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Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 38, 2008 - Issue 5
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Original Articles

Practical Methylation Procedure for (1H)‐1,2,4‐Triazole

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Pages 738-745 | Received 14 Sep 2007, Published online: 15 Feb 2008

References

  • Paquette , L. A. 1968 . Principles of Modern Heterocyclic Chemistry New York : W. A. Benjamin . Heterocyclic chemistry encompasses a vast area of knowledge. For a general overview and introduction to the discipline, the following books are useful
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  • Montgomery , J. A. 1981 . The Chemistry of Heterocyclic Compounds Edited by: Montgomery , J. A. Vol. 37 , New York : John Wiley & Sons . The chemistry and practical applications of triazoles are well‐developed. For several highly selected examples, among many publications, see Temple, C. 1,2,4‐Triazoles
  • Turnbull , K. 1998 . Five‐membered ring systems with more than one N Atom . Prog. Heterocycl. Chem. , 10 : 153 – 171 .
  • Garratt , P. J. 1996 . “ 1,2,4‐Triazoles ” . In Comprehensive Heteroaromatic Chemistry II Edited by: Katritzky , A. R. , Rees , C. W. and and Scriven , E. F. V. Vol. 4 , 127 – 163 . Oxford : Pergamon Press . 905–1006
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  • Heeres , J. , Hendrickx , R. and Van Cutsem , J. 1983 . Antimycotic azoles, 6: synthesis and antifungal properties of terconazole, a novel triazole ketal . J. Med. Chem. , 26 : 611 – 613 .
  • Atkinson , M. R. and Polya , J. B. 1954 . Triazoles, part II: N‐Substitution of some 1,2,4‐triazoles . J. Chem. Soc. , : 141 – 145 .
  • Mirzael , Y. R. , Twamley , B. and Shreeve , J. M. 2002 . Syntheses of 1‐alkyl‐1,2,4‐triazoles and the formation of quaternary 1‐alkyl‐4‐polyfluoralk‐1,2,4‐triazolium salts leading to ionic liquids . J. Org. Chem. , 67 : 9340 – 9345 .
  • Bulger , P. G. , Cottrell , I. F. , Cowdon , C. J. , Davies , A. J. and Dolling , U.‐H. 2000 . An investigation into the alkylation of 1,2,4‐triazole . Tetrahedron Lett. , 41 : 1297 – 1301 .
  • Astleford , B. A. , Goe , G. L. , Keay , J. G. and Scriven , E. F. V. 1989 . Synthesis of 1‐alkyl 1,2,4‐triazoles: a new one‐pot regiospecific procedure . J. Org. Chem. , 54 : 731 – 732 .

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