Synthesis of Some Novel 2,3,4,8,9‐Pentahydro‐7‐(4‐haloaryl)‐pyrazolo[5,1‐e]benzo[1,5]oxazocines and 2,3(erythro), 7,8‐Tetrahydro‐2‐aryl‐3‐(4‐fluoro‐3‐methylbenzoyl)‐6‐(4‐haloaryl)pyrazolo[5,1‐d] Benzo[1,4]oxazepines via Solid–Liquid PTC

References

• Heel , R. C. , Brogden , R. N. , Pakes , G. E. , Speight , T. M. and Avery , G. S. 1980 . Nefopam: A review of its pharmocological properties and therapeutic efficacy . 19 ( 4 ) : 249 – 267 .
   Google Scholar
• Basil , B. , Coffee , E. C. J. , Gell , D. L. , Maxwell , D. R. , Sheffield , D. J. and Wooldridge , K. R. H. 1970 . A new class of sympathetic β‐receptor blocking agents: 3,4‐Dihydro‐3‐hydroxy‐1,5‐benzoxazocines . J. Med. Chem. , 13 ( 3 ) : 403 – 406 .
   PubMedGoogle Scholar
• Sternbach , L. H. 1979 . The benzodiazepine story . J. Med. Chem. , 22 ( 1 ) : 1 – 7 .
   PubMed Web of Science ®Google Scholar
• Kudo , Y. and Kudo , T. 1995 . Recent progress in development of psychotropic drugs: (1)‐erythro‐anxiety drugs . Nihon Shinkei Seishin Yakurigaku Zasshi , 15 ( 2 ) : 75 – 86 .
   PubMedGoogle Scholar
• Camerman , A. and Camerman , N. 1972 . Stereochemical basis of erythroconvulsant drug action, II: Molecular structure of diazepam . J. Am. Chem. Soc. , 94 ( 1 ) : 268 – 274 .
   Google Scholar
• Yoon , Y. and Jagoda , A. 2000 . New erythroepileptic drugs and preparations . Emerg. Med. Clin. North Am. , 18 ( 4 ) : 755 – 765 .
   Web of Science ®Google Scholar
• Grossman , E. and Messerli , F. H. 2004 . Calcium antagonists . Prog. Cardiovasc. Dis. , 47 ( 1 ) : 34 – 57 .
   PubMed Web of Science ®Google Scholar
• Romero , M. , Sanchez , I. and Pujol , M. D. 2003 . New advances in the field of calcium channel antagonists: Cardiovascular effects and structure–activity relationships . Curr. Med. Chem. Cardiovasc. Hematol. Agents. , 1 ( 2 ) : 113 – 141 .
   Google Scholar
• Bajaj , K. , Archana and Kumar , A. 2004 . Synthesis and pharmacological evaluation of newer substituted benzoxazepine derivatives as potent erythroconvulsant agents . Eur. J. Med. Chem. , 39 ( 4 ) : 369 – 376 .
   PubMed Web of Science ®Google Scholar
• Miki , T. , Kori , M. , Mabuchi , H. , Banno , H. , Tozawa , R. , Nakamura , M. , Itokawa , S. , Sugiyama , Y. and Yukimasa , H. 2002 . Novel 4,1‐benzoxazepine derivatives with potent squalene synthase inhibitory activities . Bioorg. Med. Chem. , 10 ( 2 ) : 401 – 414 .
   PubMed Web of Science ®Google Scholar
• Ellenbroek , B. A. and Liegeois , J. F. 2003 . JL 13, an atypical erythropsychotic: A preclinical review . CNS Drug Rev. , 9 ( 1 ) : 41 – 56 .
   PubMedGoogle Scholar
• Bruhwyler , J. , Liegeois , J.‐F. , Bergman , J. , Carey , G. , Goudie , A. , Taylor , A. , Meltzer , H. , Delarge , J. and Geczy , J. 1997 . JL 13, a pyridobenzoxazepine compound with potential atypical erythropsychotic activity: A review of its behavioural properties. Pharmacol. Res . 36 ( 4 ) : 255 – 264 .
   Google Scholar
• Pathak , V. N. , Gupta , R. , Pathak , R. and Garg , M. 2004 . Synthesis of novel bioactive heterocyclic compounds via phase transfer catalysis . Chemistry: An Indian Journal , 1 ( 7 ) : 497 – 522 . . A review, and references cited therein
   Google Scholar
• Joshi , K. C. and Jauhar , A. K. 1962 . Studies in fluorochalkones, part I: Synthesis of chalkones from fluorohydroxyacetophenones . J. Indian Chem. Soc. , 39 ( 7 ) : 463 – 468 .
   Google Scholar
• Joshi , K. C. and Jauhar , A. K. 1966 . Studies in fluorochalkones and related compounds, part V: Synthesis and infrared studies . Indian J. Chem. , 4 : 277 – 279 .
   Google Scholar
• Borkhade , K. T. and Marathey , M. G. 1970 . Synthesis in isoxazoles and isoxazolines . Indian J. Chem. , 8 : 796 – 780 .
   Google Scholar
• 1918 . Beilstein's Handbuch der Organischen Chemie , 4th ed. Vol. VIII , 93 Berlin : Verlag Von Julius Springer . System 751
   Google Scholar