki A, Valaee L, Barzegar-Jalali M, et al. Comparison of various cosolvency models for calculating solute solubility in water–cosolvent mixtures. Int J Pharm. 1999;177:93–101.
   PubMed Web of Science ®Google Scholar
• Ruidiaz MA, Rodríguez SJ, Neita PC, et al. Performance of the Jouyban-Acree model for correlating the solubility of indomethacin and ethylhexyl triazone in ethyl acetate+ ethanol mixtures. Vitae. 2010;17:309–316.
   Web of Science ®Google Scholar
• Patel SV, Patel S. Prediction of the solubility in lipidic solvent mixture: investigation of the modeling approach and thermodynamic analysis of solubility. Eur J Pharm Sci. 2015;77:161–169.
   PubMed Web of Science ®Google Scholar
• Jouyban A, Fakhree MAA. Chapter 9: Experimental and computational methods pertaining to drug solubility. In: Acree WE Jr, editor. Toxicity and drug testing. New York (NY): Intech Co; 2012.
   Google Scholar
• Wei T, Wang C, Du S, et al. Measurement and correlation of the solubility of penicillin V potassium in ethanol+ water and 1-butyl alcohol+ water systems. J Chem Eng Data. 2015;60:112–117.
   Web of Science ®Google Scholar
• Vahdati S, Shayanfar A, Hanaee J, et al. Solubility of carvedilol in ethanol + propylene glycol mixtures at various temperatures. Ind Eng Chem Res. 2013;52:16630–16636.
   Web of Science ®Google Scholar
• Jouyban-Gharamaleki A, Acree WE Jr. Comparison of models for describing multiple peaks in solubility profiles. Int J Pharm. 1998;167:177–182.
   Web of Science ®Google Scholar
• Jouyban A, Khoubnasabjafari M, Chan HK, et al. Mathematical representation of solubility of amino acids in binary aqueous-organic solvent mixtures at various temperatures using Jouyban-Acree model. Pharmazie. 2006;61:789–792.
   PubMed Web of Science ®Google Scholar
• Mota FL, Carneiro AP, Queimada AJ, et al. Temperature and solvent effects in the solubility of some pharmaceutical compounds: measurements and modeling. Eur J Pharm Sci. 2009;37:499–507.
   PubMed Web of Science ®Google Scholar
• Ali HSM, York P, Blagden N, et al. Solubility of budesonide, hydrocortisone, and prednisolone in ethanol+ water mixtures at 298.2 K. J Chem Eng Data. 2009;55:578–582.
   Web of Science ®Google Scholar
• Kishi H, Hashimoto Y. Evaluation of the procedures for the measurement of water solubility and n-octanol/water partition coefficient of chemicals results of a ring test in Japan. Chemosphere. 1989;18:1749–1759.
   Web of Science ®Google Scholar
• Sajedi-Amin S, Barzegar-Jalali M, Fathi-Azarbayjani A, et al. Solubilization of bosentan using ethanol as a pharmaceutical cosolvent. J Mol Liq. 2017;232:152–158.
   Web of Science ®Google Scholar
• Jouyban A. Handbook of solubility data for pharmaceuticals. Boca Raton (FL): CRC Press; 2010.
   Google Scholar