References
- Villhauer , E. B. , Brinkman , J. A. , Naderi , G. B. , Burkey , B. F. , Dunning , B. E. , Prasas , K. , Mangold , B. L. , Russel , M. E. and Hughes , T. E. 2003 . 1‐[3‐Hydroxy‐1‐adamantyl)amino]acetyl]‐2‐cyano‐(S)‐pyrrolidine: A potent, selective and orally bioavailable dipetidyl peptidase IV inhibitor with antihyperglycemic properties . J. Med. Chem. , 46 : 2774 – 2789 .
- Augustyns , K. , Van der Veken , P. , Senten , K. and Haemers , A. 2003 . Dipeptidyl peptidase IV inhibitors as new therapeutic agents in the treatment of type II diabetes . Expert Opin. Ther. Pat. , 13 ( 4 ) : 499 – 510 .
- Drucker , D. J. 2003 . Therapeutic potential of dipeptidyl peptidase IV inhibitors for the treatment of type II diabetes . Expert Opin. Invest. Drugs. , 12 : 87 – 100 .
- Senten , K. , Van der Veken , P. , De Meester , I. , Lambeir , A. M. , Scharpe , S. , Haemers , A. and Augustyns , K. 2003 . Design, synthesis, and SAR of potent and selective dipeptide‐derived inhibitors for dipeptidyl peptidases . J. Med. Chem. , 46 : 5005 – 5014 .
- Senten , K. , Van der Veken , P. , De Meester , I. , Lambeir , A. M. , Scharpe , S. , Haemers , A. and Augustyns , K. 2004 . γ‐Amino‐substituted analogues of 1‐[(S)‐2,4‐diaminobutanoyl]piperidine as highly potent and selective dipeptidyl peptidase II inhibitors . J. Med. Chem. , 47 : 2906 – 2916 .
- Scharpe , S. , Gustyns , K. , Haemers , A. , Lambeir , A. M. , Demeester , I. , Senten , K. and Van Der Veken , P. Inhibitors of proline‐specific dipeptidyl peptidases: DPP IV inhibitors as a novel approach for the treatment of type 2 diabetes . WO2004076434 . 10/09/2004 .
- Radhakrishna , A. S. , Parham , M. E. , Riggs , R. M. and Loudon , G. M. 1979 . New method for direct conversion of amides to amines . J. Org. Chem. , 44 : 1746
- Waki , M. , Kitajima , Y. and Izumiya , N. 1981 . A facile synthesis of N 2‐protected L‐2,3‐diaminopropanoic acid . Synthesis , 4 : 266
- Merrick , R. , Almond , J. B. , Stimmel , E. , Thompson , A. and Loudon , G. M. 1993 . Hofmann rearrangement under mildly acidic conditions using [1,1‐bis(trifluoroacetoxy)]iodobenzene . Org. Synth. Coll. , 8 : 132