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Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 36, 2006 - Issue 18
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Original Articles

Synthesis of Tadalafil Analogues

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Pages 2627-2632 | Published online: 16 Feb 2007

References

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  • Daugan , A. , Grondin , P. , Ruault , C. , Coste , H. A. C. L. M. G. , Linget , J. M. , Kirilovsky , J. , Hyafil , F. and Labaudiniere , R. 2003 . The discovery of tadalafil: A novel and highly selective PDE5 inhibitor, 2: 2,3,6,7,12,12a‐Hexahydropyrazino[1,2:1,6]pyrido[3, 4‐b]indole‐1,4‐dione analogues . J. Med. Chem. , 46 : 4533 – 4542 .

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