One‐Step Synthesis of 2‐Aminothiazoline Derivatives Free of Lachrymatory Intermediates

References

• von Waltner , R. 1907 . Zur Kenntnis der Einwirkung von Bromacetophenon auf Thioharnstoffe . J. Prakt. Chemie , 75 : 187 – 189 .
   Google Scholar
• Hann , R. M. and Reid , E. E. 1933 . Isomeric 2‐iminotolyl‐3‐tolyl‐4‐p‐chloro and p‐bromophemyl‐Δ4‐thiazolines . J. Am. Chem. Soc. , 55 : 4998 – 5000 .
   Google Scholar
• Wilson , W. and Woodger , R. 1955 . 4′,5′‐Dihydroglyoxalino(2′,1′‐2, 3)thiazolium salts, and the ultraviolet light absorbtion of thiazole derivatives . J. Chem. Soc. , : 2943 – 2947 .
   Google Scholar
• Ivanov , Y. Y. , Tkachenko , S. E. , Proshin , A. N. and Bachurin , S. O. 2003 . 2‐Amino‐2‐thiazoline derivatives—a novel chemotype possessing muscarinomimetic effect . Biomed. Khim. , 49 ( 1 ) : 92 – 95 .
   Google Scholar
• Baumann , R. J. , Mayer , G. D. , Fite , L. D. , Gill , L. M. and Harrison , B. L. 1991 . In vitro and in vivo candicidal activities of 2‐(p‐n‐hexylphenylamino)‐1,3‐thiazoline . Chemotherapy , 37 ( 3 ) : 157 – 165 .
   Google Scholar
• Bonde , C. G. and Gaikwad , N. J. 2004 . Synthesis and preliminary evaluation of some pyrazine containing thiazolines and thiazolidinones as antimicrobial agents . Bioorg. Med. Chem. , 12 ( 9 ) : 2151 – 2161 .
   PubMed Web of Science ®Google Scholar
• Becker , H. G. O. , Domschke , G. , Fanghaenel , E. , Fischer , M. , Gewald , K. , Mayer , R. , Pavel , D. , Schmidt , K. , Berger , W. , Faust , J. , Gentz , F. , Gluch , R. , Mueler , K. , Schollberg , K. , Seiler , E. and Zeppenfeld , G. 1990 . Organikum, Organisch‐chemisches Grundpraktikum , 18th Ed. 521 Berlin : Deutscher Verlag der Wissenschaften .
   Google Scholar
• Kosolapoff , G. M. 1953 . Direct halogenation of some aromatic amines . J. Am. Chem. Soc. , 75 : 3596 – 3597 .
   Web of Science ®Google Scholar