76
Views
2
CrossRef citations to date
0
Altmetric
Articles

Measurement and modelling of solubility data for bosentan in 1-propanol + water mixtures at various temperatures

, , , , ORCID Icon & ORCID Icon
Pages 640-649 | Received 04 Aug 2018, Accepted 06 Aug 2018, Published online: 30 Aug 2018

References

  • Krupa A, Majda D, Mozgawa W, et al. Physicochemical properties of Bosentan and selected PDE-5 inhibitors in the design of drugs for rare diseases. Aaps Pharmscitech. 2017;18:1318–1331.
  • Abraham S, Steen V. Optimal management of digital ulcers in systemic sclerosis. Ther Clin Risk Manag. 2015;11:939–947.
  • Azim MS, Husain A, Mitra M, et al. Pharmacological and pharmaceutical profile of Bosentan: a review. Am J Pharm Tech Res. 2012;4:135–147.
  • Jouyban A. Handbook of solubility data for pharmaceuticals. Boca Raton (FL): CRC Press; 2010.
  • Khoubnasabjafari M, Shayanfar A, Martinez F, et al. Generally trained models to predict solubility of drugs in carbitol + water mixtures at various temperatures. J Mol Liq. 2016;219:435–438.
  • Khan AD, Singh L. Various techniques of bioavailibility enhancement: a review. J Drug Deliv Ther. 2016;6:34–41.
  • Jouyban A, Majidi MR, Jalilzadeh H, et al. Modeling drug solubility in water–cosolvent mixtures using an artificial neural network. Farmaco. 2004;59:505–512.
  • Bai TC, Yan GB, Zhang HL, et al. Solubility of silybin in aqueous dextran solutions. J Chem Eng Data. 2005;50:1596–1601.
  • Rubino JT, Swarbrick J, Boylan J. Encyclopedia of pharmaceutical technology. Dekker Inc. 1988;3:375–398.
  • Sajedi-Amin S, Barzegar-Jalali M, Fathi-Azarbayjani A, et al. Solubilization of bosentan using ethanol as a pharmaceutical cosolvent. J Mol Liq. 2017;232:152–158.
  • Babaei M, Shayanfar A, Rahimpour E, et al. Phys Chem Liq. 2018. DOI:10.1080/00319104.2018.14618721-11.
  • Barzegar-Jalali M, Mirheydari SN, Rahimpour E, Shekaari H, Martinezi F, Jouyban A. Experimental determination and correlation of bosentan solubility in (PEG 200 + water) mixtures at T= (293.15–313.15) K. Phys Chem Liq. 2018. DOI:https://doi.org/10.1080/00319104.2018.1491574
  • Barzegar-Jalali M, Mirheydari SN, Shekaari H, Martinezi F, Jouyban A. The solubility of bosentan in aqueous-2-propanol mixtures at several temperatures, measurement and data correlation. Phys Chem Liq. 2018. DOI: https://doi.org/10.1080/00319104.2018.1499911.
  • Barzegar-Jalali M, Jouyban-Gharamaleki A. Models for calculating solubility in binary solvent systems. Int J Pharm. 1996;140:237–246.
  • Delgado DR, Martínez F. Solubility and solution thermodynamics of sulfamerazine and sulfamethazine in some ethanol + water mixtures. Fluid Phase Equilib. 2013;360:88–96.
  • Wang S, Qin L, Zhou Z, et al. Solubility and solution thermodynamics of betaine in different pure solvents and binary mixtures. J Chem Eng Data. 2012;57:2128–2135.
  • Maher A, Croker D, Åc R, et al. Solubility of form III piracetam in a range of solvents. J Chem Eng Data. 2010;55:5314–5318.
  • Ruidiaz MA, Delgado DR, Martínez F, et al. Solubility and preferential solvation of indomethacin in 1,4-dioxane + water solvent mixtures. Fluid Phase Equilib. 2010;299:259–265.
  • Aragón DM, Rosas JE, Martínez F. Thermodynamic study of the solubility of ibuprofen in acetone and dichloromethane. Braz J Pharm Sci. 2010;46:227–235.
  • Panahi-Azar V, Ahmadian S, Martínez F, et al. Thermodynamic studies of fluphenazine decanoate solubility in PEG 200 + water mixtures. Fluid Phase Equilib. 2012;330:36–43.
  • Jouyban A, Acree JWE. Prediction of drug solubility in ethanol-ethyl acetate mixtures at various temperatures using the Jouyban-Acree model. J Drug Deliv Sci Tech. 2007;17:159–160.
  • Delgado DR, Rodríguez GA, Martínez F. Thermodynamic study of the solubility of sulfapyridine in some ethanol + water mixtures. J Mol Liq. 2013;177:156–161.
  • Jouyban A, Khoubnasabjafari M, Chan HK, et al. Mathematical representation of solubility of amino acids in binary aqueous-organic solvent mixtures at various temperatures using the Jouyban-Acree model. Pharmazie. 2006;61:789–792.
  • Fathi-Azarbayjani A, Abbasi M, Vaez-Gharamaleki J, et al. Measurement and correlation of deferiprone solubility: investigation of solubility parameter and application of van’t Hoff equation and Jouyban–acree model. J Mol Liq. 2016;215:339–344.
  • Jouyban-Gharamaleki A. The modified Wilson model and predicting drug solubility in water-cosolvent mixtures. Chem Pharm Bull. 1998;46:1058–1061.
  • Yalkowsky SH, Roseman TJ. Solubilization of drugs by Co-Solvents. In: Yalkowsky SH, editor. Techniques of solubilization of drugs. Vol. 12. New York (NY): Marcel Dekker Inc; 1981. p. 91–134.
  • Delgado DR, Martínez F. Solubility and solution thermodynamics of some sulfonamides in 1-propanol + water mixtures. J Solution Chem. 2014;43:836–852.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.