Publication Cover
Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 38, 2008 - Issue 16
286
Views
6
CrossRef citations to date
0
Altmetric
Original Articles

Synthesis of Ethyl Nicotinate-5-Boronic Acid Pinacol Ester and Its Application Toward Suzuki Coupling

&
Pages 2775-2781 | Received 31 Jul 2008, Accepted 18 Oct 2007, Published online: 25 Aug 2010

REFERENCES

  • Carlson , L. A. J. Nicotinic acid: the broad-spectrum lipid drug . Int. Med. , 2005 , 258 , 94 – 114 .
  • Mrochek , J. E. ; Jolley , R. L. ; Young , D. S. ; Turner , W. Metabolic response of humans to ingestion of nicotinic acid and nicotinate . J. Chem. 1976 , 22 , 1821 – 1827 .
  • Hallé , J.-C. ; Lelievre , J. ; Terrier , F. Solvent effect on preferred protonation sites in nicotinate and isonicotinate anions . J. Chem. 1996 , 74 , 613 – 620 .
  • Arnold , W. D. ; Gosberg , A. ; Li , Z. ; Steensma , R. W. ; Wilson , M. E. Fused ring heterocycle kinase modulators . WO 2006015124 , 2006 .
  • Miyaura , N. ; Suzuki , A. Palladium-catalized cross-coupling reactions of organoboron compounds . Chem. Rev. 1995 , 95 , 2457 – 2483 .
  • Ishiyama , T. ; Ishida , K. ; Miyaura , N. Synthesis of pinacol arylboronates via the cross-coupling reaction of bis(pinacolato)diboron with chloroarenes catalyzed by palladium (0)-tricyclohexylphosphine complexes . Tetrahedron 2001 , 57 , 9813 – 9816 .
  • Kudo , N. ; Perseghini , M. ; Fu , G. C. A versatile method for Suzuki cross-coupling reactions of nitrogen heterocycles . Angew. Chem. Int. Ed 2006 , 45 , 1282 – 1284 .
  • Roy , P. ; Boisvert , M. ; Leblanc , Y. Preparation of substituted 5-azaindoles: Methyl 4-chloro-1H-pyrrolo[3,2-c]pyridine-2-carboxylate . Org. Synth. 2007 , 24 , 262 – 271 .
  • Cusack , K. ; Salmeron-Garcia , J.-A. ; Gordon , T. D. ; Barberis , C. E. ; Allen , H. J. ; Bischoff , A. K. ; Ericson , A. M. ; Friedman , M. M. ; George , D. M. ; Roth , G. P. ; Talanian , R. V. ; Thomas , C. ; Wallace , G. A. ; Wishart , N. ; Yu , Z. Kinase inhibitors as therapeutic agents . WO2005110410 , 2005 .

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.